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A Pharmacokinetic Study: Ranibizumab, Aflibercept and the Effect of Vitrectomy.

Not Applicable
Completed
Conditions
Age Related Macular Degeneration
Interventions
Registration Number
NCT02174211
Lead Sponsor
King's College Hospital NHS Trust
Brief Summary

To study the effect of pars plana vitrectomy on the intravitreal pharmacokinetics of ranibizumab and to compare the half-life of ranibizumab and aflibercept.

Detailed Description

This study is a prospective, pharmacokinetic study comparing ranibizumab clearance in two groups of patients; those with and without prior vitrectomy. Additionally it will compare ranibizumab clearance to aflibercept clearance as well as the effect on systemic circulating inflammatory and safety markers. Patients will already be receiving ranibizumab or aflibercept therapy - the injection is itself administered irrespective of their participation in this study and therefore this study will not alter medical management or the choice of therapy.

To estimate ranibizumab and aflibercept clearance, it is important to measure serum concentrations at several intervals within the first 24 hours. Participants will ideally have venous blood sampling at the following times after their ranibizumab or aflibercept injection:

* 1 hour

* 2 hours

* 3 hours

* 4 hours

* 6 hours

* 24 hours

* 2 days

* 4 days

* 1 week\*

* 2 weeks

* 4 weeks\*

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
59
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Arm A: Ranibizumab (Lucentis)RanibizumabPrevious Vitrectomy
Arm B: Ranibizumab (Lucentis)RanibizumabNon-vitrectomised, PVD / no PVD
Arm C: Aflibercept (Eylea)AfliberceptNon-vitrectomised, PVD / no PVD
Primary Outcome Measures
NameTimeMethod
Ranibizumab half-life12 Months

Vitrectomised and non-vitrectomised patients

Aflibercept half-life12 Months

Non-vitrectomised patients only

Secondary Outcome Measures
NameTimeMethod
Sub-group analysis of the effect of PVD on ranibizumab half-life12 months

Measurement of half-life (drug assay)

The effect of ranibizumab and aflibercept concentrations on serum inflammatory and safety marker levels.12 months

Assay levels of cytokines and inflammatory/safety markers

Trial Locations

Locations (1)

King's College Hospital NHS Foundation Trust

🇬🇧

London, UK, United Kingdom

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