MedPath

Efficacy of Early Administration of Clotinab in Acute Myocardial Infarction

Phase 4
Completed
Conditions
Myocardial Infarction
Interventions
Drug: Clotinab
Registration Number
NCT00841438
Lead Sponsor
Yonsei University
Brief Summary

The ADMIRAL (Platelet glycoprotein IIb/IIIa inhibition with coronary stenting for acute myocardial infarction) study demonstrated that early administration of abciximab in patients with ST elevation acute myocardial infarction prior to PCI improves clinical outcomes but no specifically designed randomized study has addressed the issue of early upstream use of GP IIb/IIIa inhibitors in ST elevation acute myocardial infarction who are undergoing PCI, especially in the era of routine pretreatment with 600 mg of clopidogrel. Therefore, the objective of the randomized ECLAT-STEMI study was to assess the hypothesis that the early upstream use of Clotinab is a useful therapy in patients with ST elevation MI undergoing PCI compared to "provisional use", even after pretreatment with a 600-mg loading dose of clopidogrel.

Detailed Description

It is well known that platelet-mediated thrombosis is account for the pathophysiology of acute coronary syndrome (ACS) (1,2). In the treatment of ACS, intravenous platelet glycoprotein (GP) IIb/IIIa receptor antagonists for platelet aggregation may reduce the risk of ischemic complications (3-7). Therefore, in the management of ACS, Platelet GP IIb/IIIa receptor inhibitors have been developed as a promising new therapy for the reduction of coronary events and the improvement of clinical outcomes.

Abciximab, one of platelet GP IIb/IIIa receptor blockers, was developed by Coller in 1985 and named as 7E3(8). Abciximab is a chimeric human monoclonal antibody and binds to platelet surface GP IIb/IIIa receptor competitively with adhesive molecules such as fibrinogen and von Willebrand factor, and blocks the final stage of platelet aggregation(9). The effect of Abciximab has been proved in many clinical trials such as the EPIC trial(9), EPILOG trial(10), TARGET(11) etc. The contribution of GP IIb/IIIa inhibition in ACS (Tirofiban) is shown in placebo-controlled trials in which upstream GP IIb/IIIa inhibition was initiated upon admission (12,13). Although these results are encouraging, there are few other data to support the use of upstream GP IIb/IIIa inhibitors. Moreover, according to the GUSTO-IV trial (14), the use of Abciximab was not recommended in the manner of upstream use. To evaluate the role of abciximab in conservatively treated non-ST-elevation ACS patients, the GUSTO-IV study randomized 7800 patients with non-ST-elevation ACS to receive either placebo or an Abciximab bolus (0.25 mg/kg) and 24-hour or 48-hour infusion(0.125 ยตg/kg/min). However, in fact, a trend was noted for potential harm with the higher abciximab dose. Even subgroup analyses including high-risk troponin-positive patients showed no benefit with either abciximab regimen (9.7% with placebo, 10.2% with 24-hour abciximab, 11.7% with 48-hour abciximab for death or MI at 30 days, P = NS). Because of these results, the majority of patients received abciximab relatively late, at the time of PCI in clinical practices.

However, the ADMIRAL study (3) demonstrated that early administration of abciximab in patients with ST elevation acute myocardial infarction prior to PCI improves clinical outcomes and also no specifically designed randomized study has addressed the issue of early upstream use of GP IIb/IIIa inhibitors in ST elevation acute myocardial infarction who are undergoing PCI, especially in the era of routine pretreatment with 600 mg of clopidogrel. Therefore, the objective of the randomized ECLAT-STEMI study was to assess the hypothesis that the early upstream use of Clotinab is a useful therapy in patients with ST elevation MI undergoing PCI compared to "provisional use", even after pretreatment with a 600-mg loading dose of clopidogrel.

The Clotinab, a product made in ISU ABXIS CO., LTD, was produced by inserting anti- platelet GP IIb/IIIa DNA into Chinese hamster's ovary cell. Since it contains identical active ingredient as ReoProยฎ on the domestic market, it is expected that the Clotinab has same efficacy to ReoProยฎ as a platelet GP IIb/IIIa receptor inhibitor. Recently, the Clotinab is shown to be safe and effective in preventing ischemic heart complications for high-risk patients who will undergo PCI.

2. Study Protocol 2-1. Objectives: Randomized, controlled, single blind, multi-center trial To assess the hypothesis that the early upstream use of Clotinab is a useful therapy in patients with ST elevation myocardial infarction undergoing PCI compared to "provisional use", even after pretreatment with a 600-mg loading dose of clopidogrel.

2-2. Study Design: Efficacy of CLotinab in ST-elevation Acute myocardial infarction Trial - ST Elevation Myocardial Infarction (The ECLAT - STEMI study)

2-3. Study Endpoints:

1. Primary Endpoint: Efficacy To evaluate the effect of early upstream use of Clotinab (started at emergency room) co-administered with clopidogrel loading dose 600mg in STEMI

- 30 Days MACCE (death, MI, TVR, cerebrovascular event)

2. Secondary Endpoint: Efficacy and Safety To evaluate the safety of early upstream use of Clotinab (started at emergency room) co-administered with clopidogrel loading dose 600mg in STEMI

* TIMI flow at before and after PCI

* Corrected TIMI frame count after PCI

* Procedural success (No reflow incidence)

* MACCE at 9 month

* Major bleeding event (According to TIMI criteria)

* 9 month Angiography Finding

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
786
Inclusion Criteria
  1. The patient must be at least 18-80 years of age.
  2. The patient had the symptoms of acute myocardial infarction within 12 hours with ST segment elevation of more than 1 mm in at least two contiguous leads of EKG or new onset LBBB.
  3. The patient or guardian agrees to the study protocol and provides informed, written consent.
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Exclusion Criteria
  1. Patients to whom PCI can not be undergone within 12 hours from receiving the study drug
  2. Cardiogenic shock or symptomatic hypotension or sitting SBP < 95 mmHg
  3. The history of major surgery, trauma, retinal hemorrhage, significant gastrointestinal or genitourinary bleeding within recent 6 weeks;
  4. History of cerebrovascular attack within two years, or cerebrovascular attack with a significant residual neurological deficit
  5. Severe or malignant hypertension (= sitting SBP > 180 mmHg and/or sitting DBP > 105 mmHg)
  6. The patients who require oral anticoagulants during the trial; patients who have been administrated oral anticoagulants within 7 days
  7. The history or diagnosis of vasculitis; renal insufficiency (the level of serum creatinine is two times higher than the upper limit of normal of each center)
  8. The patients who could not take anti-platelet drugs
  9. The patients who might die of other disease than cardiac disease during the trial.
Read More

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Provisional use of ClotinabClotinabProvisional use of clotinab
Upstream use of clotinabClotinabearly upstream use of clotinab
Primary Outcome Measures
NameTimeMethod
MACCE (death, MI, TVR, cerebrovascular event)30 days
Secondary Outcome Measures
NameTimeMethod
Corrected TIMI frame count after PCIImmediate postprocedure
TIMI flow at before and after PCIImmediate post procedure
MACCE (death, MI, TVR, cerebrovascular event)9 months

Trial Locations

Locations (31)

Dankook University Hospital

๐Ÿ‡ฐ๐Ÿ‡ท

Cheonan, Korea, Republic of

Yeungnam University Hospital

๐Ÿ‡ฐ๐Ÿ‡ท

Daegu, Korea, Republic of

Keimyung University Dongsan Medical Center

๐Ÿ‡ฐ๐Ÿ‡ท

Daegu, Korea, Republic of

Chungnam National University Hospital

๐Ÿ‡ฐ๐Ÿ‡ท

Daejeon, Korea, Republic of

Kyungpook National University Hospital

๐Ÿ‡ฐ๐Ÿ‡ท

Daegu, Korea, Republic of

National Health Insurance Corporation Ilsan Hospital

๐Ÿ‡ฐ๐Ÿ‡ท

Goyang, Korea, Republic of

Chonbuk National University Hospital

๐Ÿ‡ฐ๐Ÿ‡ท

Cheonju, Korea, Republic of

Dongguk University International Hospital

๐Ÿ‡ฐ๐Ÿ‡ท

Goyang, Korea, Republic of

Myongji Hospital

๐Ÿ‡ฐ๐Ÿ‡ท

Goyang, Korea, Republic of

Chonnam National University Hospital

๐Ÿ‡ฐ๐Ÿ‡ท

Gwangju, Korea, Republic of

Inje University Pusan Paik Hospital

๐Ÿ‡ฐ๐Ÿ‡ท

Pusan, Korea, Republic of

Hallym University sacred Heart Hospital

๐Ÿ‡ฐ๐Ÿ‡ท

Pyungchon, Korea, Republic of

Seoul National University Bundang Hospital

๐Ÿ‡ฐ๐Ÿ‡ท

Seongnam, Korea, Republic of

Kyung Hee University Medical Center

๐Ÿ‡ฐ๐Ÿ‡ท

Seoul, Korea, Republic of

Eulji General Hospital

๐Ÿ‡ฐ๐Ÿ‡ท

Seoul, Korea, Republic of

Yonsei University

๐Ÿ‡ฐ๐Ÿ‡ท

Seoul, Korea, Republic of

Samsung Medical Center

๐Ÿ‡ฐ๐Ÿ‡ท

Seoul, Korea, Republic of

Kyung Hee University East-West Nea Medical Center

๐Ÿ‡ฐ๐Ÿ‡ท

Seoul, Korea, Republic of

Inje University Sanggye Paik Hospital

๐Ÿ‡ฐ๐Ÿ‡ท

Seoul, Korea, Republic of

Korea University Anam Hospital

๐Ÿ‡ฐ๐Ÿ‡ท

Seoul, Korea, Republic of

Yonsei University Youngdong Severance Hospital

๐Ÿ‡ฐ๐Ÿ‡ท

Seoul, Korea, Republic of

Catholic University of Korea, St. Mary's Hospital

๐Ÿ‡ฐ๐Ÿ‡ท

Seoul, Korea, Republic of

Ajou University Hospital

๐Ÿ‡ฐ๐Ÿ‡ท

Suwon, Korea, Republic of

Hallym University kangnam sacred Heart Hospital

๐Ÿ‡ฐ๐Ÿ‡ท

Seoul, Korea, Republic of

Wonju Christian Hospital

๐Ÿ‡ฐ๐Ÿ‡ท

Wonju, Korea, Republic of

Korea University Guro Hospital

๐Ÿ‡ฐ๐Ÿ‡ท

Seoul, Korea, Republic of

Pusan National University Hospital

๐Ÿ‡ฐ๐Ÿ‡ท

Pusan, Korea, Republic of

Ulsan University Hospital

๐Ÿ‡ฐ๐Ÿ‡ท

Ulsan, Korea, Republic of

Gachon University Gil Medical Center

๐Ÿ‡ฐ๐Ÿ‡ท

Seoul, Korea, Republic of

Catholic University of Korea, kangnam St. Mary's Hospital

๐Ÿ‡ฐ๐Ÿ‡ท

Seoul, Korea, Republic of

Asan Medical Center

๐Ÿ‡ฐ๐Ÿ‡ท

Seoul, Korea, Republic of

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