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Efficacy of Temocillin in Urinary Tract Infection Due to ESBL Producing and AmpC Hyperproducing Enterobacteriaceae

Phase 4
Conditions
Urinary Tract Infections
Interventions
Registration Number
NCT02681263
Lead Sponsor
University Hospital, Grenoble
Brief Summary

The present study aims at demonstrating the efficacy of temocillin in the treatment of UTI requiring parenteral therapy due to a confirmed ESBL producing or AmpC hyperproducing Enterobacteriaceae, resistant to quinolones and Bactrim® in France. In addition, this study will describe and support the use of high dose (6g/day) of temocillin which could be of interest for the treatment urinary tract infection due to multi-resistant bacteria having high MIC (up to 32 mg/L). The investigators will also evaluate the tolerance of the drug by monitoring the adverse event and the incidence of eventual Clostridium difficile associated infection.

Detailed Description

Not available

Recruitment & Eligibility

Status
UNKNOWN
Sex
All
Target Recruitment
25
Inclusion Criteria
  • Age of at least 18 year old
  • Patient benefits from social security
  • Signed informed consent
  • A urinary tract infection due to a confirmed ESBL producing strain (detected by the use of a rapid diagnostic test applied on the urine) requiring parenteral antimicrobial therapy
  • Hospitalized patient
  • For women able to procreate: Use of an acceptable method of birth control throughout the study. Acceptable methods of birth control are: oral contraceptives, intrauterine device (IUD), diaphragm with spermicide and condom. (All forms of hormonal contraception are acceptable
Exclusion Criteria
  • Patient infected with a bacteria which is not an ESBL-producing or AmpC hyperproducing Enterobacteriaceae
  • Patients infected with a strain sensible to both fluoroquinolones and trimethoprim/sulfamethoxazole
  • Patients infected with a strain resistant to temocillin
  • Hospital-acquired urinary tract infection (defined as a urinary infection that occurred at least 48h post admission in the hospital)
  • Patients has received any dose of active antimicrobial therapy (an antibiotic to which the infecting bacterium is susceptible) in the last 48h (prior to enrolment) except ≤ 2 dose of gentamicin.
  • Patients presenting another site of infection than urinary (except onset of bacteraemia from urinary tract origin) due to Gram negative bacteria.
  • Patients needing concomitant antimicrobial therapy.
  • Septic shock
  • Children (up to 18 years old)
  • Women who is pregnant, breastfeeding, or expecting to conceive at any time during the study (pregnancy test will be conducted for woman without menopause)
  • Patients with any kind of urinary/bladder catheter (JJ ureteral probe, ...)
  • Hypersensitivity to the active substance, to penicillins or to any other type of beta-lactam agent
  • Chronically dialyzed patients
  • Patients having a creatinine clearance < 30 mL/min
  • Complete obstruction of the urinary tract
  • Perinephretic or intrarenal abscesses
  • Tutorship or curatorship patient
  • Patient unable to give his consent

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
TemocillinTemocillinTreatment duration with a minimum of 5 days administration of the study drug: Temocillin (Negaban®) 6g/day (2g/tid) and as monotherapy. Total antibiotic treatment between 10 and 14 days according to local guidelines (up to 21 days in immunosuppressed patients).
Primary Outcome Measures
NameTimeMethod
Microbiological efficacy at Test of Cure in patients microbiologically evaluable7 days post end of Temocillin Treatment

The microbiological efficacy will be assessed by quantitative urine culture and defined as follows:

* Eradication : \< 10\^3 CFU/mL of the baseline pathogen

* Persistence : ≥ 10\^3 CFU/ml of the baseline pathogen

* Superinfection : ≥ 10\^5 CFU/ml of another uropathogen during therapy

* New infection : ≥ 10\^5 CFU/ml of another uropathogen after therapy

* Relapse : eradication at TOC but ≥ 10\^3 CFU/mL of the baseline pathogen at FU Overall microbiological response will be determined as "unfavorable" if persistence or superinfection or new infection or relapse.

Secondary Outcome Measures
NameTimeMethod
Clinical efficacy in clinical evaluable group3 weeks for end of Temocillin Treatment

Each patient's response will be categorized as cure (resolution of all clinical symptoms), improvement (normalization of body temperature but persistence of either urinary syndrome or flank pain) or failure (persistence of baseline clinical symptoms or emergence of new symptoms related to UTI).

Development of resistance to temocillin during treatment3 weeks for end of Temocillin Treatment

The acquisition of resistance will be monitored in the central laboratory and is defined as an increase in MIC of at least 4 dilutions.

Microbiological efficacy3 weeks for end of Temocillin Treatment

The microbiological efficacy will be assessed by quantitative urine culture and defined as follows:

* Eradication : \< 10\^3 CFU/mL of the baseline pathogen

* Persistence : ≥ 10\^3 CFU/ml of the baseline pathogen

* Superinfection : ≥ 10\^5 CFU/ml of another uropathogen during therapy

* New infection : ≥ 10\^5 CFU/ml of another uropathogen after therapy

* Relapse : eradication at TOC but ≥ 10\^3 CFU/mL of the baseline pathogen at FU

Trial Locations

Locations (19)

APHP - Avicenne Hospital

🇫🇷

Bobigny, France

APHP - Bicêtre Hospital

🇫🇷

Kremlin-Bicêtre, France

APHP - St Louis

🇫🇷

Paris, France

APHP - Bichat Hospital

🇫🇷

Paris, France

CHU de Rouen

🇫🇷

Rouen, France

CHU de Saint Etienne

🇫🇷

Saint Etienne, France

APHP - Beaujon Hospital

🇫🇷

Clichy, France

CHU de Martinique

🇫🇷

Fort De France, France

CH de Perpignan

🇫🇷

Perpignan, France

CHU de Nice

🇫🇷

Nice, France

CH Ajaccio

🇫🇷

Ajaccio, France

CH Annecy Genevois

🇫🇷

Annecy, France

CHU de Pointe à Pitre

🇫🇷

Pointe À Pitre, France

CHU de Poitiers

🇫🇷

Poitiers, France

CHU de Tours

🇫🇷

Tours, France

APHP - Cochin Hospital

🇫🇷

Paris, France

CHU de Grenoble

🇫🇷

Grenoble, France

CHU de Lille

🇫🇷

Lille, France

CHU de Nantes

🇫🇷

Nantes, France

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