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Safety and Efficacy Study of Adjunctive Antiplatelet Therapy Prior to Primary PCI in Patients With STEMI

Phase 2
Terminated
Conditions
Myocardial Infarction
Interventions
Registration Number
NCT00546260
Lead Sponsor
Portola Pharmaceuticals
Brief Summary

Safety and efficacy of adjunctive antiplatelet therapy prior to primary percutaneous intervention (PCI) in patients with ST-Elevation Myocardial Infarction (STEMI)

Detailed Description

Patients with STEMI who are to undergo primary PCI will be randomized to an intravenous (iv) bolus of placebo vs. PRT060128 prior to angiography.

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
70
Inclusion Criteria
  • Persistent ST elevation ≥ 1mm (≥ 0.1mV) in two contiguous limb leads OR ≥ 2 mm (≥ 0.2mV) in two contiguous precordial leads, AND chest pain ≥ 20 minutes with onset within 6 hours of hospital presentation.
Exclusion Criteria
  • Cardiogenic shock (systolic blood pressure < 90 mm Hg requiring vasopressor or hemodynamic support)
  • Uncontrolled hypertension defined as any measured systolic blood pressure (SBP) > 180 mm Hg or diastolic blood pressure (DBP) ≥ 110 mm Hg after the time -- History or symptoms of a congenital or acquired bleeding disorder or vascular malformation.
  • Recent gastrointestinal bleeding within the last 30 days.
  • Known thrombocytopenia (platelet count < 100,000/mm3).
  • Any treatment with a fibrinolytic agent within the last 7 days.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
1placeboPlacebo for each Dose cohort: 10, 20, 40, and 60 mg
2PRT060128 PotassiumExperimental drug for each Dose cohort: 10, 20, 40, and 60 mg
Primary Outcome Measures
NameTimeMethod
Number of Patients With Thrombolysis in Myocardial Infarction (TIMI) Major/Minor Bleeding, Global Use of Strategies to Open Occluded Coronary Arteries (GUSTO) Severe/Moderate Bleeding Through Hospital Discharge, and Intracranial Hemorrhage Through 30 Days30 days

TIMI Major:Intracranial bleeding or a decrease in the hemoglobin concentration of 5g/dL or more, or 15% or greater decrease in hematocrit.

TIMI Minor:Hemoglobin concentration decreased by 3g/dL (but \<5g/dL) or the hematocrit decreased by 10-15%.

GUSTO Severe/life threatening:Intracranial hemorrhage or bleeding that causes hemodynamic compromise requiring intervention.

GUSTO Moderate:Bleeding that requires bloodtransfusion but does not lead to hemodynamic compromise requiring intervention.

Stroke:New focal neurologic deficit that does not resolve within 24 hours.

Secondary Outcome Measures
NameTimeMethod
Corrected TIMI Frame Count (cTFC) in the Infarct Artery on the Initial Diagnostic Angiogram Before Primary PCITime for contrast to reach a standardized distal coronary landmark in the culprit vessel

This measure was used to assess flow in the epicardial artery. It is the number of cine frames required for contrast to reach a standardized distal coronary landmark in the culprit vessel and was to be counted using an electronic frame counter.

Percentage ST-segment Resolution Prior to PCIBefore primary PCI

The relative effect of PRT060128 on ST-segment measured after PCI and expressed as a percent of ST-Segment prior to PCI. This measure was used to evaluate the dethrombotic and early reperfusion effects of PRT060128 in STEMI.

Trial Locations

Locations (31)

Maine Medical Center

🇺🇸

Portland, Maine, United States

Tallahassee Memorial Medical Center

🇺🇸

Tallahassee, Florida, United States

William Beaumont Hospital - Troy Cardiology

🇺🇸

Troy, Michigan, United States

Geisinger Medical Center

🇺🇸

Danville, Pennsylvania, United States

Trillium Health Centre - Mississaugua

🇨🇦

Mississauga, Ontario, Canada

Genesys Regional Medical Center

🇺🇸

Grand Blanc, Michigan, United States

Foothills Hospital

🇨🇦

Calgary, Alberta, Canada

Victoria Heart Institute, Royal Jubilee Hospital

🇨🇦

Victoria, British Columbia, Canada

Atlantic Health Services

🇨🇦

St. John, New Brunswick, Canada

London Health Sciences

🇨🇦

London, Ontario, Canada

Hospital du Sacre Coeur

🇨🇦

Montreal, Quebec, Canada

St. Joseph Mercy - Oakland

🇺🇸

Pontiac, Michigan, United States

St. Paul's Hospital

🇨🇦

Vancouver, British Columbia, Canada

Sunnybrook Health Sciences Centre

🇨🇦

Toronto, Ontario, Canada

Centre Hospitalier Universitaire de Montreal - Hotel Dieu

🇨🇦

Montreal, Quebec, Canada

Regina General Hospital

🇨🇦

Regina, Saskatchewan, Canada

Hamilton Health Sciences

🇨🇦

Hamilton, Ontario, Canada

William Beaumont Hospital

🇺🇸

Royal Oak, Michigan, United States

Soutlake Regional Health Centre

🇨🇦

Newmarket, Ontario, Canada

Lindner Clinical Trial Center

🇺🇸

Cincinnati, Ohio, United States

General Hospital - Heath Sciences Centre

🇨🇦

St. John's, Newfoundland and Labrador, Canada

Montreal Heart Institute

🇨🇦

Montreal, Quebec, Canada

The Heart Center

🇺🇸

Kingsport, Tennessee, United States

Vancouver General Hospital

🇨🇦

Vancouver, British Columbia, Canada

Washington Adventist Hospital

🇺🇸

Takoma Park, Maryland, United States

Henry Ford Hospital

🇺🇸

Detroit, Michigan, United States

Iowa Heart Center

🇺🇸

Des Moines, Iowa, United States

University of Kentucky Hospital, Gill Heart Center

🇺🇸

Lexington, Kentucky, United States

Royal Alexandria Hospital

🇨🇦

Edmonton, Alberta, Canada

University of Alberta Hospital

🇨🇦

Edmonton, Alberta, Canada

Queen Elizabeth II Health Sciences Centre

🇨🇦

Halifax, Nova Scotia, Canada

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