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Luminal Fructose Kinetics (MARTINI Study)

Phase 2
Recruiting
Conditions
MASLD
Interventions
Registration Number
NCT06539494
Lead Sponsor
Academisch Medisch Centrum - Universiteit van Amsterdam (AMC-UvA)
Brief Summary

In this study the investigators aim is to explore the dynamics of (small) intestinal fructose catabolism in humans and ethanol production in relation to small intestinal signalling pathways and changes in pH, using 13C fructose isotope tracing techniques complemented with direct luminal sampling via small intestinal catheter in biopsy proven MASLD/MASH patients vs healthy (BMI\<25) subjects. Additionally the investigators will repeat the experiment after four weeks of administering omeprazole at a dose of 40 mg twice daily. Omeprazole is a proton pump inhibitor, known to elevate pH from 2-6.

Detailed Description

The investigators will perform a non blinded single centre intervention study in 2x 11 participants

Participants will be either healthy volunteers with a BMI \< 25 and Age 18-65 or patients with MASLD with a BMI \>25, Age 18-65

The objective of the investigators is to study the fructose host/microbial kinetics in humans and to establish the role of (small) intestinal pH on fructose fermentation and endogenous ethanol production in a MASLD/MASH population versus healthy subjects

Subjects will be given omeprazole orally given twice a day 40mg for four weeks

At baseline and after four weeks of omeprazole, a fructose challenge test with labelled fructose and fomepizole and a gastroscopy will be performed, during which a nasal-intestinal catheter will be placed to allow for luminal sampling during the fructose challenge test.

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
22
Inclusion Criteria

In case of the healthy subject group:

  • Adult individuals, age > 18 <65 years
  • Male or postmenopauzal females
  • BMI <25
  • Ability to give informed consent In case of the MASLD/MASH group
  • Adult individuals, age > 18 <65 years
  • Male or postmenopauzal females
  • BMI > 25
  • Biopsy proven MASLD/MASH
  • Ability to give informed consent
Exclusion Criteria
  • History of sustained excess alcohol ingestion: daily consumption >30g/day (3 drinks per day) for males and >20 g/day (2 drinks per day) for females
  • Patients with diabetes
  • Bariatric surgery
  • Other forms of liver disease (e.g. Hepatitis B,C, Wilson disease, hemochromatosis)
  • Proton-pump inhibitor usage one year prior to study participation
  • GLP1, SGLT2i or insulin use
  • Antibiotic use for the past 3 months
  • Probiotic or symbiotic usage
  • Pregnant women
  • Chronic illness (including a known history of heart failure, renal failure (eGFR <30 ml/min), pulmonary disease, gastrointestinal disorders, or hematologic diseases), or other inflammatory diseases
  • Active infection
  • Use of ascal, clopidogrel or other platelet inhibition
  • Smoking
  • Blood thinners
  • Heart failure

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Healthy volunteerOmeprazole 40 MGhealthy volunteers who will get omeprazol daily 2dd40 mg for 4 weeks
Sujbects with MASLDOmeprazole 40 MGPatients with MASLD who will get omeprazol daily 2dd40 mg for 4 weeks
Primary Outcome Measures
NameTimeMethod
Changes in ethanol concentrations before and after omeprazol usagefour weeks

mM (serum, intestinal fluid, urine and feces)

Fructose metabolites in feces before and after omeprazol usage4 weeks

Using 24h feces, the investigators will measure fecal concentrations of fructose metabolites such as ethanol, as well as short chain fatty acids (SCFAs) and bile acids.

Fructose metabolites in urine4 weeks

Using 24h urine, the investigators will measure fecal concentrations of fructose metabolites such as ethanol, as well as SCFAs and bile acids.

Changes in fructose concentrations in peripheral blood before and after omeprazol usage4 weeks

Area under the curve of fructose in peripheral blood upon ingestion of 1 gram / kg unlabeled fructose in combination with 1000mg of D-fructose-13C6 measured during fructose challange test

Changes in fructose metabolites in breath before and after omeprazol usage4 weeks

Area under the curve of various metabolites (e.g. ethanol) will be measured in breath samples upon ingestion of 1 gram / kg unlabeled fructose in combination with 1000mg of D-fructose-13C6 measured during fructose challange test

Changes in serum glucose concentrations before and after omeprazol4 weeks

mmol/l measured during fructose challange test

Secondary Outcome Measures
NameTimeMethod
Changes in dietary intakefour weeks

Participants are asked to fill out an online dietary questionnaire for the 3 days prior to study visits

Bioreactor analysesfour weeks

Using specific anaerobic culturing, ethanol production of fecal samples will be assessed of bacterial strains.

Differences in gene expression in small intestinal biopsies4 weeks

measured by RNA sequencing

Changes in microbiota composition in luminal samplesfour weeks

changes in relative abundance (%) of bacterial phyla, genera and species between groups and after intervention with omeprazol measured by 16sRNA sequencing and shotgun metagenome analysis

Changes in Oral microbiota compositionfour weeks

changes in relative abundance (%) of bacterial phyla, genera and species between groups and after intervention with omeprazol measured by 16sRNA sequencing.

Changes in Fecal microbiota composition4 weeks

changes in relative abundance (%) of bacterial phyla, genera and species between groups and after intervention with omeprazol measured by 16sRNA sequencing and shotgun metagenome analysis

Changes in abundance of post prandial plasma metabolites4 weeks

Postprandial plasma samples will be prepared for the analysis of mainly: organic acids, amino acids, fatty acids, uric acid, glucose and fructose before and after intervention with omeprazol

Trial Locations

Locations (1)

Amsterdam UMC location AMC

🇳🇱

Amsterdam, Netherlands

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