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Dose Finding Trial With a New Treatment (Degarelix) for Prostate Cancer

Phase 2
Completed
Conditions
Prostate Cancer
Interventions
Registration Number
NCT00819156
Lead Sponsor
Ferring Pharmaceuticals
Brief Summary

The purpose of the trial was to evaluate the safety and efficacy of degarelix when comparing six different doses. The patients participating in the trial were treated with degarelix every month for a year. During the treatment the patients had to visit the clinic for investigations. Blood samples for testosterone, dihydrotestosterone, luteinizing hormone, follicle stimulating hormone, and Prostate Specific Antigen were taken and analysed throughout the trial.

Detailed Description

Degarelix was not FDA regulated at the time of the trial. After completion of the trial degarelix has been approved by the FDA and is thus an FDA regulated intervention.

Recruitment & Eligibility

Status
COMPLETED
Sex
Male
Target Recruitment
189
Inclusion Criteria
  • Written informed consent prior to any study related procedures
  • Proven prostate cancer in need for endocrine treatment, except for neoadjuvant hormonal therapy, but including patients with a rising PSA further to prostatectomy or radiotherapy
  • ECOG score to be equal to or above 2
  • Testosterone level within age-specific normal range
  • PSA value equal to or above 2 ng/ml
  • Life expectancy of at least 6 months
Exclusion Criteria
  • Previous or current hormonal treatment of prostate cancer
  • Recent or current treatment with any drugs modifying the testosterone level
  • Candidate for curative treatment such as prostatectomy or radiotherapy
  • History of severe asthma, anaphylactic reactions, angioedema, angioneurotic oedema or Quincke's Oedema
  • Hypersensitivity towards any component of degarelix or mannitol
  • Cancer disease within the last 5 years except for prostate cancer and some skin cancers
  • Signs of liver impairment shown as elevated serum ALT or serum bilirubin
  • Known hepatic disease
  • Other laboratory abnormalities that judged by the investigator would interfere with the patients participation in the trial or the evaluation of the trial results
  • Clinically significant disorder including excessive alcohol or drug abuse that may interfere with trial participation or influence the conclusion of the trial as judged by the investigator
  • Mental incapacity or language barrier precluding adequate understanding or cooperation
  • Having received an investigational product within the last 12 weeks preceding the trial
  • Previous participation in this trial

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Degarelix 240/160degarelixCycle 1 was an initial 240 milligram dose of Degarelix. Cycles 2-13 were maintenance doses of 160 milligrams each of Degarelix. Each cycle was 28 days.
Degarelix 240/120degarelixCycle 1 was an initial 240 milligram dose of Degarelix. Cycles 2-13 were maintenance doses of 120 milligrams each of Degarelix. Each cycle was 28 days.
Degarelix 200/80degarelixCycle 1 was an initial 200 milligram dose of Degarelix. Cycles 2-13 were maintenance doses of 80 milligrams each of Degarelix. Each cycle was 28 days.
Degarelix 200/120degarelixCycle 1 was an initial 200 milligram dose of Degarelix. Cycles 2-13 were maintenance doses of 120 milligrams each of Degarelix. Each cycle was 28 days.
Degarelix 200/160degarelixCycle 1 was an initial 200 milligram dose of Degarelix. Cycles 2-13 were maintenance doses of 160 milligrams each of Degarelix. Each cycle was 28 days.
Degarelix 240/80degarelixCycle 1 was an initial 240 milligram dose of Degarelix. Cycles 2-13 were maintenance doses of 80 milligrams each of Degarelix. Each cycle was 28 days.
Primary Outcome Measures
NameTimeMethod
Number of Patients With Testosterone <=0.5 Nanograms/Milliliter From Day 28 to Day 36412 months

Number of patients who achieved a testosterone level considered a castration level.

Secondary Outcome Measures
NameTimeMethod
Number of Patients With Testoterone <=0.5 Nanogram/Milliliter at Day 3.Day 3

The number of patients who achieved the \<=0.5 nanogram/milliliter level for serum testosterone after 3 days.

Days to 50 Percent Reduction in Prostate-Specific AntigenDay 0 (post dose) to Day 364

Median number of days after the first dose of Degarelix when the prostate-specific antigen levels fell to 50 percent of the baseline value.

Number of Patients With Testosterone Level <=0.5 Nanogram/Milliliter From Day 28 to Day 364 for Patients With Testosterone <=0.5 Nanogram/Milliliter at Day 28Day 28 - 364

Number of patients who maintained a castration level of testosterone (\<=0.5 Nanogram/Milliliter) while on a maintenance dose of Degarelix from Day 28 - 364.

Number of Patients With Testosterone <=0.5 Nanogram/Milliliter at Day 28.Day 28

The number of patients who achieved the \<=0.5 nanogram/milliliter level for serum testosterone after the initial dose cycle.

Days to 90 Percent Reduction in Prostate-Specific AntigenDay 0 (post dose) to Day 364

Median number of days after the first dose of Degarelix when the prostate-specific antigen levels fell to 90 percent of the baseline value.

Days to Prostate-Specific Antigen ProgressionDay 0 (post dose) to Day 364

Median days to prostate-specific antigen increase of \>= 50 percent and \>=5 nanograms/milliliter compared to nadir on two consecutive visits at least two weeks apart.

Median Serum Testosterone LevelsDay 0 (Baseline), Days 1,3,7,14, and 364
Median Prostate-specific Antigen LevelsDay 0 (Baseline), Days 3, 7, 14, and 364
Median Values of Di-HydrotestosteroneDay 0 (Baseline), Days 1, 3, 7, 14, and 364
Median Values for Serum Luteinizing HormoneDay 0 (Baseline), Days 1, 3, 7, 14, and 364
Median Values for Follicle Stimulation HormoneDay 0 (Baseline), Days 1, 3, 7, 14, and 364
The Number of Patients With Abnormal Liver Function Tests364 days

The number of patients who had abnormal (defined as above upper limit of normal range(ULN)) alanine aminotransferase(ALT), aspartate aminotransferase levels, and bilirubin levels. Also includes the number of patients who had ALT increases \>3x ULN, and patients with ALT increases \>3x ULN with concurrent increases in bilirubin \>1.5 ULN.

The Number of Patients With Markedly Abnormal Changes in Vital Signs or Body WeightDay 364

Vital sign and body weight values at the end of the trial are compared to baseline values. The table represents the number of patients in each group with normal baseline values and markedly abnormal end-of-study values.

Trial Locations

Locations (38)

UZ Gasthuisberg

🇧🇪

Leuven, Belgium

Urologische Universitätsklinikum

🇩🇪

Mannheim, Germany

Pez Aladar County Hospital

🇭🇺

Györ, Hungary

Vivantes Klinikum am Urban

🇩🇪

Berlin, Germany

Pavlov medical School, Urology

🇷🇺

St Petersburg, Russian Federation

UCL Saint Luc

🇧🇪

Brussels, Belgium

UZ Gent

🇧🇪

Gent, Belgium

Loretto Krankenhaus

🇩🇪

Freiburg, Germany

Bajcsy-Zsilinszky Hospital, Urology

🇭🇺

Budapest, Hungary

Jahn Ferenc Dél Pesti Hospital, Urology

🇭🇺

Budapest, Hungary

BAZ County Hospital

🇭🇺

Miskolc, Hungary

Hospital of Local Gov. Szeged, Urology

🇭🇺

Szeged, Hungary

Wojewódzki Szpital Specjalisttyczny

🇵🇱

Slupsk, Poland

MÁV Hospital, Urology

🇭🇺

Szolnok, Hungary

AMC

🇳🇱

Amsterdam, Netherlands

CF2 Hospital

🇷🇴

Bucharest, Romania

Atrium MC

🇳🇱

Heerlen, Netherlands

Dr. Th Burghele Hospital

🇷🇴

Bucharest, Romania

Botkin Clinical Hospital

🇷🇺

Moscow, Russian Federation

City Hospital #1

🇷🇺

Moscow, Russian Federation

City Hospital #60

🇷🇺

Moscow, Russian Federation

City Hospital #50

🇷🇺

Moscow, Russian Federation

City Hospital #29

🇷🇺

Moscow, Russian Federation

Institute of Urology of MoH

🇷🇺

Moscow, Russian Federation

"Andros" Urology Clinic

🇷🇺

St Petersburg, Russian Federation

City Hospital #15

🇷🇺

St Petersburg, Russian Federation

Pavlov Medical School Outpatient

🇷🇺

St Petersburg, Russian Federation

City Hospital #26

🇷🇺

St Petersburg, Russian Federation

Sct Petersburg State Medical Academy

🇷🇺

St Petersburg, Russian Federation

370 Clarke Road

🇿🇦

Glenwood, Durban, South Africa

Military Medical Academy, Urology

🇷🇺

St Petersburg, Russian Federation

Pretoria Urology Hospital

🇿🇦

Hatfield, Pretoria, South Africa

WITS Medical School

🇿🇦

Parktown, South Africa

Sunninghill Clinic

🇿🇦

Sunninghill, South Africa

401B Medical Centre

🇿🇦

Pietermaritzburg, South Africa

Euromed AG Klinik

🇩🇪

Fürth, Germany

Fundeni Hospital

🇷🇴

Bucharest, Romania

Sf. Ioan Hospital

🇷🇴

Bucharest, Romania

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