MedPath

Study Comparing Combination of LGX818 Plus MEK162 Versus Vemurafenib and LGX818 Monotherapy in BRAF Mutant Melanoma

Phase 3
Completed
Conditions
Melanoma
Interventions
Registration Number
NCT01909453
Lead Sponsor
Pfizer
Brief Summary

This is 2-part, randomized, open label, multi-center, parallel group, phase III study comparing the efficacy and safety of LGX818 plus MEK162 to vemurafenib and LGX818 monotherapy in patients with locally advanced unresectable or metastatic melanoma with BRAF V600 mutation. A total of approximately 900 patients will be randomized.

Part 1:

Patients will be randomized in a 1:1:1 ratio to one of 3 treatment arms:

1. LGX818 450 mg QD plus MEK162 45 mg BID (denoted as Combo 450 arm)

2. LGX818 300 mg QD monotherapy (denoted as LGX818 arm) or

3. vemurafenib 960 mg BID (denoted as vemurafenib arm)

Part 2:

Patients will be randomized in a 3:1 ratio to one of the 2 treatment arms:

1. LGX818 300 mg QD plus MEK162 45 mg BID (denoted as Combo 300 arm) or

2. LGX818 300 mg QD monotherapy (denoted as LGX818 arm)

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
922
Inclusion Criteria
  • Diagnosis of locally advanced, unresectable or metastatic cutaneous melanoma or unknown primary melanoma (AJCC Stage IIIB, IIIC, or IV)
  • Presence of BRAF V600E or V600K mutation in tumor tissue prior to randomization
  • Naïve untreated patients or patients who have progressed on or after prior first line immunotherapy for resectable locally advanced or metastatic melanoma; prior adjuvant therapy is permitted (e.g. IFN, IL-2 therapy, any other immunotherapy, radiotherapy or chemotherapy), except the administration of BRAF or MEK inhibitors
  • Evidence of at least one measurable lesion as detected by radiological or photographic methods
  • ECOG performance status of 0 or 1
  • Adequate bone marrow, organ function, cardiac and laboratory parameters
  • Normal functioning of daily living activities
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Exclusion Criteria
  • Any untreated central nervous system (CNS) lesion
  • Uveal and mucosal melanoma
  • History of leptomeningeal metastases
  • History of or current evidence of central serous retinopathy (CSR), retinal vein occlusion (RVO) or history of retinal degenerative disease
  • Any previous systemic chemotherapy treatment, extensive radiotherapy or investigational agent other than immunotherapy, or patients who have received more than one line of immunotherapy for locally advanced unresectable or metastatic melanoma; Ipilimumab (adjuvant) or other immunotherapy treatment must have ended at least 6 weeks prior to randomization
  • History of Gilbert's syndrome
  • Prior therapy with a BRAF inhibitor and/or a MEK- inhibitor
  • Impaired cardiovascular function or clinically significant cardiovascular diseases
  • Uncontrolled arterial hypertension despite medical treatment
  • HIV positive or active Hepatitis B, and/or active Hepatitis C
  • Impairment of gastrointestinal function
  • Patients with neuromuscular disorders that are associated with elevated CK
  • Pregnant or nursing (lactating) women
  • Medical, psychiatric, cognitive or other conditions that may compromise the patient's ability to understand the patient information, give informed consent, comply with the study protocol or complete the study

Other protocol-defined inclusion/exclusion criteria may apply

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Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
LGX818 300 mg + MEK162LGX818LGX818 300 mg QD + MEK162 45 mg BID
LGX818 300 mg + MEK162MEK162LGX818 300 mg QD + MEK162 45 mg BID
LGX818 450 mg + MEK162LGX818LGX818 450 mg QD + MEK162 45 mg BID
LGX818 450 mg + MEK162MEK162LGX818 450 mg QD + MEK162 45 mg BID
LGX818LGX818LGX818 300 mg QD
VemurafenibvemurafenibVemurafenib 960 mg BID
Primary Outcome Measures
NameTimeMethod
Part 1: Progression Free Survival (PFS) by Blinded Independent Review Committee (BIRC) in Combo 450 Group as Compared to Vemurafenib GroupFrom randomization until documented disease progression (PD), initiation of new anti-cancer therapy, censoring date or death, whichever occurred first (up to 29 months)

PFS was defined as the time from the date of randomization to the date of the first documented disease progression (PD) or death due to any cause, whichever occurs first. PFS was determined based on tumor assessment (RECIST version 1.1 criteria) as per BIRC/central review and survival information. If a participant did not had an event at the time of the analysis cut-off or at the start of any new anti-cancer therapy, data was censored at the date of last adequate tumor assessment. PD was defined as at least a 20% increase in the sum of diameter of all measured target lesions, taking as reference the smallest sum of diameter of all target lesions recorded at or after baseline. In addition to the relative increase of 20%, the sum must demonstrate an absolute increase of at least 5 square millimeter (mm\^2).

Part 1: Progression Free Survival (PFS) by Blinded Independent Review Committee (BIRC) in Combo 450 Group as Compared to LGX818 GroupFrom randomization until documented disease progression (PD), initiation of new anti-cancer therapy, censoring date or death, whichever occurred first (up to 29 months), excluding Part 1: LGX818 300 mg group; up to 35 months for Part 1: LGX 300 mg group

PFS was defined as the time from the date of randomization to the date of the first documented disease progression (PD) or death due to any cause, whichever occurs first. PFS was determined based on tumor assessment (RECIST version 1.1 criteria) as per BIRC and survival information. If a participant did not had an event at the time of the analysis cut-off or at the start of any new anti-cancer therapy, data was censored at the date of last adequate tumor assessment. PD was defined as at least a 20% increase in the sum of diameter of all measured target lesions, taking as reference the smallest sum of diameter of all target lesions recorded at or after baseline. In addition to the relative increase of 20%, the sum must demonstrate an absolute increase of at least 5 mm\^2.

Secondary Outcome Measures
NameTimeMethod
Part 1: Number of Participants With Worst Post-baseline Left Ventricular Dysfunction Events (LVEF) Values by Multigated Acquisition (MUGA) Scans or Transthoracic Echocardiograms (ECHO), by CTCAE GradeBaseline up to 30 days from last dose of study drug (up to 30 months), excluding Part 1: LGX818 300 mg group; up to 36 months for Part 1 LGX 300 mg group

Participants with worst post-baseline LVEF Values were graded as Grade 0: Non missing value below Grade 2; Grade 2: LVEF between 40% and 50% or absolute reduction from baseline \>=10% and \< 20%; Grade 3: LVEF between 20% and 39% or absolute reduction from baseline \>=20%; Grade 4: LVEF lower than 20%. Baseline was defined as the last non-missing value prior to the first dose of study treatment. Missing data were due to participants who died or withdrew consent prior to the first scheduled evaluation or missed evaluations as protocol deviations.

Part 1: Number of Participants With Ocular-related Adverse Events of Special Interest (AESI) Graded According to the National Cancer Institute Common Terminology Criteria (NCI-CTCAE) v4.03Baseline up to 30 days from last dose of study drug (up to 30 months), excluding Part 1: LGX818 300 mg group; up to 36 months for Part 1 LGX 300 mg group

AESI consisted of events for which there was a specific clinical interest with regard to LGX818 and/or MEK162 treatment. Ocular-related AESI included retinopathy excluding retinal vein occlusion (RVO), RVO and uveitis-type events. As per NCI-CTCAE version 4.03, severity was graded as Grade 1: asymptomatic/mild symptoms, clinical/diagnostic observations only, intervention not indicated; Grade 2: moderate, minimal, local/noninvasive intervention indicated, limiting age-appropriate instrumental ADL; Grade 3: severe/medically significant but not immediately life-threatening, hospitalization/prolongation of existing hospitalization indicated, disabling, limiting self-care ADL; Grade 4: life-threatening consequence, urgent intervention indicated; Grade 5: death related to AE. AEs of grade 3 or 4 are reported in this outcome measure.

Part 2: Number of Participants With Newly Occurring Notably Abnormal Vital SignsBaseline up to 30 days after last dose of study drug (up to 36 months)

Notably abnormal vital signs were: Low/high systolic blood pressure (SBP) in millimeter of mercury (mmHg): less than or equal to (\<=) 90 mmHg with decrease from baseline of greater than or equal to (\>=) 20 mmHg/\>= 160 mmHg with increase from baseline of \>=20 mmHg, Low/high diastolic blood pressure (DBP) \[mmHg\]: \<=50 mmHg with decrease from baseline of \>=15 mmHg/\>=100 mmHg with increase from baseline of \>=15 mmHg, Low/high pulse rate \[bpm\]: \<=50 bpm with decrease from baseline of \>=15 bpm/\>=120 bpm with increase from baseline of \>=15 bpm, Low/high weight (kg): \>=20 % decrease from baseline/\>= 10% increase from baseline Low/high Body temperature degree C): \<= 36°C/\>= 37.5 degree C.

Part 1: Percentage of Participants With Adverse Events (AEs) and Serious Adverse Events (SAEs) as Graded by National Cancer Institute Common Terminology Criteria (NCI-CTCAE), Version 4.03Baseline up to 30 days from last dose of study drug (up to 30 months), excluding Part 1: LGX818 300 mg group; up to 36 months for Part 1 LGX 300 mg group

AE was any untoward medical occurrence in a participant who received study drug without regard to possibility of causal relationship. SAE was any untoward medical occurrence at any dose that results in death; is life-threatening; requires inpatient hospitalization/prolongation of existing hospitalization; results in persistent/significant disability/incapacity; results in congenital anomaly/birth defect or that is considered to be important medical event. As per NCI-CTCAE version 4.03, severity was graded as Grade 1: asymptomatic/mild symptoms, clinical/diagnostic observations only; Grade 2: moderate, minimal, local/noninvasive intervention indicated, limiting age-appropriate instrumental activities of daily life (ADL); Grade 3: severe/medically significant but not immediately life-threatening, hospitalization/prolongation of existing hospitalization indicated, disabling, limiting self-care ADL; Grade 4: life-threatening consequence; Grade 5: death. AEs of all grades were reported.

Part 1: Number of Participants With Newly Occurring Notably Abnormal Vital SignsBaseline up to 30 days from last dose of study drug (up to 30 months), excluding Part 1: LGX818 300 mg group; up to 36 months for Part 1 LGX 300 mg group

Notably abnormal vital signs were: Low/high systolic blood pressure (SBP) (millimeter of mercury \[mmHg\]): less than or equal to (\<=) 90 mmHg with decrease from baseline of greater than or equal to (\>=) 20 mmHg/\>= 160 mmHg with increase from baseline of \>=20 mmHg. Low/high diastolic blood pressure (DBP) \[mmHg\]: \<= 50 mmHg with decrease from baseline of \>=15 mmHg/\>=100 mmHg with increase from baseline of \>=15 mmHg. Low/high Pulse rate: \<=50 beats per minute (bpm) with decrease from baseline of \>=15 bpm/\>= 120 bpm with increase from baseline of \>=15 bpm. Low/high Weight \[kilogram\]: \>=20 percent (%) decrease from baseline/\>= 10% increase from baseline. Low/high Body temperature degree Celsius (C): \<= 36 degree C/\>= 37.5 degree C.

Part 1: Overall Survival (OS)From randomization until documented disease progression (PD), initiation of new anti-cancer therapy, censoring date or death, whichever occurred first (up to 38 months)

Overall survival was defined as the time from the date of randomization to the date of death due to any cause. If a death had not been observed by the date of analysis cutoff, OS was censored at the date of last contact.

Part 1: Number of Participants With Clinically Notable Shift From Baseline in Laboratory Parameter Values Based on National Cancer Institute Common Terminology Criteria (NCI-CTCAE) Grade, Version 4.03Baseline up to 30 days from last dose of study drug (up to 30 months), excluding Part 1: LGX818 300 mg group; up to 36 months for Part 1 LGX 300 mg group

Number of participants with clinically notable shift from baseline in laboratory parameter values based on national cancer institute common terminology criteria (NCI-CTCAE) grade, Version 4.03 were graded from Grades 1 to 5. Grade 1: Mild; asymptomatic or mild symptoms; clinical or diagnostic observations only; intervention not indicated. Grade 2: Moderate; minimal, local or noninvasive intervention indicated. Grade 3: Severe or medically significant but not immediately life-threatening; hospitalization or prolongation of hospitalization indicated. Grade 4: Life-threatening consequences; urgent intervention indicated. Grade 5: Death. Clinically notable shift from baseline in laboratory parameter = worsening by at least 2 grades or to \>=grade 3.

Part 1: Number of Participants With Dermatologic-related Adverse Events of Special Interest (AESI) Graded According to the National Cancer Institute Common Terminology Criteria (NCI-CTCAE) v4.03Baseline up to 30 days from last dose of study drug (up to 30 months), excluding Part 1: LGX818 300 mg group; up to 36 months for Part 1 LGX 300 mg group

AESI consisted of events for which there was a specific clinical interest with regard to LGX818 and/or MEK162 treatment. Dermatologic-related AESI included rash, photosensitivity, nail disorders, skin infections, severe cutaneous adverse reactions and Palmar-plantar erythrodysaesthesia (PPE) syndrome. As per NCI-CTCAE version 4.03, severity was graded as Grade 1: asymptomatic/mild symptoms, clinical/diagnostic observations only, intervention not indicated; Grade 2: moderate, minimal, local/noninvasive intervention indicated, limiting age-appropriate instrumental ADL; Grade 3: severe/medically significant but not immediately life-threatening, hospitalization/prolongation of existing hospitalization indicated, disabling, limiting self-care ADL; Grade 4: life-threatening consequence, urgent intervention indicated; Grade 5: death related to AE. AEs of grade 3 or 4 are reported in this outcome measure.

Part 2: Progression Free Survival (PFS) by BIRC in Combo 300 Group as Compared to LGX818 GroupFrom randomization until documented disease progression (PD), initiation of new anti-cancer therapy, censoring date or death, whichever occurred first (up to 35 months)

PFS was defined as the time from the date of randomization to the date of the first documented disease progression (PD) or death due to any cause, whichever occurs first. PFS was determined based on tumor assessment (RECIST version 1.1 criteria) as per BIRC and survival information. If a participant did not had an event at the time of the analysis cut-off or at the start of any new anti-cancer therapy, data was censored at the date of last adequate tumor assessment. PD was defined as at least a 20% increase in the sum of diameter of all measured target lesions, taking as reference the smallest sum of diameter of all target lesions recorded at or after baseline. In addition to the relative increase of 20%, the sum must demonstrate an absolute increase of at least 5 mm\^2.

Part 1: Number of Participants With Newly Occurring Notable Electrocardiogram (ECG) ValuesBaseline up to 30 days from last dose of study drug (up to 30 months), excluding Part 1: LGX818 300 mg group; up to 36 months for Part 1 LGX 300 mg group

Newly occurring notable ECG values were reported for QT (millisecond \[ms\]), QTcF (millisecond), QTcB (millisecond) and heart rate (beats per minute). Newly occurring was defined as participants not meeting criterion at baseline and meeting criterion post-baseline. Ranges for newly occurring notable ECG values (QT, QTcF, QTcB) are New greater than (\>) 450, New \>480, New \>500, Increase from baseline \>30, Increase from baseline \>60. Heart rate: New \<60, New \>100 was considered as newly occurring notable value.

Part 2: Percentage of Participants With Adverse Events (AEs) and Serious Adverse Events (SAEs) as Graded by National Cancer Institute Common Terminology Criteria (NCI-CTCAE), Version 4.03Baseline up to 30 days after last dose of study drug (up to 36 months)

AE was any untoward medical occurrence in a participant who received study drug without regard to possibility of causal relationship. SAE was any untoward medical occurrence at any dose that results in death; is life-threatening; requires inpatient hospitalization/prolongation of existing hospitalization; results in persistent/significant disability/incapacity; results in congenital anomaly/birth defect or that is considered to be important medical event. As per NCI-CTCAE version 4.03, severity was graded as Grade 1: asymptomatic/mild symptoms, clinical/diagnostic observations only; Grade 2: moderate, minimal, local/noninvasive intervention indicated, limiting age-appropriate instrumental activities of daily life (ADL); Grade 3: severe/medically significant but not immediately life-threatening, hospitalization/prolongation of existing hospitalization indicated, disabling, limiting self-care ADL; Grade 4: life-threatening consequence; Grade 5: death. AEs of all grades were reported.

Part 2: Number of Participants With Newly Occurring Notable ECG ValuesBaseline up to 30 days after last dose of study drug (up to 36 months)

Newly occurring notable ECG values were reported for QT (ms), QTcF (ms), QTcB (ms) and heart rate (bpm). Newly occurring was defined as participants not meeting criterion at baseline and meeting criterion post-baseline. Ranges for newly occurring notable ECG values (QT, QTcF, QTcB) are New \>450, New \>480, New \>500, increase from baseline \>30, Increase from baseline \>60. Heart rate: New \< 60, New \>100 was considered as newly occurring notable value.

Part 2: Number of Participants With Worst Post-baseline Left Ventricular Dysfunction Events (LVEF) Values by Multigated Acquisition (MUGA) Scans or Transthoracic Echocardiograms (ECHO), by CTCAE GradeBaseline up to 30 days after last dose of study drug (up to 36 months)

Participants with worst post-baseline LVEF Values were graded as Grade 0: Non missing value below Grade 2; Grade 2: LVEF between 40% and 50% or absolute reduction from baseline \>=10% and \< 20%;Grade 3: LVEF between 20% and 39% or absolute reduction from baseline \>=20%; Grade 4: LVEF lower than 20%. Baseline was defined as the last non-missing value prior to the first dose of study treatment. Missing data were due to participants who died or withdrew consent prior to the first scheduled evaluation or missed evaluations as protocol deviations.

Part 2: Number of Participants With Dermatologic-related Adverse Events of Special Interest (AESI) Graded According to the National Cancer Institute Common Terminology Criteria (NCI-CTCAE) v4.03Baseline up to 30 days after last dose of study drug (up to 36 months)

AESI consisted of events for which there was a specific clinical interest with regard to LGX818 and/or MEK162 treatment. Dermatologic-related AESI included rash, photosensitivity, nail disorders, skin infections, severe cutaneous adverse reactions and PPE syndrome. As per NCI-CTCAE version 4.03, severity was graded as Grade 1: asymptomatic/mild symptoms, clinical/diagnostic observations only, intervention not indicated; Grade 2: moderate, minimal, local/noninvasive intervention indicated, limiting age-appropriate instrumental ADL; Grade 3: severe/medically significant but not immediately life-threatening, hospitalization/prolongation of existing hospitalization indicated, disabling, limiting self-care ADL; Grade 4: life-threatening consequence, urgent intervention indicated; Grade 5: death related to AE. AEs of grade 3 or 4 are reported are reported in this outcome measure.

Part 2: Number of Participants With Clinically Notable Shift From Baseline in Laboratory Parameter Values Based on National Cancer Institute Common Terminology Criteria (NCI-CTCAE) Grade, Version 4.0Baseline up to 30 days after last dose of study drug (up to 36 months)

Number of participants with clinically notable shift from baseline in laboratory parameter values based on national cancer institute common terminology criteria (NCI-CTCAE) grade, Version 4.0 were graded from Grades 1 to 5. Grade 1: Mild; asymptomatic or mild symptoms; clinical or diagnostic observations only; intervention not indicated. Grade 2: Moderate; minimal, local or noninvasive intervention indicated. Grade 3: Severe or medically significant but not immediately life-threatening; hospitalization or prolongation of hospitalization indicated. Grade 4: Life-threatening consequences; urgent intervention indicated. Grade 5: Death. Clinically notable shift from baseline in laboratory parameter = worsening by at least 2 grades or to \>=grade 3.

Part 1 and Part 2: Objective Response Rate (ORR)From randomization until disease progression, censoring date or death, whichever occurred first (up to 29 months for Part 1, excluding Part 1: LGX818 300 mg group; up to 35 months for Part 2 and Part 1 LGX 300 mg group)

ORR, calculated as the percentage of participants with a best overall response of complete response (CR) or partial response (PR). CR was defined as disappearance of all non-nodal target lesions. In addition, any pathological lymph nodes assigned as target lesions must have a reduction in short axis to \< 10 mm. PR was defined as at least a 30% decrease in the sum of diameter of all target lesions, taking as reference the baseline sum of diameters. Results are reported for confirmed BIRC response.

Part 1 and Part 2: Time to Objective Response (TTR)From randomization until disease progression, censoring date or death, whichever occurred first (up to 29 months for Part 1, excluding Part 1: LGX818 300 mg group; up to 35 months for Part 2 and Part 1 LGX 300 mg group)

TTR was the time between date of randomization until first documented response of CR or PR. Participants who did not achieve a PR or CR were censored at the last adequate tumor assessment date when they did not have a PFS event or at maximum follow-up (i.e. first patient first visit \[FPFV\] to last patient last visit \[LPLV\] used for the analysis) when they had a PFS event. CR was defined as disappearance of all non-nodal target lesions. In addition, any pathological lymph nodes assigned as target lesions must have a reduction in short axis to \<10 mm. PR was defined as at least a 30% decrease in the sum of diameter of all target lesions, taking as reference the baseline sum of diameters. TTR was estimated in the treatment arms using a Kaplan-Meier method. TTR was based on central review.

Part 1 and Part 2: Change From Baseline in Global Health Status Score of EORTC QLQ-C30 at Day 1 of Cycle 3, 5, 7, 9, 11, 13, 15, 17, 19, 21, 23, 25 and End of Treatment VisitBaseline (Day 1 of Cycle 1), Day 1 of Cycle 3, 5, 7, 9, 11, 13, 15, 17, 19, 21, 23, 25 and end of treatment visit (within14 days after the last dose of study drug)

EORTC QLQ-C30 contains 30 items and is composed of multi-item and single-item measures. These include 5 functional scales (physical, role, emotional, cognitive and social functioning), 3 symptom scales (fatigue, nausea/vomiting, and pain), 6 single items (dyspnea, insomnia, appetite loss, constipation, diarrhea and financial impact) and a global health status/quality of life (QOL) scale. The questionnaire employs 28 4-point Likert scales with responses from "not at all" to "very much" and two 7-point Likert scales for global health and overall QOL. Responses to all items converted to 0 to 100 scale. For functional and global QOL scales, higher scores represent a better level of functioning/QOL. For symptom-oriented scales, a higher score represents more severe symptoms.

Part 1: Plasma Concentrations of MEK162Cycle 1 Day 1: pre-dose, 0.5, 1.5, 4 to 8, hours post dose; Cycle 2 Day 1: pre-dose; Cycle 3 Day 1: pre-dose
Part 2: Number of Participants With Ocular-related Adverse Events of Special Interest (AESI) Graded According to the National Cancer Institute Common Terminology Criteria (NCI-CTCAE) v4.03Baseline up to 30 days after last dose of study drug (up to 36 months)

AESI consisted of events for which there was a specific clinical interest with regard to LGX818 and/or MEK162 treatment. Ocular-related AESI included retinopathy excluding RVO, RVO and uveitis-type events. As per NCI-CTCAE version 4.03, severity was graded as Grade 1: asymptomatic/mild symptoms, clinical/diagnostic observations only, intervention not indicated; Grade 2: moderate, minimal, local/noninvasive intervention indicated, limiting age-appropriate instrumental ADL; Grade 3: severe/medically significant but not immediately life-threatening, hospitalization/prolongation of existing hospitalization indicated, disabling, limiting self-care ADL; Grade 4: life-threatening consequence, urgent intervention indicated; Grade 5: death related to AE. AEs of grade 3 or 4 are reported in this outcome measure.

Part 2: Overall Survival (OS)From randomization until documented disease progression (PD), initiation of new anti-cancer therapy, censoring date or death, whichever occurred first (up to 38 months)
Part 1 and Part 2: Number of Participants With Change From Baseline in Eastern Cooperative Oncology Group Performance Status (ECOG PS)Part 1 and Part 2: Baseline, Day 1 of each cycle (Cycle 2 to Cycle 31)

ECOG: participant's performance status was measured on a 6-point scale: 0= fully active/able to carry on all pre-disease activities without restriction; 1= restricted in physically strenuous activity but ambulatory and able to carry out work of a light and sedentary nature; 2= ambulatory and capable of all self-care, but unable to carry out any work activities, up and about more than 50% of waking hours; 3= capable of only limited self-care, confined to bed/chair \>50% of waking hours; 4= completely disabled, cannot carry on any self-care, totally confined to bed/chair: 5= dead.

Part 1 and Part 2: Time to Definitive 1 Point Deterioration in Eastern Cooperative Oncology Group Performance Status (ECOG PS)Baseline up to 30 days from last dose of study drug (up to 30 months for Part 1, excluding Part 1: LGX818 300 mg group; up to 36 months for Part 2 and Part 1 LGX 300 mg group)

ECOG: participant's performance status was measured on a 6-point scale: 0= fully active/able to carry on all pre-disease activities without restriction; 1= restricted in physically strenuous activity but ambulatory and able to carry out work of a light and sedentary nature; 2= ambulatory and capable of all self-care, but unable to carry out any work activities, up and about more than 50 percent (%) of waking hours; 3= capable of only limited self-care, confined to bed/chair \>50% of waking hours; 4= completely disabled, cannot carry on any self-care, totally confined to bed/chair: 5= dead. Definitive deterioration was defined as death due to any cause or decrease in ECOG PS by at least one category from baseline score with no subsequent improvement.

Part 1 and Part 2: Disease Control Rate (DCR)From randomization until disease progression or death, whichever occurred first (up to 29 months for Part 1, excluding Part 1: LGX818 300 mg group; up to 35 months for Part 2 and Part 1 LGX 300 mg group)

DCR was calculated as the percentage of participants with a best overall response (BOR) of CR, PR, or stable disease (SD). CR was defined as disappearance of all non-nodal target lesions. In addition, any pathological lymph nodes assigned as target lesions must have a reduction in short axis to \<10 mm. PR was defined as at least a 30% decrease in the sum of diameter of all target lesions, taking as reference the baseline sum of diameters. Two sets of DCR were considered, one for confirmed and one for unconfirmed responses. Results are reported for confirmed and unconfirmed responses combined. SD: Neither sufficient shrinkage to qualify for PR or CR nor an increase in lesions which would qualify for PD. DCR was based on central review.

Part 1 and Part 2: Time to Definitive 10% Deterioration in the Function Assessment Cancer Therapy-melanoma (FACT-M) SubscaleDate of randomization to date of event or death due to any cause, which ever occurred first (up to 29 months for Part 1, excluding Part 1: LGX818 300 mg group; up to 35 months for Part 2 and Part 1 LGX 300 mg group)

FACT-M:melanoma specific questionnaire to assess participant health-related quality of life. Melanoma specific subscale consists of 16 items related to signs,symptoms,physical/social activities most relevant to participants with advanced-stage melanoma. Other items include physical, functional and social/family well-being (7 items each),emotional well-being (6 items),surgery specific concerns related to melanoma(8 items,not included in this study). Each item range from 0(not at all) to 4(very much), combined to produce subscale scores.Total score range for FACT-M excluding surgery specific items is 0 to 172,higher scores represent better quality of life.Melanoma subscale score range from 0(worst response) to 64(best response),higher score indicated better quality of life. Time to definitive 10% deterioration:time from date of randomization to date of event with at least 10% relative to baseline worsening of corresponding scale score with no later improvement or death due to any cause.

Part 1 and Part 2: Time to Definitive 10% Deterioration in the Global Health Status Score of the European Organization for Research and Treatment of Cancer's Core Quality of Life Questionnaire (EORTC QLQ-C30)Date of randomization to date of event or death due to any cause, which ever occurred first (maximum up to 29 months for Part 1, excluding Part 1: LGX818 300 mg group; up to 35 months for Part 2 and Part 1 LGX 300 mg group)

EORTC QLQ-C30 is 30 item questionnaire composed of 5 multi-item functional subscales (physical, role, cognitive, emotional, social functioning), 3 multi-item symptom scales (fatigue, nausea/vomiting, and pain), global health/quality of life (QOL) subscale and 6 single items assessing other cancer related symptoms (dyspnea, sleep disturbance, appetite, diarrhea, constipation and financial impact of cancer). It employed twenty-eight 4 point Likert scales with responses from "not at all" to "very much" and two 7 point Likert scales for global health and overall QOL. Global health status scale score ranged from 0 to 100. Higher score represented better level of functioning. Time to definitive 10% deterioration: time from date of randomization to date of event with at least 10% relative to baseline worsening of corresponding scale score with no later improvement or death due to any cause.

Part 1 and Part 2: Duration of Response (DOR)From randomization until disease progression, censoring date or death, whichever occurred first (up to 29 months for Part 1, excluding Part 1: LGX818 300 mg group; up to 35 months for Part 2 and Part 1 LGX 300 mg group)

DOR was calculated, as the time from the date of first documented response (CR or PR) to the first documented progression or death due to underlying cancer. DOR was estimated for responders (i.e. participants achieving at least once CR or PR) only using a Kaplan-Meier method. CR was defined as disappearance of all non-nodal target lesions. In addition, any pathological lymph nodes assigned as target lesions must have a reduction in short axis to \<10 mm. PR was defined as at least a 30% decrease in the sum of diameter of all target lesions, taking as reference the baseline sum of diameters. If a participant with a CR or PR had no progression or death due to underlying disease, the participant was censored at the date of last adequate tumor assessment. Results are based on confirmed BIRC response.

Part 1 and Part 2: Change From Baseline in the Function Assessment Cancer Therapy-melanoma (FACT-M) Subscale at Day 1 of Cycle 3, 5, 7, 9, 11, 13, 15, 17, 19, 21, 23, 25 and End of Treatment VisitBaseline (Day 1 of Cycle 1), Day 1 of Cycle 3, 5, 7, 9, 11, 13, 15, 17, 19, 21, 23, 25 and end of treatment visit (within14 days after the last dose of study drug)

FACT-M: melanoma specific questionnaire to assess participant health-related quality of life. Melanoma specific subscale consists of 16 items related to signs, symptoms, physical/social activities most relevant to participants with advanced-stage melanoma. Other items include physical, functional and social/family well-being (7 items each),emotional well-being (6 items),surgery specific concerns related to melanoma(8 items, not included in this study). Each item range from 0(not at all) to 4(very much), combined to produce subscale scores. Total score range for FACT-M excluding surgery specific items is 0 to 172,higher scores represented better quality of life. Melanoma subscale score range from 0(worst response) to 64(best response),higher score indicated better quality of life.

Part 1 and Part 2: Change From Baseline in EuroQoL-5 Dimension-5 Level (EQ-5D-5L) Index Score at Day 1 of Cycle 3, 5, 7, 9, 11, 13, 15, 17, 19, 21, 23, 25 and End of Treatment VisitBaseline (Day 1 of Cycle 1), Day 1 of Cycle 3, 5, 7, 9, 11, 13, 15, 17, 19, 21, 23, 25 and end of treatment visit (within14 days after the last dose of study drug)

EQ-5D-5L is a standardized participant completed questionnaire that measures health status in terms of a single index value or utility score. EQ-5D-5L consisted of two components: a health state profile (descriptive system) and a visual analogue scale (VAS) in which participants rate their overall health status from 0 (worst imaginable) to 100 (best imaginable), where higher scores indicated better health status. EQ-5D health state profile is comprised of 5 dimensions: mobility, self-care, usual activities, pain/discomfort and anxiety/depression. Each dimension has 5 response levels: 1=no problems, 2=slight problems, 3=moderate problems, 4=severe problems and 5=extreme problems. EQ-5D-5L health status index score range between 0 to 1. Higher score indicated better health status.

Part 1 and Part 2: Change From Baseline in Emotional Functioning Scale Score of the EORTC QLQ-C30 at Day 1 of Cycle 3, 5, 7, 9, 11, 13, 15, 17, 19, 21, 23, 25 and End of Treatment VisitBaseline (Day 1 of Cycle 1), Day 1 of Cycle 3, 5, 7, 9, 11, 13, 15, 17, 19, 21, 23, 25 and end of treatment visit (within14 days after the last dose of study drug)

EORTC QLQ-C30 contains 30 items and is composed of multi-item and single-item measures. These include 5 functional scales (physical, role, emotional, cognitive and social functioning), 3 symptom scales (fatigue, nausea/vomiting, and pain), 6 single items (dyspnea, insomnia, appetite loss, constipation, diarrhea and financial impact) and a global health status/quality of life (QOL) scale. The questionnaire employs 28 4-point Likert scales with responses from "not at all" to "very much" and two 7-point Likert scales for global health and overall QOL. Responses to all items converted to 0 to 100 scale. For functional and global QOL scales, higher scores represent a better level of functioning/QOL. For symptom-oriented scales, a higher score represented more severe symptoms.

Part 1 and Part 2: Change From Baseline in Physical Functioning Scale Score of the EORTC QLQ-C30 at Day 1 of Cycle 3, 5, 7, 9, 11, 13, 15, 17, 19, 21, 23, 25 and End of Treatment VisitBaseline (Day 1 of Cycle 1), Day 1 of Cycle 3, 5, 7, 9, 11, 13, 15, 17, 19, 21, 23, 25 and end of treatment visit (within14 days after the last dose of study drug)

EORTC QLQ-C30 contains 30 items and is composed of multi-item and single-item measures. These include 5 functional scales (physical, role, emotional, cognitive and social functioning), 3 symptom scales (fatigue, nausea/vomiting, and pain), 6 single items (dyspnea, insomnia, appetite loss, constipation, diarrhea and financial impact) and a global health status/quality of life (QOL) scale. The questionnaire employs 28 4-point Likert scales with responses from "not at all" to "very much" and two 7-point Likert scales for global health and overall QOL. Responses to all items converted to 0 to 100 scale. For functional and global QOL scales, higher scores represented a better level of functioning/QOL. For symptom-oriented scales, a higher score represented more severe symptoms.

Part 1 and Part 2: Change From Baseline in Social Functioning Scale Score of the EORTC QLQ-C30 at Day 1 of Cycle 3, 5, 7, 9, 11, 13, 15, 17, 19, 21, 23, 25 and End of Treatment VisitBaseline (Day 1 of Cycle 1), Day 1 of Cycle 3, 5, 7, 9, 11, 13, 15, 17, 19, 21, 23, 25 and end of treatment visit (within14 days after the last dose of study drug)

EORTC QLQ-C30 contains 30 items and is composed of multi-item and single-item measures. These include 5 functional scales (physical, role, emotional, cognitive and social functioning), 3 symptom scales (fatigue, nausea/vomiting, and pain), 6 single items (dyspnea, insomnia, appetite loss, constipation, diarrhea and financial impact) and a global health status/quality of life (QOL) scale. The questionnaire employs 28 4-point Likert scales with responses from "not at all" to "very much" and two 7-point Likert scales for global health and overall QOL. Responses to all items converted to 0 to 100 scale. For functional and global QOL scales, higher scores represented a better level of functioning/QOL. For symptom-oriented scales, a higher score represented more severe symptoms.

Part 1: Plasma Concentrations of LGX 818Cycle 1 Day 1: pre-dose, 0.5, 1.5, 4 to 8 hours post dose; Cycle 2 Day 1: pre-dose; Cycle 3 Day 1: pre-dose
Part 2: Plasma Concentrations of LGX 818Cycle 1 Day 1: pre-dose, 0.5, 1.5, 4 to 8 hours post dose; Cycle 2 Day 1: pre-dose; Cycle 3 Day 1: pre-dose
Part 2: Plasma Concentrations of MEK162Cycle 1 Day 1: pre-dose, 0.5, 1.5, 4 to 8, hours post dose; Cycle 2 Day 1: pre-dose; Cycle 3 Day 1: pre-dose

Trial Locations

Locations (349)

Tulsa Cancer Institute PLLC

🇺🇸

Tulsa, Oklahoma, United States

University of Pittsburgh Cancer Institute

🇺🇸

Pittsburgh, Pennsylvania, United States

University of Tennessee Medical Center Cancer Institute

🇺🇸

Knoxville, Tennessee, United States

Universitatsklinikum Leipzig

🇩🇪

Leipzig, Sachsen, Germany

University Hospital Schleswig-Holstein, Campus Kiel

🇩🇪

Kiel, Germany

Universitatsklinikum Schleswig-Holstein

🇩🇪

Lübeck, Germany

Universitatsklinikum Schleswig-Holstein - Kiel

🇩🇪

Kiel, Germany

Universitatsklinikum Schleswig-Holstein, Campus Lubeck

🇩🇪

Lübeck, Schleswig-holstein, Germany

Charite-Universitaetsmedizin Berlin

🇩🇪

Berlin, Germany

Universitätsklinikum Bonn

🇩🇪

Bonn, Germany

University Hospital Carl Gustav Carus at the Technical University of Dresden

🇩🇪

Dresden, Germany

Universitätsklinikum Carl Gustav Carus an der TU Dresden

🇩🇪

Dresden, Germany

Überörtliche Radiologische Gemeinschaftspraxis Dresden

🇩🇪

Dresden, Germany

Diagnostische und interventionelle Radiologie und Neuroradiologie

🇩🇪

Erfurt, Germany

Klinik fur Hautkrankheiten und Allergologie, Helios Hauttumorzentrum Erfurt, Helios Klinikum Erfurt

🇩🇪

Erfurt, Germany

Zuyderland Medisch Centrum

🇳🇱

Heerlen, Limburg, Netherlands

VU Medisch Centrum

🇳🇱

Amsterdam, Noord Holland, Netherlands

Amphia Ziekenhuis

🇳🇱

Breda, Noord-brabant, Netherlands

Hospital Civil (Hospital Regional Universitario de Malaga)

🇪🇸

Malaga, Spain

Hospital Regional Universitario de Malaga ? Hospital General

🇪🇸

Malaga, Spain

Hospital Universitario Virgen del Rocio - PPDS

🇪🇸

Sevilla, Spain

Fundacion Instituto Valenciano de Oncologia

🇪🇸

Valencia, Spain

Gävle Sjukhus

🇸🇪

Gavle, Sweden

Sahlgrenska Universitetssjukhuset

🇸🇪

Göteborg, Sweden

Skanes Universitetssjukhus Lund

🇸🇪

Lund, Sweden

Karolinska Universitetssjukhuset Solna

🇸🇪

Solna, Sweden

Uppsala Universitet

🇸🇪

Uppsala, Sweden

Universitätsspital Zürich

🇨🇭

Zurich Flughafen, Switzerland

Inselspital Bern

🇨🇭

Bern, Switzerland

Dr. med. Nicole Gasser

🇨🇭

Zürich, Switzerland

Dr.med. Ursula Urner

🇨🇭

Zürich, Switzerland

Institut für diagnostische und interventionelle Radiologie

🇨🇭

Zürich, Switzerland

Ege University Medical Faculty

🇹🇷

Bornova, Turkey

Ege University Medical aculty

🇹🇷

Izmir, Turkey

Sifa Universitesi Bornova Egitim Arastirma Hastanesi

🇹🇷

Izmir, Turkey

Addenbrookes Hospital

🇬🇧

Cambridge, Cambridgeshire, United Kingdom

Mid Essex Hospital Services NHS Trust

🇬🇧

Broomfield, Chelmsford, Essex, United Kingdom

The Royal Marsden NHS Foundation Trust

🇬🇧

London, Chelsea, United Kingdom

CHU de Reims - Hôpital Robert Debré

🇫🇷

Reims, France

Nouvel Hopital Civil

🇫🇷

Strasbourg, France

Cardiologist Private Practice

🇫🇷

Templemars, France

Fondazione IRCCS Policlinico San Matteo di Pavia

🇮🇹

Pavia, Italy

Azienda Ospedaliera Civile Maria Paternò Arezzo Ragusa

🇮🇹

Ragusa, Italy

S. C. Oncologia Medica Presidio Ospedaliero Maria Paterno Arezzo

🇮🇹

Ragusa, Italy

Policlinico Universitario Campus Biomedico

🇮🇹

Rome, Italy

Azienza Ospedaliera Universitaria Senese

🇮🇹

Siena, Italy

Ospedale Koelliker

🇮🇹

Torino, Italy

Azienda Sanitaria Universitaria Integrata di Udine - PO Universitario Santa Maria della Misericordia

🇮🇹

Udine, Italy

Kyushu University Hospital

🇯🇵

Fukuoka-shi, Fukuoka, Japan

Shinshu University Hospital

🇯🇵

Matsumoto, Nagano, Japan

Niigata Cancer Center Hospital

🇯🇵

Niigata, Japan

National Cancer Center Hospital

🇯🇵

Chuo-ku, Tokyo, Japan

National Hospital Organization Osaka National Hospital

🇯🇵

Osaka, Ôsaka, Japan

Samsung Medical Center - PPDS

🇰🇷

Seoul, Korea, Republic of

Asan Medical Center - PPDS

🇰🇷

Seoul, Korea, Republic of

Seoul National University Hospital

🇰🇷

Seoul, Korea, Republic of

Severance Hospital Yonsei University Health System - PPDS

🇰🇷

Seoul, Korea, Republic of

Instituto Nacional de Cancerologia

🇲🇽

Mexico, DF, Mexico

Medica Sur, S. A. B de C. V. (Centro de Investigación Farmacológica y Biotecnológica CIF-BIOTEC)

🇲🇽

Mexico, Mexico

Instituto Nacional de Cardiología Ignacio Chavez

🇲🇽

Mexico, Mexico

Radboud University Nijmegen Medical Centre

🇳🇱

Nijmegen, Gelderland, Netherlands

Singapore General Hospital (SGH)

🇸🇬

Singapore, Singapore

Hospital Arnau de Vilanova

🇪🇸

Lleida, Spain

Hospital Universitari Arnau de Vilanova

🇪🇸

Lleida, Spain

Hospital General Universitario Gregorio Maranon

🇪🇸

Madrid, Spain

Hospital Universitario 12 de Octubre

🇪🇸

Madrid, Spain

Hospital Universitario Ramon y Cajal

🇪🇸

Madrid, Spain

University of Miami

🇺🇸

Miami, Florida, United States

Hattiesburg Clinic Oncology Hem

🇺🇸

Hattiesburg, Mississippi, United States

UT Southwestern Medical Center at Dallas

🇺🇸

Dallas, Texas, United States

The Queen Elizabeth Hospital

🇦🇺

Woodville, South Australia, Australia

AMO - Assistência Multidisciplinar em Oncologia

🇧🇷

Salvador, Bahia, Brazil

Klinikum Bayreuth GmbH

🇩🇪

Bayreuth, Bayern, Germany

Istituto Dermopatico dell'Immacolata IRCCS

🇮🇹

Roma, Lazio, Italy

Hospital Universitario Dr. Jose Eleuterio Gonzalez

🇲🇽

Monterrey, Nuevo LEON, Mexico

Vision Optical

🇦🇺

Southport, Queensland, Australia

Cancun Oncology Center Galenia

🇲🇽

Cancun, Quintana ROO, Mexico

Gazi University Medical Faculty Gazi Hospital

🇹🇷

Ankara, Turkey

Medisch Centrum Leeuwarden

🇳🇱

Leeuwarden, Friesland, Netherlands

Hospital Universitario La Paz - PPDS

🇪🇸

Madrid, Spain

Universitetssjukhuset i Linköping

🇸🇪

Linköping, Sweden

ASST degli Spedali Civili di Brescia - Spedali Civili di Brescia - INCIPIT - PIN

🇮🇹

Brescia, Lombardia, Italy

Istituto Nazionale Dei Tumori

🇮🇹

Milano, Lombardia, Italy

ASST Grande Ospedale Metropolitano Niguarda - Presidio Ospedaliero Ospedale Niguarda

🇮🇹

Milano, Lombardia, Italy

Mount Vernon Hospital

🇬🇧

Northwood, London, CITY OF, United Kingdom

UAB Comprehensive Cancer Center

🇺🇸

Birmingham, Alabama, United States

University of Illinois Hospital and Health Sciences System - Investigational Drug Service

🇺🇸

Chicago, Illinois, United States

Eye & Ear Infirmary- Opthalmology

🇺🇸

Chicago, Illinois, United States

UAB The Kirklin Clinic

🇺🇸

Birmingham, Alabama, United States

Retinal Consultants of Alabama P.C.

🇺🇸

Birmingham, Alabama, United States

UAB Callahan Eye Hospital

🇺🇸

Birmingham, Alabama, United States

University of Alabama at Birmingham

🇺🇸

Birmingham, Alabama, United States

Highlands Oncology Group

🇺🇸

Rogers, Arkansas, United States

Highlands Oncology Group - Fayetteville

🇺🇸

Springdale, Arkansas, United States

UC Irvine Medical Center

🇺🇸

Orange, California, United States

Rocky Mountain Cancer Centers (Williams) - USOR

🇺🇸

Denver, Colorado, United States

Rocky Mountain Cancer Centers

🇺🇸

Pueblo, Colorado, United States

Specialty Eye Care

🇺🇸

Parker, Colorado, United States

University Cancer Institute

🇺🇸

Boynton Beach, Florida, United States

University of Illinois at Chicago

🇺🇸

Chicago, Illinois, United States

University of Illinois Hospital and Health Sciences System

🇺🇸

Chicago, Illinois, United States

University of Illinois Medical Center

🇺🇸

Chicago, Illinois, United States

University of Vermont Medical Center

🇺🇸

Burlington, Vermont, United States

University of Vermont Cancer Center

🇺🇸

Burlington, Vermont, United States

Goshen Center For Cancer Care

🇺🇸

Goshen, Indiana, United States

Lack's Cancer Center at Mercy Health Saint Mary's

🇺🇸

Grand Rapids, Michigan, United States

Mercy Health Hauenstein Neuroscience Center Neuro-Ophthalmology (Clinic)

🇺🇸

Grand Rapids, Michigan, United States

Retina Specialists of Michigan

🇺🇸

Grand Rapids, Michigan, United States

Jackson Oncology Associates - St. Dominic Hospital

🇺🇸

Jackson, Mississippi, United States

Jackson Oncology Associates, PLLC

🇺🇸

Jackson, Mississippi, United States

Hackensack University Medical Center

🇺🇸

Hackensack, New Jersey, United States

Hackensack University Medical Cente

🇺🇸

Hackensack, New Jersey, United States

Investigational Drug Service, Department of Pharmacy (Investigational Product)

🇺🇸

Rochester, New York, United States

University of Rochester Medical Center - PPDS

🇺🇸

Rochester, New York, United States

Dr. Dennis B. Kay (Ophthalmologist)

🇺🇸

Dallas, Texas, United States

Texas Oncology - Baylor Charles A. Sammons Cancer Center

🇺🇸

Dallas, Texas, United States

Virginia Cancer Specialists, PC

🇺🇸

Leesburg, Virginia, United States

Virginia Cancer Specialists

🇺🇸

Fairfax, Virginia, United States

Virginia Cancer Specialists (Leesburg) - USOR

🇺🇸

Leesburg, Virginia, United States

Northern Virginia Ophthalmology Associates

🇺🇸

Falls Church, Virginia, United States

Wenatchee Valley Hospital & Clinics

🇺🇸

Wenatchee, Washington, United States

Wenatchee Valley Hospitals & Clinics

🇺🇸

Wenatchee, Washington, United States

Wenatchee Valley Medical Center

🇺🇸

Wenatchee, Washington, United States

Lake Macquarie Private Hospital

🇦🇺

Gateshead, New South Wales, Australia

HPS Pharmacy

🇦🇺

Southport, Queensland, Australia

Tasman Oncology Research

🇦🇺

Southport, Queensland, Australia

Fundación CENIT para la Investigación en Neurociencias

🇦🇷

Caba, Buenos Aires, Argentina

Organización Médica de Investigación

🇦🇷

Buenos Aires, Ciudad Autónoma DE Buenosaires, Argentina

Fundación Investigar

🇦🇷

Buenos Aires, Ciudad Autónoma DE Buenosaires, Argentina

Sanatorio de La Providencia

🇦🇷

Buenos Aires, Ciudad Autónoma DE Buenosaires, Argentina

Hospital Italiano de Buenos Aires

🇦🇷

Buenos Aires, Ciudad Autónoma DE Buenosaires, Argentina

Instituto Médico Especializado Alexander Fleming

🇦🇷

Buenos Aires, Ciudad Autónoma DE Buenosaires, Argentina

Centro de Diagnóstico Dr. Enrique Rossi

🇦🇷

Buenos Aires, Ciudad Autónoma DE Buenosaires, Argentina

Princess Alexandra Hospital

🇦🇺

Woolloongabba, Queensland, Australia

The Alfred Hospital

🇦🇺

Prahran, Victoria, Australia

Sir Charles Gairdner Hospital Pharmacy Department

🇦🇺

Nedlands, Western Australia, Australia

Sir Charles Gairdner Hospital

🇦🇺

Nedlands, Western Australia, Australia

Instituto de Medicina Integral Professor Fernando Figueira

🇧🇷

Recife, Pernambuco, Brazil

Associação Hospital de Caridade Ijuí

🇧🇷

Ijuí, RIO Grande DO SUL, Brazil

Hospital de Clinicas de Porto Alegre (HCPA) - PPDS

🇧🇷

Porto Alegre, RIO Grande DO SUL, Brazil

Fundação PIO XII

🇧🇷

Barretos, SÃO Paulo, Brazil

Liga Norte Riograndense Contra O Cancer

🇧🇷

Natal, Brazil

Hospital do Cancer I - Instituto Nacional de Cancer - INCA

🇧🇷

Rio de Janeiro, Brazil

INCA Instituto Nacional de Cancer

🇧🇷

Rio de Janeiro, Brazil

Hospital BP Mirante

🇧🇷

Sao Paulo, Brazil

Tom Baker Cancer Centre

🇨🇦

Calgary, Alberta, Canada

SunnyBrook Health Sciences Centre

🇨🇦

Toronto, Ontario, Canada

Sunnybrook Research Institute

🇨🇦

Toronto, Ontario, Canada

Toronto General Hospital

🇨🇦

Toronto, Ontario, Canada

Princess Margaret Cancer Centre

🇨🇦

Toronto, Ontario, Canada

Centre Hospitalier De L'Universite De Montreal Hospital Notre Dame

🇨🇦

Montreal, Quebec, Canada

CHUM Notrea Dame Hospital

🇨🇦

Montreal, Quebec, Canada

Centre Hospitalier de l'Universite de Montreal

🇨🇦

Montreal, Quebec, Canada

McGill University Health center

🇨🇦

Montreal, Quebec, Canada

CHU de Quebec-Universite Laval

🇨🇦

Quebec City, Quebec, Canada

CHU de Quebec- L'Hotel-Dieu de Quebec

🇨🇦

Québec, Quebec, Canada

Centre de Sante Et Services Sociaux Richelieu Yamaska

🇨🇦

Sainte Hyacinthe, Quebec, Canada

Centre Hospitalier Universitaire de Quebec - Hotel - Dieu de Quebec - Universite Laval

🇨🇦

Quebec, Canada

CHU de Quebec-Universite Laval - L' Hotel - Dieu de Quebec

🇨🇦

Quebec, Canada

Service de PneumologieCHU Lyon Sud

🇫🇷

Pierre-bénite, France

Hospital Universitario San Ignacio

🇨🇴

Bogotá, Pbx (57-1), Colombia

Mou/Mmci - Ppds

🇨🇿

Brno, Jihomoravský KRAJ, Czechia

Fakultni nemocnice Ostrava

🇨🇿

Ostrava Poruba, Czechia

Fakultni nemocnice Kralovske Vinohrady

🇨🇿

Praha 10, Praha, Hlavní Mesto, Czechia

Vseobecna Fakultni Nemocnice V Praze

🇨🇿

Praha, Czechia

Fakultni nemocnice u sv. Anny v Brne

🇨🇿

Brno, Czechia

Fakultni nemocnice Olomouc

🇨🇿

Olomouc, Czechia

General Faculty Hospital

🇨🇿

Praha 2, Czechia

Vseobecna Fakultni Nemocnice V Praze-U Nemocnice 499/2

🇨🇿

Praha, Czechia

CHU de Nice

🇫🇷

Nice, Alpes-maritimes, France

Hôpital Saint-André

🇫🇷

Bordeaux, Gironde, France

CHU de Grenoble

🇫🇷

Grenoble, Isère, France

Hôpital Robert Debré

🇫🇷

Reims, Marne, France

CHRU de Lille - Hôpital Huriet

🇫🇷

Lille, Nord, France

Centre Léon Bérard Centre Régional de Lutte Contre Le Cancer Rhône Alpes

🇫🇷

Lyon, Rhone, France

Hôpital de La Croix Rousse

🇫🇷

Lyon, Rhône, France

Centre Hospitalier Le Mans

🇫🇷

Le Mans, Sarthe, France

Institut Gustave Roussy

🇫🇷

Villejuif, France

CHU de Bordeaux - Hopital Saint Andre

🇫🇷

Bordeaux, France

Hopital Saint Andre Unite de Cancerologie Service de Dermatologie

🇫🇷

Bordeaux, France

Centre Hospitalier Universitaire Ambroise Paré

🇫🇷

Boulogne-Billancourt, France

Clinique de la Louvière

🇫🇷

Lille, France

Hôpital D'Instruction des Armées Desgenettes

🇫🇷

Lyon, France

Groupe Hospitalier Archet I Et II

🇫🇷

Nice, France

Hopital Lariboisiere

🇫🇷

Paris, France

Institut Mutualiste Montsouris

🇫🇷

Paris, France

Ophtalmologist office

🇫🇷

Paris, France

Hôpital Saint louis

🇫🇷

Paris, France

Hospices Civils de Lyon - Hopital Lyon Sud

🇫🇷

Pierre Benite, France

Universitaetsklinikum Freiburg

🇩🇪

Freiburg im Breisgau, Baden-württemberg, Germany

University Clinic Heidelberg - PPDS

🇩🇪

Heidelberg, Germany

Klinikum Mannheim Universitätsklinikum gGmbH

🇩🇪

Mannheim, Baden-württemberg, Germany

Universitätsklinikum Tübingen

🇩🇪

Tübingen, Germany

Universitätsklinikum Ulm

🇩🇪

Ulm, Germany

Hautklinik, Klinikum Nürnberg, Universitätsklinik der Paracelsus Medizinischen Privatuniversität

🇩🇪

München, Germany

LMU Klinikum der Universität München

🇩🇪

München, Bayern, Germany

LMU Klinikum

🇩🇪

München, Bayern, Germany

Institut für Röntgendiagnostik

🇩🇪

Regensburg, Bayern, Germany

University Clinic Regensburg - PPDS

🇩🇪

Regensburg, Bayern, Germany

Universitätsklinikum Würzburg

🇩🇪

Würzburg, Bayern, Germany

Universitätsklinikum Frankfurt

🇩🇪

Frankfurt, Hessen, Germany

Gesundheit Nordhessen Holding AG

🇩🇪

Kassel, Hessen, Germany

Klinikum Kassel

🇩🇪

Kassel, Hessen, Germany

Zentrum für Radiologie

🇩🇪

Kassel, Hessen, Germany

Augenarztzentrum Buxtehude

🇩🇪

Buxtehude, Niedersachsen, Germany

Elben Klinken Stade ? Buxtehude

🇩🇪

Buxtehude, Niedersachsen, Germany

Augenklinik Universitätsklinikum Bonn

🇩🇪

Bonn, Nordrhein-westfalen, Germany

Institut für Diagnostische Radiologie, Neuroradiologie und Nuklearmedizin

🇩🇪

Minden, Nordrhein-westfalen, Germany

Johannes Wesling Klinikum Minden

🇩🇪

Minden, Nordrhein-westfalen, Germany

Mühlenkreiskliniken - Johannes Wesling Klinikum Minden

🇩🇪

Minden, Nordrhein-westfalen, Germany

Universitätsmedizin der Johannes Gutenberg-Universität Mainz

🇩🇪

Mainz, Rheinland-pfalz, Germany

Universitätsklinik Magdeburg

🇩🇪

Magdeburg, Sachsen-anhalt, Germany

Universitätsklinikum Magdeburg A.ö.R.

🇩🇪

Magdeburg, Sachsen-anhalt, Germany

Klinik und Poliklinik für Augenheilkunde

🇩🇪

Dresden, Sachsen, Germany

Universitatsklinikum Leipzig AoR

🇩🇪

Leipzig, Sachsen, Germany

Universitätsklinikum Essen

🇩🇪

Essen, Germany

Goethe-University Frankfurt/Main

🇩🇪

Frankfurt/Main, Germany

Universitätsklinikum Freiburg, Klinik für Radiologie

🇩🇪

Freiburg, Germany

Institut für Diagnostische und Interventionelle Radiologie

🇩🇪

Gera, Germany

SRH Wald-Klinikum Gera GmbH

🇩🇪

Gera, Germany

Klinik für Augenheilkunde

🇩🇪

Gera, Germany

Universitätsklinik Hamburg Eppendorf

🇩🇪

Hamburg, Germany

Augenärzte am Kröpcke

🇩🇪

Hannover, Germany

Medizinische Hochschule Hannover (Hannover Medical School)

🇩🇪

Hannover, Germany

Institut für Diagnostische und Interventionelle Radilogie

🇩🇪

Hannover, Germany

Universität des Saarlandes

🇩🇪

Homburg, Germany

Universitätsaugenklinik

🇩🇪

Magdeburg, Germany

Universitätsklinik für Radiologie und Nuklearmedizin

🇩🇪

Magdeburg, Germany

University Hospital Mainz

🇩🇪

Mainz, Germany

Augenklinik Universitätsklinikum Mannheim

🇩🇪

Mannheim, Germany

Augen-Praxis_Minden

🇩🇪

Minden, Germany

LMU Klinikum der Universität

🇩🇪

München, Germany

Fachklinik Hornheide Abteilung für Internistische Onkologie und Hämatologie

🇩🇪

Münster, Germany

Klinikum Nürnberg - Campus Nord

🇩🇪

Nürnberg, Germany

Klinik & Poliklinik für Augenheilkunde

🇩🇪

Regensburg, Germany

Internistische Schwerpunktpraxis Kardiologie Hämatologie Onkologie

🇩🇪

Ulm, Germany

Hygeia Diagnostic and Therapeutic Centre of Athens

🇬🇷

Athens, Attiki, Greece

Laiko General Hospital of Athens

🇬🇷

Athens, Greece

Metropolitan Hospital

🇬🇷

Piraeus, Greece

Debreceni Egyetem Klinikai Kozpont

🇭🇺

Debrecen, Hungary

Magyar Honvédség Egészségügyi Központ

🇭🇺

Budapest, Hungary

Eszak-Pesti Centrumkorhaz -Honvedkorhaz- Podmaniczky utcai telephely

🇭🇺

Budapest, Hungary

Orszagos Onkologiai Intezet

🇭🇺

Budapest, Hungary

Jasz-Nagykun-Szolnok Megyei Hetenyi Geza Korhaz-Rendelointezet

🇭🇺

Szolnok, Hungary

Jasz-Nagykun-Szolnok Varmegyei Hetenyi Geza Korhaz-Rendelointezet

🇭🇺

Szolnok, Hungary

Rambam Health Care Campus

🇮🇱

Haifa, Ḥeifā, Israel

Sheba Medical Center - PPDS

🇮🇱

Ramat Gan, Tel-aviv, Israel

Hadassah Medical Center - PPDS

🇮🇱

Jerusalem, Israel

Azienda Ospedaliero Universitaria Ospedali Riuniti di Ancona-Umberto I G.M. Lancisi G. Salesi

🇮🇹

Torrette Site, Ancona, Italy

Azienda Ospedaliera Universitaria Federico II

🇮🇹

Napoli, Campania, Italy

Azienda Ospedaliero Universitaria Di Bologna Policlinico S Orsola Malpighi-Via Massarenti

🇮🇹

Bologna, Emilia-romagna, Italy

Azienda Ospedaliero Universitaria Di Bologna Policlinico S Orsola Malpighi

🇮🇹

Bologna, Emilia-romagna, Italy

Policlinico Universitario Campus Biomedico Di Roma

🇮🇹

Roma, Lazio, Italy

Istituto Nazionale Tumori Regina Elena

🇮🇹

Roma, Lazio, Italy

Azienda Ospedaliera Sant'Andrea

🇮🇹

Roma, Lazio, Italy

Azienda Ospedaliera Ospedale Di Lecco

🇮🇹

Lecco, Lombardia, Italy

Istituto Europeo Di Oncologia

🇮🇹

Milano, Italy

ASST di Monza - Azienda Ospedaliera San Gerardo

🇮🇹

Monza, Lombardia, Italy

Azienda Ospedaliera San Gerardo

🇮🇹

Monza, Lombardia, Italy

Istituto Clinico Humanitas - Humanitas Cancer Center

🇮🇹

Rozzano, Lombardia, Italy

Istituto Clinico Humanitas

🇮🇹

Rozzano, Lombardia, Italy

Fondazione del Piemonte per l'Oncologia (IRCCS)

🇮🇹

Candiolo, Torino, Italy

Azienda Ospedaliero Universitaria Pisana

🇮🇹

Pisa, Toscana, Italy

Azienda Ospedaliera S Maria Di Terni

🇮🇹

Terni, Umbria, Italy

Azienda Ospedaliera Santa Maria di Terni

🇮🇹

Terni, Umbria, Italy

Clinica Oculistica

🇮🇹

Padua, Veneto, Italy

IRCCS Az. Osp. Universitaria San Martino- IST

🇮🇹

Genoa, Italy

IRCCS Giovanni Paolo II Cancer Institute

🇮🇹

Bari, Italy

ASST Papa Giovanni XXIII - Azienda Ospedaliera Papa Giovanni XXIII

🇮🇹

Bergamo, Italy

Azienda Ospedaliero Universitaria Di Bologna - Policlinico S.Orsola Malpighi

🇮🇹

Bologna, Italy

Istituto Nazionale per lo studio e la cura dei tumori Fondazione Giovanni Pascale

🇮🇹

Napoli, Italy

Istituto Nazionale Tumori IRCCS Fondazione Giovanni Pascale

🇮🇹

Napoli, Italy

Istituto Oncologico Veneto - I.R.C.C.S.

🇮🇹

Padova, Italy

Maxima Medisch Centrum

🇳🇱

Veldhoven, Noord-brabant, Netherlands

Medisch Spectrum Twente

🇳🇱

Enschede, Netherlands

Isala Zwolle

🇳🇱

Zwolle, Overijssel, Netherlands

Medisch Spectrum Twente - Hospital

🇳🇱

Ariënsplein Enschede, Netherlands

Universitair Medisch Centrum Groningen

🇳🇱

Groningen, Netherlands

Zuyderland Medisch Centrum - Heerlen

🇳🇱

Heerlen, Netherlands

Leids Universitair Medisch Centrum

🇳🇱

Leiden, Netherlands

Maastricht University Medical Center

🇳🇱

Maastricht, Netherlands

Erasmus MC

🇳🇱

Rotterdam, Netherlands

Erasmus MC-Daniel den Hoed Oncologisch Centrum

🇳🇱

Rotterdam, Netherlands

Zuyerland Medisch Centrum

🇳🇱

Sittard-Geleen, Netherlands

Oslo universitetssykehus HF, Utprøvingsenheten

🇳🇴

Oslo, Norway

Oslo universitetssykehus HF

🇳🇴

Oslo, Norway

Oslo Myeloma Center - PPDS

🇳🇴

Oslo, Norway

Narodowy Instytut Onkologii im. Marii Sklodowskiej-Curie - Panstwowy Instytut Badawczy w Warszawie

🇵🇱

Warsaw, Mazowieckie, Poland

Centrum Medyczne MAVIT Sp. z o.o.

🇵🇱

Warszawa, Mazowieckie, Poland

Lux Med

🇵🇱

Warszawa, Poland

Instituto Português de Oncologia de Lisboa Francisco Gentil, E.P.E.

🇵🇹

Lisboa, Portugal

Instituto Portugues de Oncologia Do Porto Francisco Gentil Epe - PPDS

🇵🇹

Porto, Portugal

Hospital Garcia de Orta*E.P.E.

🇵🇹

Almada, Portugal

Centro Hospitalar de Lisboa Norte, E.P.E- Hospital de Santa Maria

🇵🇹

Lisboa, Portugal

Centro Hospitalar Universitario Lisboa Norte E.P.E

🇵🇹

Lisboa, Portugal

Hospital de Santa Maria-Avenida Prof. Egas Moniz - PPDS

🇵🇹

Lisboa, Portugal

Hospital de Santa Maria

🇵🇹

Lisboa, Portugal

Russian Oncology Research Center n a N N Blokhin

🇷🇺

Moscow, Russian Federation

Ryazan Regional Clinical Oncology Dispensary

🇷🇺

Ryazan, Russian Federation

Ryazan Clinical Hospital n.a. Semashko

🇷🇺

Ryazan, Russian Federation

Scientific Research Institute of Oncology n.a. N.N. Petrov

🇷🇺

St. Petersburg, Russian Federation

National Cancer Centre - 30 Hospital Blvd

🇸🇬

Singapore, Singapore

National Cancer Centre Singapore

🇸🇬

Singapore, Singapore

Singapore National Eye Research Centre

🇸🇬

Singapore, Singapore

Nemocnica Svateho Michala, a.s.

🇸🇰

Bratislava, Slovakia

Narodny onkologicky ustav - PPDS

🇸🇰

Bratislava, Slovakia

BIONT, a.s.

🇸🇰

Bratislava, Slovakia

POKO POPRAD, s.r.o.

🇸🇰

Poprad, Slovakia

Steve Biko Academic Hospital

🇿🇦

Pretoria, South Africa

Mary Potter Oncology Centre

🇿🇦

Pretoria, South Africa

Hospital Universitario de Jerez

🇪🇸

Jerez De La Frontera, Andalucía, Spain

Hospital Universitario Central de Asturias

🇪🇸

Oviedo, Asturias, Spain

Hospital Universitario Germans Trias i Pujol

🇪🇸

Badalona, Spain

Cetir, Centre Mèdic, S.L

🇪🇸

Barcelona, Cataluña, Spain

Hospital Universitario Puerta de Hierro Majadahonda

🇪🇸

Majadahonda, Madrid, Spain

Hospital Universitario Puerta de Hierro - Majadahonda

🇪🇸

Majadahonda, Spain

Hospital Clinico Universitario Virgen de la Arrixaca

🇪🇸

El Palmar, Murcia, Spain

Clinica Universidad Navarra

🇪🇸

Pamplona, Navarra, Spain

Clinica Universidad de Navarra

🇪🇸

Pamplona, Navarra, Spain

Complejo Hospitalario de Navarra

🇪🇸

Pamplona, Navarra, Spain

Hospital Universitario de Navarra

🇪🇸

Pamplona, Navarra, Spain

Hospital Nuestra Señora de Valme

🇪🇸

Seville, Sevilla, Spain

Hospital General Universitario de Alicante

🇪🇸

Alicante, Spain

Hospital General Universitario Dr. Balmis

🇪🇸

Alicante, Spain

Centro de Oftalmologia Barraquer

🇪🇸

Barcelona, Spain

Hospital Universitario Vall d'Hebron - PPDS

🇪🇸

Barcelona, Spain

Hospital Clinic de Barcelona

🇪🇸

Barcelona, Spain

Hospital Clinic provincial de Barcelona

🇪🇸

Barcelona, Spain

Hospital de La Santa Creu i Sant Pau

🇪🇸

Barcelona, Spain

Onkologikoa

🇪🇸

Donostia-san Sebastián, Spain

Hospital Universitario Virgen de las Nieves

🇪🇸

Granada, Spain

Hospital Universitario A Coruña

🇪🇸

La Coruna, Spain

Royal Preston Hospital

🇬🇧

Preston, Lancashire, United Kingdom

Royal Marsden Hospital - Surrey

🇬🇧

London, London, CITY OF, United Kingdom

The Royal Marsden in Sutton, Surrey - Downs Rd

🇬🇧

London, London, CITY OF, United Kingdom

Royal Surrey County Hospital

🇬🇧

Guildford, Surrey, United Kingdom

Clatterbridge Hospital - NWCRN - PPDS

🇬🇧

Bebbington, Wirral, United Kingdom

Clatterbridge Hospital - PPDS

🇬🇧

Bebington, Wirral, United Kingdom

The Clatterbridge Cancer Centre NHS Foundation Trust

🇬🇧

Bebington, Wirral, United Kingdom

Weston Park Hospital

🇬🇧

Sheffield, York, United Kingdom

Broomfield Hospital

🇬🇧

Broomfield, United Kingdom

Cambridge University Hospitals NHS Foundation Trust

🇬🇧

Cambridge, United Kingdom

St James University Hospital

🇬🇧

Leeds, United Kingdom

Royal Free Hospital

🇬🇧

London, United Kingdom

The Christie NHS Foundation Trust - PPDS

🇬🇧

Manchester, United Kingdom

Churchill Hospital

🇬🇧

Oxford, United Kingdom

Royal Preston Hospital - NWCRN- PPDS

🇬🇧

Preston, United Kingdom

Royal Preston Hospital - PPDS

🇬🇧

Preston, United Kingdom

Clatterbridge Cancer Centre

🇬🇧

Wirral, United Kingdom

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