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A Study Evaluating the Safety and Efficacy of GLPG5101 (19CP02) in Participants With Non-Hodgkin Lymphoma

Phase 1
Recruiting
Conditions
Relapsed/Refractory B-cell Non-Hodgkin Lymphoma
Lymphomas Non-Hodgkin's B-Cell
Interventions
Genetic: GLPG5101
Registration Number
NCT06561425
Lead Sponsor
Galapagos NV
Brief Summary

This study is evaluating whether an experimental treatment called GLPG5101 helps to treat non-Hodgkin lymphoma (NHL) and if it is safe to use.

This study will be carried out in 2 phases:

* The first phase is to see which doses of GLPG5101 work best with the least number of side effects.

* In the second phase, participants will receive the selected dose(s) based on the results in the first phase.

Detailed Description

Phase 1 Dose escalation phase:

The dose escalation phase is designed to select the doses for dose expansion based on efficacy and safety outcomes.

Three dose levels of GLPG5101 will be evaluated to determine the recommended phase 2 doses (RP2Ds).

Participants with aggressive or indolent forms of Relapsed/Refractory B-cell Non-Hodgkin Lymphoma (r/r NHL) including follicular lymphoma (FL), marginal zone lymphoma (MZL), mantle cell lymphoma (MCL), and Diffuse large B-cell lymphoma (DLBCL) will be enrolled. In case any safety or efficacy differences based on histological subtype of the disease are observed, it may be decided to make decisions regarding dose escalation for a specific subtype(s) independently, upon recommendation by the Safety Review Committee (SRC). Hence the RP2Ds may be different for different subtypes.

Phase 2 Dose expansion phase:

After determination of the RP2Ds, the study continues with the dose expansion phase. Different doses deemed safe by the SRC within the same indication may be explored in the dose-expansion phase to help select the optimal dose for further development.

During this phase, participants will be enrolled into separate disease cohorts as defined by their NHL subtype:

* Cohort 1a: DLBCL second line or greater (2L+)

* Cohort 1b: DLBCL 2L+ with secondary central nervous system lymphoma (SCNSL)

* Cohort 2: High-risk first-line DLBCL

* Cohort 3: Indolent B-cell NHL (FL and MZL third-line or greater \[3L+\])

* Cohort 4: MCL 2L+

* Cohort 5: BL 2L+

* Cohort 6a: PCNSL 2L+

* Cohort 6b: PCNSL first-line consolidation

* Cohort 7: DLBCL-RT 2L+

Participants per disease cohort will be treated at the selected RP2Ds for that disease subtype.

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
250
Inclusion Criteria
  • Histologically confirmed diagnosis of one of the following NHL subtypes: DLBCL, FL grade 1, 2 or 3A, MZL, MCL, BL, PCNSL, DLBCL-RT, High Grade B-cell Lymphoma (HGBL)
  • Relapsed or refractory disease
  • Presence of at least one measurable lesion according to the Lugano classification (except for PCNSL subjects ineligible for ASCT after induction therapy, Cohort 6b)
  • Eastern Cooperative Oncology Group (ECOG) performance status of 0-2 (Participants with ECOG 2 must have serum albumin ≥ 3.4 gram/deciliter)
  • Adequate bone marrow function
  • Adequate renal, hepatic and pulmonary function
  • Women of childbearing potential must have a negative serum pregnancy test at screening and prior to the first dose of conditioning chemotherapy
  • Women of childbearing potential and all male subjects must agree to use highly effective methods of contraception and agree to remain on a highly effective method of contraception from the time of signing the informed consent form until at least 12 months after GLPG5101 infusion. Subjects must agree to not donate eggs or sperm during this period.

Key

Exclusion Criteria
  • Selected prior treatments as defined in the protocol
  • History of another primary malignancy that requires intervention beyond surveillance or that has not been in remission for at least 3 years. (exceptions per protocol)
  • Toxicity from previous anticancer therapy that has not resolved to baseline levels or to ≤ Grade 2
  • Active central nervous system (CNS) involvement (lesion on contrast-enhanced CT/MRI brain, malignant B cells in CSF) by disease under study (exceptions per protocol)
  • Clinically significant cardiac disease
  • Primary immunodeficiency
  • Stroke or seizure within 6 months of screening
  • History of autoimmune disease requiring systemic immunosuppression or disease modifying treatment within 28 days before screening
  • Infection with human immunodeficiency virus (HIV), active hepatitis B or active hepatitis C virus
  • Systemic fungal, bacterial, viral, or other infection that is not controlled

Study & Design

Study Type
INTERVENTIONAL
Study Design
SEQUENTIAL
Arm && Interventions
GroupInterventionDescription
Phase 1 (Dose escalation phase): Dose level 1GLPG5101Participants will receive a single dose of GLPG5101 intravenous (IV) cell suspension for infusion at dose level 1 on Day 0.
Phase 2 (Dose expansion phase): Indolent B-cell NHLGLPG5101Participants with indolent B-cell NHL (FL and MZ) will receive a single dose of GLPG5101 IV cell suspension for infusion at RP2D level on Day 0.
Phase 2 (Dose expansion phase): BLGLPG5101Participants with BL will receive a single dose of GLPG5101 IV cell suspension for infusion at RP2D level on Day 0.
Phase 2 (Dose expansion phase): PCNSLGLPG5101Participants with PCNSL will receive a single dose of GLPG5101 IV cell suspension for infusion at RP2D level on Day 0.
Phase 1 (Dose escalation phase): Dose level 3GLPG5101Participants will receive a single dose of GLPG5101 IV cell suspension for infusion at dose level 3 on Day 0.
Phase 1 (Dose escalation phase): Dose level 2GLPG5101Participants will receive a single dose of GLPG5101 IV cell suspension for infusion at dose level 2 on Day 0.
Phase 2 (Dose expansion phase): DLBCLGLPG5101Participants with DLBCL will receive a single dose of GLPG5101 IV cell suspension for infusion at RP2D level on Day 0.
Phase 2 (Dose expansion phase): High-risk DLBCLGLPG5101Participants with High-risk DLBCL will receive a single dose of GLPG5101 IV cell suspension for infusion at RP2D level on Day 0.
Phase 2 (Dose expansion phase): MCLGLPG5101Participants with MCL will receive a single dose of GLPG5101 IV cell suspension for infusion at RP2D level on Day 0.
Primary Outcome Measures
NameTimeMethod
Phase 1: Number of participants with adverse events (AEs) and serious adverse events (SAEs)2 years
Phase 1: Number of participants with Dose-Limiting Toxicities (DLTs)From first dose up to Day 28
Phase 2: Number of participants with objective response (OR) per the Lugano Classification or International Primary central nervous system lymphoma Collaborative Group (IPCG) criteria for PCNSL2 years

For all cohorts except cohort 6b

Phase 2: Progression-free survival (PFS)2 years

For cohort 6b only

Secondary Outcome Measures
NameTimeMethod
Number of participants without minimal Residual Disease (MRD) at CR (DLBCL, MCL and DLBCL-RT)2 years
Pharmacokinetics (PK): Levels of anti-CD19 CAR T cells in blood at peak and over time2 years
Pharmacodynamics (PD): Levels of chemokines in serum over timeDay 7 before infusion, Day 0, Day 1, Day 4, Day 7, Day 10, Day 14, Day 21, Day 28
PD: Levels of cytokines in serum over timeDay 7 before infusion, Day 0, Day 1, Day 4, Day 7, Day 10, Day 14, Day 21, Day 28
Percentage of successfully manufactured GLPG5101 products within the predefined release specificationsFrom leukapheresis to infusion
Phase 2: Number of participants with AEs and SAEs2 years
Number of participants with AEs of special interests2 years
Number of participants with OR per the Lugano Classification or IPCG criteria2 years

For phase 1 and cohort 6b only

Number of participants with OR per International workshop on Chronic Lymphocytic Leukemia (iwCLL) criteria (DLBCL-RT [cohort 7] only2 years
Number of participants with complete response (CR) per Lugano Classification or IPCG criteria for PCNSL2 years
Duration of response (DOR)2 years
Duration of complete response (DOCR)2 years
Event-free survival (EFS)2 years
Progression-free survival (PFS)2 years
Overall survival (OS)2 years
Phase 2: Change from baseline in measurement of health-related Quality of Life (HRQoL) using the European Organization for Research and Treatment of Cancer (EORTC) QLQ-C30 and its CLL-specific module QLQ-CLL-17 (DLBCL-RT only), and EuroQol EQ-5D-5L2 years

Trial Locations

Locations (9)

Beth Israel Deaconess Medical Center

🇺🇸

Boston, Massachusetts, United States

Tufts Medical Center

🇺🇸

Boston, Massachusetts, United States

Antwerp University Hospital

🇧🇪

Edegem, Belgium

UZ Leuven

🇧🇪

Leuven, Belgium

CHU De Liège

🇧🇪

Liège, Belgium

Cliniques Universitaires Saint-Luc

🇧🇪

Woluwe-Saint-Lambert, Belgium

Academisch Medisch Centrum

🇳🇱

Amsterdam, Netherlands

Leiden University Medical Center

🇳🇱

Leiden, Netherlands

Erasmus Universitair Medisch Centrum Rotterdam (Erasmus MC)

🇳🇱

Rotterdam, Netherlands

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