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Efficacy and Safety of Ramelteon in Subjects With Mild to Moderate Alzheimer's Disease

Phase 2
Completed
Conditions
Chronic Insomnia
Interventions
Drug: Placebo
Registration Number
NCT00325728
Lead Sponsor
Takeda
Brief Summary

The purpose of this study is to determine the efficacy of ramelteon, once daily (QD), in subjects with mild to moderate Alzheimer's Disease and sleep disturbance

Detailed Description

Epidemiological data for 2005 show that an estimated 4.2 million people in the US suffer from Alzheimer's disease, often necessitating caregiver assistance, which can in many cases progress to institutionalization. Subjects with Alzheimer's disease dementia frequently experience disturbed sleep patterns characterized by insufficient nocturnal sleep and excessive daytime napping, which has been associated with both cognitive and behavioral pathology such as impaired daytime functioning, agitation, and nocturnal wandering.

Although the causality of sleep disturbances in Alzheimer's disease remains unclear; some research suggests that the fragmented sleep and associated behavioral disturbances could be related to the degeneration of the serotonergic and noradrenergic innervation of suprachiasmatic nucleus andsubsequent disruption in melatonin secretion patterns. Additionally, research suggests that melatonin levels are decreased in patients with Alzheimer's disease

In the United States, ramelteon is marketed for the treatment of insomnia characterized by difficulty with sleep onset and is under global development for the treatment of transient, chronic insomnia and circadian rhythm sleep disorders. It is believed that ramelteon works by binding melatonin to MT1/MT2 receptors in the suprachiasmatic nucleus which inhibits firing of specific neurons, which is thought to attenuate the alerting signal and allows the homeostatic mechanism to express itself and promote sleep.

Study participation is anticipated to be about 11 weeks (approximately 3 months).

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
74
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
PlaceboPlacebo-
Ramelteon 8 mg QDRamelteon-
Primary Outcome Measures
NameTimeMethod
Mean Nighttime Total Sleep Time as determined by actigraphy.Week 1
Secondary Outcome Measures
NameTimeMethod
Change from Baseline in Nighttime Total Sleep TimeWeeks 2, 4, 6, and 8 or Final Visit
Change from Baseline in Nighttime Wake After Sleep Onset per ActigraphyWeeks 2, 4, 6, and 8 or Final Visit
Change from Baseline in Nighttime Number Of Awakenings per ActigraphyWeeks 2, 4, 6, and 8 or Final Visit
Change from Baseline in Daytime Total Sleep TimeWeeks 2, 4, 6, and 8 or Final Visit
Change from Baseline in the ratio of Daytime Total Sleep Time to Nighttime Total Sleep Time.Weeks 2, 4, 6, and 8 or Final Visit
Change from Baseline in Sleep Efficiency.Weeks 2, 4, 6, and 8 or Final Visit
Percentage of subjects who experience Increase in Nighttime Total Sleep Time of 30 minutes.Weeks 2, 4, 6, and 8 or Final Visit
Number of Daytime Naps.Weeks 2, 4, 6, and 8 or Final Visit
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