MedPath

Long-term Efficacy, Safety and Tolerability of Pramipexole in Patients With Idiopathic Moderate to Severe Restless Legs Syndrome (RLS)

Phase 4
Completed
Conditions
Restless Legs Syndrome
Interventions
Drug: Placebo
Registration Number
NCT00472199
Lead Sponsor
Boehringer Ingelheim
Brief Summary

The primary objective of the current study will be the evaluation of long-term efficacy of a 26-weeks treatment with pramipexole in patients with idiopathic moderate to severe Restless Legs Syndrome (RLS) in comparison to placebo.

The key secondary objectives are to assess the effects on clinical global impressions - global improvement (CGI-I) (based on CGI-I responder rate) and on RLS (based on IRLS responder rate) for 26 weeks under pramipexole in comparison to placebo. Further secondary objectives are to investigate the incidence and severity of augmentation and rebound and to assess the effects on patient global impression (PGI) (based on PGI responder rate), on RLS symptoms (based on the RLS-6 scales), on associated mood disturbance (based on item 10 of the IRLS), on pain in limbs (based on a visual analogue scale (VAS)), on quality of life in RLS (based on Johns Hopkins RLS-QoL), on general quality of life Short Form 36 (SF-36) and on safety (based on adverse events (AE) profile) of pramipexole in comparison to placebo.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
331
Inclusion Criteria
  1. Written informed consent consistent with International Conference on Harmonization - Good Clinical Practice (ICH-GCP) and local Institutional Review Board/Independent Ethics Committee (IRB/IEC) requirements obtained prior to any study procedures being performed and the ability and willingness to comply with study treatment regimen and to attend study assessments
  2. Male or female out-patients aged 18-85 years
  3. Diagnosis of idiopathic RLS according to the clinical RLS criteria of the International Restless Legs Syndrome Study Group (IRLSSG) [P03-03355]. All four criteria must be present to fulfil the diagnosis of RLS.
  4. RLS symptoms present at least 2 to 3 days per week during the last 3 months prior to baseline (Visit 2)
  5. IRLS total score >15 at baseline (Visit 2)
Exclusion Criteria
  1. Women of child-bearing potential (i.e. premenopausal women, or postmenopausal women less than 6 months after last menses) who do not use during the clinical trial an adequate method of contraception such as: double barrier protection (e.g. diaphragm or condom and spermicide), intrauterine device, hormonal therapy (oral, injectable, or subcutaneous), or partner's surgical sterilization
  2. Any woman of child-bearing potential not having a negative pregnancy test at screening
  3. Breastfeeding women
  4. Patients with known hypersensitivity to pramipexole or any other component of the investigational product or placebo tablets
  5. Diagnosis of augmentation under previous pharmacological RLS treatment
  6. Concomitant or previous pharmacologic therapy as follows: Any intake of dopamine agonists within 14 days prior to baseline (Visit 2); Any intake of levodopa within 14 days prior to baseline (Visit 2); Unsuccessful prior treatment with non-ergot dopamine agonists (e.g. pramipexole, ropinirole);

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
PlaceboPlacebo4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks.
PramipexolePramipexole4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase or decrease the dose in steps to 0.25 mg, 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks.
Primary Outcome Measures
NameTimeMethod
Change From Baseline in International Restless Legs Syndrome Study Group Rating Scale (IRLS) Total Score After 26 WeeksBaseline and 26 weeks

IRLS total score ranging from 0 (no RLS symptoms) to 40 (very severe RLS symptoms)

Secondary Outcome Measures
NameTimeMethod
Change From Baseline in SF-36 Dimension Social Functioning After 26 WeeksBaseline and 26 weeks

Score ranging from 0 to 100 with higher scores indicating better social functioning

Clinical Global Impression - Global Improvement (CGI-I) Responder Rateafter 26 weeks of treatment

CGI-I scores ranging from '1' (very much improved) to '7' (very much worse), CGI-I responder have scoring 1 or 2 (at least much improved)

International Restless Legs Syndrome (IRLS) Study Group Rating Scale Responder Rateafter 26 weeks of treatment

IRLS response was defined as at least 50% reduction in IRLS total score from baseline. IRLS total score ranging from 0 (no RLS symptoms) to 40 (very severe symptoms)

Patient Global Impression (PGI) Responder Rateafter 26 weeks of treatment

PGI scores ranging from '1' (very much better) to '7' (very much worse), PGI responder have scoring 1 or 2 (at least much better)

Change From Baseline in Restless Legs Syndrome-6 (RLS-6) Score "Satisfaction With Sleep" After 26 Weeksbaseline and 26 weeks of treatment

The score is an 11-point Likert scale, ranging from "none/not at all" (0) to "very severe" (10), to reflect the patient's condition during the previous week

Change From Baseline in RLS-6 Score "Severity Falling Asleep" After 26 WeeksBaseline and 26 weeks of treatment

The score is an 11-point Likert scale, ranging from "none/not at all" (0) to "very severe" (10), to reflect the patient's condition during the previous week

Change From Baseline in RLS-6 Score "Severity During the Night" After 26 Weeksbaseline and 26 weeks of treatment

The question was rated on an 11-point Likert scale, ranging from "none/not at all" (0) to "very severe" (10), to reflect the patient's condition during the previous week

Change From Baseline in RLS-6 Score "Severity During the Day When at Rest" After 26 WeeksBaseline and 26 weeks of treatment

The score is an 11-point Likert scale, ranging from "none/not at all" (0) to "very severe" (10), to reflect the patient's condition during the previous week

Change From Baseline RLS-6 Score "Severity During the Day Engaged in Activities" After 26 WeeksBaseline and 26 weeks of treatment

The score is an 11-point Likert scale, ranging from "none/not at all" (0) to "very severe" (10), to reflect the patient's condition during the previous week

Change From Baseline in RLS-6 Score "Tired or Sleepy During the Day" After 26 WeeksBaseline and 26 weeks of treatment

The score is an 11-point Likert scale, ranging from "none/not at all" (0) to "very severe" (10), to reflect the patient's condition during the previous week

Change From Baseline in IRLS Mood Disturbance Score (Item 10) After 26 WeeksBaseline and 26 weeks of treatment

Mood disturbance associated with RLS symptoms ranging from 0 (none) to 4 (very severe)

Change From Baseline in Visual Analogue Scale (VAS) Score for Pain in Limbs After 26 WeeksBaseline and 26 weeks of treatment

The scale measures pain on a continuous 100 mm axis ranging from no pain (0 mm) to unbearable pain (100 mm)

Change From Baseline in Quality of Life in RLS (RLS QoL) Score After 26 WeeksBaseline and 26 weeks of treatment

RLS QoL total score ranging from 0 to 100 with higher values indicating better quality of life

Change From Baseline in Short Form-36 (SF-36) Dimension Bodily Pain After 26 WeeksBaseline and 26 weeks

Score ranging from 0 to 100 with higher scores indicating less bodily pain

Change From Baseline in SF-36 Dimension General Health After 26 WeeksBaseline and 26 weeks

Score ranging from 0 to 100 with higher scores indicating better health status

Change From Baseline in SF-36 Dimension Mental Health After 26 WeeksBaseline and 26 weeks

Score ranging from 0 to 100 with higher scores indicating better mental health

Change From Baseline in SF-36 Dimension Physical Functioning After 26 WeeksBaseline and 26 weeks

Score ranging from 0 to 100 with higher scores indicating better physical functioning

Change From Baseline in SF-36 Dimension Role Limitations Due to Emotional Problems After 26 WeeksBaseline and 26 weeks

Score ranging from 0 to 100 with higher scores indicating less limitations due to emotional problems

Change From Baseline in SF-36 Dimension Role Limitations Due to Physical Problems After 26 WeeksBaseline and 26 weeks

Score ranging from 0 to 100 with higher scores indicating less limitations due to physical problems

Change From Baseline in SF-36 Dimension Vitality After 26 WeeksBaseline and 26 weeks

Score ranging from 0 to 100 with higher scores indicating better vitality

Change From Baseline in SF-36 Dimension Mental Component Summary After 26 WeeksBaseline and 26 weeks

Score ranging from 0 to 100 with higher scores indicating better health

Change From Baseline in SF-36 Dimension Physical Component Summary After 26 WeeksBaseline and 26 weeks

Score ranging from 0 to 100 with higher scores indicating better health

Diagnosis of Classified Augmentation According to Independent Expert Panelafter at least 4 weeks of treatment

Augmentation is a worsening of RLS symptoms and may manifest as increased severity and the involvement of other extremities or as a shift of RLS symptoms to a time period that is 2 or more hours earlier than was typical of the time of symptom onset during the initial course of beneficial stable treatment or the state before recently starting treatment.

Worsening of RLS Symptoms (by at Least 4 Points in the IRLS Total Score Compared to Baseline) After Treatment Discontinuationafter at least 1 week of treatment discontinuation

Worsening of RLS symptoms, in comparison to baseline, following abrupt treatment discontinuation (for patients with no added RLS therapy after study drug discontinuation).

Assessment of worsening of RLS was based on the IRLS total score assessed 7 ± 1 days after treatment discontinuation (the end of the study or premature discontinuation) compared with that at baseline. Analysis considered the number of patients experiencing a clinically relevant deterioration of ≥4 points in total IRLS score 7 ± 1 days after discontinuation of trial medication compared with baseline.

Baseline, Week 26 Mean Supine Systolic Blood PressureBaseline, Week 26
Baseline, Week 26 Mean Standing Systolic Blood PressureBaseline, Week 26
Baseline, Week 26 Mean Supine Diastolic Blood PressureBaseline, Week 26
Baseline, Week 26 Mean Standing Diastolic Blood PressureBaseline, Week 26
Baseline, Week 26 Mean Standing Pulse RateBaseline, Week 26
Baseline, Week 26 Mean Supine Pulse RateBaseline, Week 26

Trial Locations

Locations (42)

248.629.44003 Boehringer Ingelheim Investigational Site

🇬🇧

Chorley, United Kingdom

248.629.3402 Boehringer Ingelheim Investigational Site

🇪🇸

Barcelona, Spain

248.629.44004 Boehringer Ingelheim Investigational Site

🇬🇧

Glasgow, United Kingdom

248.629.4906 Boehringer Ingelheim Investigational Site

🇩🇪

Herborn, Germany

248.629.35303 Boehringer Ingelheim Investigational Site

🇮🇪

Co. Tipperary, Ireland

248.629.4904 Boehringer Ingelheim Investigational Site

🇩🇪

Berlin (Hellersdorf), Germany

248.629.3405 Boehringer Ingelheim Investigational Site

🇪🇸

Granada, Spain

248.629.3403 Boehringer Ingelheim Investigational Site

🇪🇸

San Sebastián, Spain

248.629.4304 Boehringer Ingelheim Investigational Site

🇦🇹

Linz, Austria

248.629.44001 Boehringer Ingelheim Investigational Site

🇬🇧

Manchester, United Kingdom

248.629.4302 Boehringer Ingelheim Investigational Site

🇦🇹

Innsbruck, Austria

248.629.35801 Boehringer Ingelheim Investigational Site

🇫🇮

Espoo, Finland

248.629.35805 Boehringer Ingelheim Investigational Site

🇫🇮

Helsinki, Finland

248.629.35804 Boehringer Ingelheim Investigational Site

🇫🇮

Joensuu, Finland

248.629.35802 Boehringer Ingelheim Investigational Site

🇫🇮

Oulu, Finland

248.629.4903 Boehringer Ingelheim Investigational Site

🇩🇪

Berlin-Steglitz, Germany

248.629.4902 Boehringer Ingelheim Investigational Site

🇩🇪

Berlin, Germany

248.629.4908 Boehringer Ingelheim Investigational Site

🇩🇪

Bochum, Germany

248.629.4901 Boehringer Ingelheim Investigational Site

🇩🇪

Ellwangen, Germany

248.629.35301 Boehringer Ingelheim Investigational Site

🇮🇪

Carrigtwohill, Ireland

248.629.31001 Boehringer Ingelheim Investigational Site

🇳🇱

Bennebroek, Netherlands

248.629.4204 Boehringer Ingelheim Investigational Site

🇸🇰

Bratislava, Slovakia

248.629.4202 Boehringer Ingelheim Investigational Site

🇸🇰

Brezno, Slovakia

248.629.3401 Boehringer Ingelheim Investigational Site

🇪🇸

Madrid, Spain

248.629.3406 Hospital Arnau de Vilanova

🇪🇸

Valencia, Spain

248.629.44006 Boehringer Ingelheim Investigational Site

🇬🇧

Edgbaston, Birmingham, United Kingdom

248.629.44002 Boehringer Ingelheim Investigational Site

🇬🇧

Reading, United Kingdom

248.629.44005 Boehringer Ingelheim Investigational Site

🇬🇧

Waterloo, Liverpool, United Kingdom

248.629.4905 Boehringer Ingelheim Investigational Site

🇩🇪

Leipzig, Germany

248.629.4909 Boehringer Ingelheim Investigational Site

🇩🇪

Schwerin, Germany

248.629.4907 Boehringer Ingelheim Investigational Site

🇩🇪

Würzburg, Germany

248.629.31005 Boehringer Ingelheim Investigational Site

🇳🇱

Hoogwoud, Netherlands

248.629.31003 Boehringer Ingelheim Investigational Site

🇳🇱

Oude Pekela, Netherlands

248.629.4205 Boehringer Ingelheim Investigational Site

🇸🇰

Bratislava, Slovakia

248.629.31002 Boehringer Ingelheim Investigational Site

🇳🇱

Oude Pekela, Netherlands

248.629.35302 Boehringer Ingelheim Investigational Site

🇮🇪

Co. Kildare, Ireland

248.629.4201 Boehringer Ingelheim Investigational Site

🇸🇰

Kosice, Slovakia

248.629.4203 Boehringer Ingelheim Investigational Site

🇸🇰

Martin, Slovakia

248.629.3201 Boehringer Ingelheim Investigational Site

🇧🇪

Edegem, Belgium

248.629.35806 Boehringer Ingelheim Investigational Site

🇫🇮

Tampere, Finland

248.629.31006 Boehringer Ingelheim Investigational Site

🇳🇱

Musselkanaal, Netherlands

248.629.31004 Boehringer Ingelheim Investigational Site

🇳🇱

Rijswijk, Netherlands

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