MedPath

Dose Finding Study of CHF 4226 for Treating Patients With COPD

Phase 2
Completed
Conditions
Chronic Obstructive Pulmonary Disease
Interventions
Registration Number
NCT00605891
Lead Sponsor
Chiesi Farmaceutici S.p.A.
Brief Summary

The purpose of this study is to identify the optimal once-daily dose of CHF 4226 to be further developed for the treatment of patients with COPD.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
278
Inclusion Criteria
  • Patient has signed an IRB-/Ethics Committee-approved Informed Consent form

  • Patient is a male or non-pregnant female between the ages of 40 - 75 years, inclusive

  • Patient has a current or past smoking history of at least 15 pack-years

  • Patient has a clinical diagnosis of COPD in accordance with the recommendations of the National Heart Lung and Blood Institute/World Health Organization (NHLBI/WHO) Global Initiative for Chronic Obstructive Lung Disease (GOLD)

  • Patient meets the following requirements after an FEV1 albuterol reversibility test (i.e., 30 minutes following 200 mcg (metered dose) albuterol/salbutamol pMDI):

  • FEV1 is at least 0.9L

  • FEV1 of 40% - 70%, inclusive, of patient's predicted normal value

  • Change in FEV1 > 4% of patient's predicted normal value

    • If change in FEV1 < 4% of patient's predicted normal value, then this requirement must be met after retesting during the run-in period, at least 24 hours prior to Day -1
  • FEV1/FVC < 70%

Exclusion Criteria
  • Patient has a history of asthma, allergic rhinitis, or atopy
  • Patient has a blood eosinophil count > 500/microliter
  • Patient had a COPD exacerbation or a lower respiratory tract infection within 8 weeks prior to screening, or during the run-in period, that resulted in the use of an antibiotic, or oral or parenteral corticosteroids
  • Patient is on an inhaled corticosteroid that has been initiated, or the effective dose has been changed, within 4 weeks prior to screening or during the run-in period
  • Patient has an uncontrolled cardiovascular (e.g., uncontrolled hypertension), respiratory, hematologic, immunologic, renal, neurologic, hepatic, endocrine (e.g., uncontrolled diabetes mellitus) or other disease, or any condition that might, in the judgment of the Investigator, place the patient at undue risk or potentially compromise the results or interpretation of the study
  • Patient has a history of coronary artery disease, cerebrovascular disease, cardiac arrhythmias
  • Patient has a concomitant disease of poor prognosis (e.g., cancer)
  • Patient has a serum potassium value ≤ 3.5 mEq/L or >5.5mEq/L and/or a fasting serum glucose value ≥ 140 mg/dL
  • Patient has an abnormal QTc Fridericia interval value in the Screening visit ECG test (i.e., > 450 msec in males or > 470 msec in females)
  • Patient has developed Cor Pulmonale
  • Patient is receiving long term oxygen therapy, i.e., ≥ 16 hours/24-hour period, every day
  • Patient has a known intolerance/hypersensitivity to Beta2-adrenergic agonists, propellant gases/excipients
  • Patient is receiving treatment with a tricyclic antidepressant or a monoamine oxidase inhibitor (MAOI)
  • Patient has received a live-attenuated virus vaccination within two weeks prior to screening or during the run-in
  • Patient is pregnant or lactating female, or female at risk of pregnancy (i.e., not using an adequate contraceptive method)
  • Patient is mentally or legally incapacitated
  • Patient has participated in another investigational study within 30 days prior to screening
  • Patient abuses alcohol or other substances
  • Patient is potentially non-compliant or unable to perform required outcome measurements of the protocol

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Ccarmoterol (CHF 4226)carmoterol (CHF 4226) 4.0 μg once a day, in the morning
Acarmoterol (CHF 4226)carmoterol (CHF 4226) 1.0 μg once a day, in the morning
Bcarmoterol (CHF 4226)carmoterol (CHF 4226) 2.0 μg once a day, in the morning
DplaceboPlacebo once a day, in the morning
EsalmeterolSalmeterol 50 μg BID, in the morning and in the evening
Primary Outcome Measures
NameTimeMethod
Change in FEV1Day 1 to Day 14 (+3 days)
Secondary Outcome Measures
NameTimeMethod
FEV110 and 30 min, 1, 2, and 3 hrs post dose on Day 1, Day 2 and Day 14 (+3)
ECG/QTcpre dose and post dose at 30' on Days 1, 2 and 14 (+3)
Fasting serum potassiumpre dose and post dose at 30' on Days 1, 2 and 14 (+3)
Fasting glucosepre dose and post dose at 30' on Days 1, 2 and 14 (+3)
Change in FEV110 and 30 min, 1, 2, and 3 hrs post dose on Day 1, Day 2 and Day 14 (+3)

Trial Locations

Locations (50)

Ordinace pro nemoci dychaciho ustroji

🇨🇿

Beroun, Czech Republic

University Clinical Research - DeLand, LLC

🇺🇸

DeLand, Florida, United States

NZOZ Non-nocere

🇵🇱

Gdansk, Poland

Klinika Pulmonologii i Alergologii

🇵🇱

Lodz, Poland

Spitalul Clinic Judetean de Urgenta Brasov

🇷🇴

Brasov, Romania

Spitalul Clinic "Sf. Maria"

🇷🇴

Bucharest, Romania

Spitalul Clinic de Urgenta Militar Central "Davila"

🇷🇴

Bucharest, Romania

UCSD - Clinical Trials Center

🇺🇸

San Diego, California, United States

The University of Texas Health Center at Tyler

🇺🇸

Tyler, Texas, United States

University of Wisconsin-Allergy/Asthma

🇺🇸

Madison, Wisconsin, United States

Plicni ambulance Rokycany

🇨🇿

Rokycany, Czech Republic

Plicni ambulance

🇨🇿

Praha 3 - Zizkov, Czech Republic

Nemocnice Na Homolce Plicni ambulance

🇨🇿

Praha 5, Czech Republic

Medars GmbH

🇩🇪

Berlin, Germany

Clopton Clinic

🇺🇸

Jonesboro, Arkansas, United States

ABM Research Center

🇺🇸

Fresno, California, United States

Institute of Healthcare Assessment Inc.

🇺🇸

San Diego, California, United States

Clinical Research of West Florida

🇺🇸

Clearwater, Florida, United States

Carolina Pharmaceutical Research

🇺🇸

Statesville, North Carolina, United States

New Horizons Clinical Research

🇺🇸

Cincinnati, Ohio, United States

Clinical Research Institute of Southern Oregon PC

🇺🇸

Medford, Oregon, United States

Lowcountry Lung and Critical Care, PA

🇺🇸

North Charleston, South Carolina, United States

National Jewish Medical and Research Center

🇺🇸

Denver, Colorado, United States

Clinical Research of West Florida, Inc.

🇺🇸

Tampa, Florida, United States

OTRAN

🇨🇿

Kutna Hora, Czech Republic

Plicni a alergologicka ambulance

🇨🇿

Kutna Hora, Czech Republic

Pneumolog, internista

🇨🇿

Lovosice, Czech Republic

Palm Beach Research Center

🇺🇸

West Palm Beach, Florida, United States

Delaware Valley Clinical Research

🇺🇸

Cherry Hill, New Jersey, United States

Toledo Center for Clinical Research

🇺🇸

Sylvania, Ohio, United States

Edward Hospital and Helath Services, Center for Clinical Trials

🇺🇸

Naperville, Illinois, United States

Community Clinical Research Center

🇺🇸

Anderson, Indiana, United States

ClinSite

🇺🇸

Canton, Michigan, United States

Pulmonary Consultants - Research Department

🇺🇸

Medford, Oregon, United States

Amarillo Center for Clinical Research, Ltd.

🇺🇸

Amarillo, Texas, United States

Lungenzentrum Geesthacht

🇩🇪

Geesthacht, Germany

Pneumologisches Forschungsinstitut GmbH

🇩🇪

Grosshansdorf, Germany

Pneumologisches Forschungsinstitut Niederlassung Hamburg

🇩🇪

Hamburg, Germany

Robert-Koch-Klinik

🇩🇪

Leipzig, Germany

SMO, MD GmbH

🇩🇪

Magdeburg, Germany

IFG GmbH

🇩🇪

Ruedersdorf, Germany

Medcare Specjalistyczna Opieka Medyczna NZOZ

🇵🇱

Gdansk, Poland

SPZOZ w Proszowicach Oddzial Chorob Pluc

🇵🇱

Proszowice, Poland

Spitalul de Urgenta "Prof. Dr. Dimitrie Gerota"

🇷🇴

Bucharest, Romania

Institutul National de Pneumoftisiologie "M. Nasta"

🇷🇴

Bucharest, Romania

Spitalul de Pneumoftiziologie Constanta

🇷🇴

Constanta, Romania

UCT Lung Institute

🇿🇦

Mowbray, Cape Town, South Africa

Tiervlei Trial Center, Karl Bremer Hospital

🇿🇦

Bellville, South Africa

ClinSite, LLC

🇺🇸

Ann Arbor, Michigan, United States

Breath of Life Research Institute

🇺🇸

Katy, Texas, United States

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