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Angiotensin II Receptor Blockade in Vascular Ehlers Danlos Syndrome (ARCADE)

Phase 3
Completed
Conditions
Ehlers-Danlos Syndrome, Vascular Type
Interventions
Drug: Placebo
Registration Number
NCT02597361
Lead Sponsor
Assistance Publique - Hôpitaux de Paris
Brief Summary

This study aims to verify the hypothesis that patients with Vascular Ehlers Danlos syndrome (vEDS) should benefit of the blockade of angiotensin (Ang) II noxious effects on their vasculature affected by a defect in type III collagen in addition to the effects celiprolol. This randomized, double blind, placebo controlled trial compares the administration of the Ang II type I receptor blocker (ARB) - irbesartan- to placebo over a 2-year period in vEDS patients with the main objective to reduce the incidence of both symptomatic and asymptomatic vascular events.

Detailed Description

vEDS is a rare life-threatening inherited condition due to mutations at the COL3A1 gene encoding the pro-alpha 1 chain of type III procollagen (OMIM #130050) with unpredictable and recurring arterial dissections/aneurysms starting in the early adulthood. The investigators have previously shown that a treatment with 200-400 mg per day of celiprolol, reduces both fatal and non-fatal vascular events in patients with vEDS. If tolerated, the treatment is now the standard treatment for vEDS. However, despite celiprolol , symptomatic and asymptomatic arterial events continue to occur in vEDS patients. Recent findings suggest a possible deleterious effect of endogenous Angiotensin II on medium size arteries in vEDS patients. The hypothesis of this study is that the blockade of endogenous Ang II will provide supplemental vascular protection and thus reduce recurrence of arterial events in vEDS patients.

The primary objective of this study is to determine in patients with molecularly proven vEDS, whether an Ang II receptor blocker, prescribed at an optimally tolerated dose combined with the reference celiprolol treatment, decreases the 24 months rate of both asymptomatic and symptomatic cardiovascular (CV) events when compared to placebo.

Methodology:

Multicenter, double-blind, randomized (1:1), placebo-controlled, parallel group, study with blind endpoint evaluation in adult vEDS patients.

Main criteria for inclusion:

Patients of both sexes aged 18 to 70 years with molecularly proven vEDS, not in an acute phase of the disease, with no contra-indication for taking an Ang II blocker.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
61
Inclusion Criteria
  • Patients with genetically-proven vEDS (presence of a pathogenic mutation at the COL3A1 gene);
  • Age ≥18 years and <70 years;
  • Men and women with reliable contraception or negative beta-HCG at screening;
  • Celiprolol at the optimal tolerated dose since at least 12 weeks;
  • vEDS patient fully intolerant to celiprolol but not treated with any other drug active on the vascular system, except another beta-blocker;
  • No compelling indication for ARB therapy (renal infarction, hypertension, proteinuric nephropathy, chronic heart failure, myocardial infarction, stroke);
  • Estimated glomerular filtration rate (GFR) ≥ 30ml/min/1,73m2 (MDRD Formula);
  • Normal or clinically acceptable 12-lead ECG;
  • Written informed consent to participate in the study.
Exclusion Criteria

General criteria

  • Unlikely to co-operate in the study and/or poor compliance anticipated by the investigator, e.g., uncooperative attitude, inability to return for follow-up visit, and unlikelihood of completing the study;
  • Participation in another interventional therapeutic study at the same time or within 3 months prior to the beginning of the present study;
  • Participant not affiliated to the French social security;
  • No written informed consent;
  • Severe contrast media allergy, not amenable to pre-treatment Medical and therapeutic criteria
  • History of previous symptomatic visceral complication (any CV event, pulmonary or digestive event) in the 3 months preceding the inclusion;
  • Formal indication for an antihypertensive medication (office BP ≥140/90 mmHg on celiprolol on at least two separated visits, confirmed by daytime ambulatory BP or home BP ≥ 135/85 mmHg);
  • Concomitant treatment with renin-angiotensin-aldosterone system blocking agents apart from the study drug, e.g. ACEI, ARB or aldosterone-antagonist or any renin inhibitor, if given for an elective indication (heart failure, renal infarction, chronic kidney disease, proteinuria, myocardial infarction, stroke);
  • Any cardiac condition that justifies a specific medical care (i.e. second or third degree auriculo-ventricular block, potentially life threatening arrhythmia or other uncontrolled arrhythmia or persistent arrhythmia, clinically significant valvular heart disease);
  • Known significant renal artery stenosis with evidence of renal ischemia (on Duplex ultrasound, CTA, or other exam);
  • Any concurrent life threatening condition other than vEDS with a life expectancy less than 2 years;
  • Likely allergy or hypersensitivity to irbesartan, based on known allergies to drugs of the same class, or which in the opinion of the investigator suggests an increased potential for an adverse hypersensitivity as well as known or suspected contraindications to the study drug;
  • Any condition that in the opinion of the investigator would jeopardize the evaluation of efficacy or safety;
  • Pregnant or nursing (lactating) women, where pregnancy is defined as the state of a female after conception and until the termination of gestation, confirmed by a positive Human Chorionic Gonadotropin (hCG) laboratory test (>5 mIU/ml);
  • Women of child-bearing potential (WOCBP) without reliable contraception.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
IrbesartanIrbesartanIrbesartan: 150 or 300 mg o.d. for 2 years.The up-titration of irbesartan from 150 mg to 300 mg o.d. occurs during the first 8 weeks following randomization and will be driven by clinical, hemodynamic and biological (plasma creatinine and K) tolerability.
PlaceboPlaceboPlacebo once or twice per day for 2 years.
Primary Outcome Measures
NameTimeMethod
Cardiovascular morbidity and mortality2 years

Total number of any non-fatal and fatal cardiovascular events or events related to vEDS

Arterial lesions2 years

number and severity of arterial lesions detected by CTA

Secondary Outcome Measures
NameTimeMethod
Time to first symptomatic clinical morbid and fatal events2 years
Total number of arterial lesions worsened during follow-up2 years
Rate of any symptomatic cardiovascular event2 years

CV death; any morbid and fatal events related to vEDS; Any non fatal CV event; Non-fatal stroke

Occurrence of new asymptomatic arterial lesions (aneurysm, dissection), detected by a systematic CTA2 years

Arterial dissection/rupture/aneurysm in any vascular bed

Number of unplanned hospitalization for any vEDS related event2 years
Total number of arterial lesions detected by vascular DUS2 years

Echo duplex ultrasound made at inclusion, 6, 12, 18 and 24 months

Changes in PWV (Pulse Wave Velocity)2 years

Applanation tonometry made at randomization visit, 6, 12, 18 and 24 months

Changes in large arteries properties (diameter, wall stress, stiffness)2 years

Echotracking made at randomization visit, 6, 12, 18 and 24 months

Decrease in office systolic/diastolic BP2 years

Vital signs (BP and HR) measured by automatic device at each visit

Change in estimated glomerular filtration rate (MDRD)2 years

eGFR evaluated at each visit

Tolerability and safety of the irbesartan assessed by orthostatic hypotension, plasma creatinine, plasma K+ evaluated at each visit2 years
Compliance to treatment2 years

Spot urine for drug determination (celiprolol and irbesartan urinary detection) made at randomization visit and 3, 12 and 24 months

Quality of life2 years

SF36 and HADS questionnaires submitted to participants at randomization visit, 6, 12 and 24 months

Trial Locations

Locations (15)

CHU DE BORDEAUX - Hopital Saint Andre

🇫🇷

Bordeaux, France

CHU DE LYON - Hopital Femme Mere Enfant

🇫🇷

Bron, France

CHU DE TOURS - Hopital Trousseau

🇫🇷

Chambray-les-Tours, France

CHU DE GRENOBLE - Hopital Albert Michallon

🇫🇷

Grenoble, France

CHU DE TOULOUSE - Hopital Rangueil

🇫🇷

Toulouse, France

CHU DE CAEN - Hopital Cote de Nacre

🇫🇷

Caen, France

CHU DE GRENOBLE - Hopital Couple Enfant

🇫🇷

Grenoble, France

CHU DE LYON - Hopital Edouard Herriot

🇫🇷

Lyon, France

CHRU DE LILLE - Hopital Claude Huriez

🇫🇷

Lille, France

CHU DE MONTPELLIER - Hopital Saint Eloi

🇫🇷

Montpellier, France

AP-HP - Hopital Europeen Georges-Pompidou

🇫🇷

Paris, France

CHU DE NANTES - Hopital Hotel-Dieu

🇫🇷

Nantes, France

CHU DE TOULOUSE - Hopital Purpan

🇫🇷

Toulouse, France

AP-HM - Hopital de la Timone

🇫🇷

Marseille, France

CHRU DE NANCY - Institut Lorrain du Coeur et des Vaisseaux

🇫🇷

Vandoeuvre-les-Nancy, France

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