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An open-label phase I study of AS-0141 in patients with advanced, metastatic, relapsed or refractory malignancies

Phase 1
Recruiting
Conditions
Solid tumors and hematologic malignancies (AML, MDS, DLBCL)
Registration Number
JPRN-jRCT2031210072
Lead Sponsor
Arimura Akinori
Brief Summary

Not available

Detailed Description

Not available

Recruitment & Eligibility

Status
Recruiting
Sex
All
Target Recruitment
75
Inclusion Criteria

Aged >18 years at time of informed consent
- Histlogically confirmed solid tumors, AML, MDS, or DLBCL for which no standard therapy is available
- Eastern Cooperative Oncology Group (ECOG) Performance Status (PS) <= 1 (solid tumors and DLBCL) or <= 2 (AML and MDS)
- Life expectancy at least 3 months (90days)

Exclusion Criteria

- Patient with known high microsatellite instability(MSH-H)
- Any of the following complicating desease
1) Uncontrolled diabetes
2) Interstitial pneumonia, pulumonary fibrosis, radiation pneumonia (including history)
3) Active infection disease requiring systemic treatment such as antimicrobial agent, antivirus agent
4) AML patients with leukocytosis over 30,000/mm^3 in peripheral leukocyte count
- Any of following serious cardiac or cardiovascular condition
1) Congestive heart failure
2) Class III/ IV heart failure according to the New York Heart Association [NYHA] criteria
3) Ischemic myocardial disease (angina pectoris which needs treatment or revascularization, miocardinal infarction, unstable and symptomatic ischemic heart disease, etc) within 6 months before study drug administration
4) Uncontrolled cardiac arrhythmia (including atrial flutter/fibrillation, ventricular fibrillation, or ventricular tachycardia)
5) Uncontrolled hypertension
6) Ischemic cerebrovascular accident (history of transient ischemic attack, arterial blood circulation reconstruction, etc.)

Study & Design

Study Type
Interventional
Study Design
Not specified
Primary Outcome Measures
NameTimeMethod
Secondary Outcome Measures
NameTimeMethod
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