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A Study Evaluating the Efficacy and Safety of Afimetoran Compared With Placebo in Participants With Active Systemic Lupus Erythematosus (SLE)

Phase 2
Recruiting
Conditions
Systemic Lupus Erythematosus
Interventions
Other: Placebo
Registration Number
NCT04895696
Lead Sponsor
Bristol-Myers Squibb
Brief Summary

The purpose of this study is to evaluate the effectiveness, safety and tolerability of Afimetoran in participants with active Systemic Lupus Erythematosus (SLE). The extension period will provide additional long-term safety and efficacy data and enable those participants initially randomized to placebo to receive treatment with Afimetoran.

Detailed Description

Not available

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
268
Inclusion Criteria
  • Diagnosed ≥ 12 weeks before the screening visit and qualify as having SLE according to the SLE International Collaborating Clinics (SLICC) Classification Criteria at the screening visit
  • Test positive, as determined by the central laboratory, for at least one of the following lupus related autoantibodies at the time of screening: antinuclear antibody ≥ 1:80, anti-double-stranded deoxyribonucleic acid (dsDNA) antibody, or anti-Smith antibody.
  • Have a total Hybrid Systemic Lupus Erythematosus Disease Activity Index (SLEDAI) score ≥ 6 points and clinical Hybrid SLEDAI score ≥ 4 points with joint involvement and/or rash
Exclusion Criteria
  • Active severe lupus nephritis (LN) as assessed by the investigator
  • Active or unstable neuropsychiatric lupus manifestations defined by the Hybrid SLEDAI
  • Diagnosis of Mixed Connective Tissue Disease for which the predominant diagnosis is not SLE
  • Antiphospholipid Syndrome

Other protocol-defined inclusion/exclusion criteria apply

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Afimetoran: Dose 1Afimetoran-
PlaceboPlacebo-
Afimetoran: Dose 2Afimetoran-
Afimetoran: Dose 3Afimetoran-
Primary Outcome Measures
NameTimeMethod
Proportion of participants that achieve an SLE (Systemic Lupus Erythematosus) Responder Index (4) (SRI(4)) response at Week 48Up to 48 Weeks
Secondary Outcome Measures
NameTimeMethod
Proportion of participants who achieve a Lupus Low Disease Activity State (LLDAS) response at Week 24 and Week 48Up to 48 Weeks
Mean change from baseline in swollen joint count using the 28-joint count at Week 24 and Week 48 in participants with ≥ 2 swollen joints at baselineUp to 48 Weeks
Change from baseline in PGA score of disease activity at Week 24 and Week 48Up to 48 Weeks

PGA = Physician Global Assessment of disease activity (score of "0" indicating no disease activity and higher scores indicating higher disease activity)

Proportion of participants who achieve CS reduction or maintenance to ≤ 7.5 mg per day at Week 48Up to 48 Weeks
Number of participants with Adverse Events (AEs)Up to 100 Weeks
Number of participants with physical examination abnormalitiesUp to 100 Weeks
Number of participants with electrocardiogram (ECG) abnormalitiesUp to 52 Weeks
Proportion of participants who achieve an SRI(4) response at Week 24Up to 24 Weeks
Proportion of participants with a Cutaneous Lupus Erythematosus Disease Area and Severity Index; Activity (CLASI-A) score ≥ 10 at baseline who achieve a decrease of ≥ 50% from baseline CLASI-A score (CLASI-50) response at Week 24 and Week 48Up to 48 Weeks
Proportion of participants with 6 or more swollen joints and 6 or more tender joints at baseline who achieve a ≥ 50% reduction from baseline in both swollen and tender joints at Week 24 and Week 48Up to 48 Weeks
Mean change from baseline in tender joint count at Week 24 and Week 48 using the 28- joint count in participants with ≥ 2 tender joints at baselineUp to 48 Weeks
Change in participant reported disease activity from baseline to Week 24 and Week 48 according to the 36-item Short Form Health Questionnaire (SF-36)Up to 48 Weeks

The SF-36 was designed as an indicator of health status in population surveys, and health policy evaluations, and for use as an outcome measure in clinical practice and research. Scores for each domain range from 0 to 100, with high scores indicating a better health status.

Number of participants with Serious Adverse Events (SAEs)Up to 100 Weeks
Proportion of participants that achieve a British Isles Lupus Assessment Group (BILAG)-based Combine Lupus Assessment (BICLA) response at Week 24 and Week 48Up to 48 Weeks
Number of participants with clinical laboratory abnormalitiesUp to 100 Weeks
Number of participants with vital sign abnormalitiesUp to 100 Weeks

Trial Locations

Locations (174)

Local Institution - 0196

🇨🇳

Baoding, Hebei, China

Private Practice - Dr. Jefrey Lieberman

🇺🇸

Decatur, Georgia, United States

Local Institution - 0100

🇺🇸

Birmingham, Alabama, United States

St Joseph Heritage Healthcare-Rheumatology

🇺🇸

Fullerton, California, United States

Christine Thai, MD

🇺🇸

Huntington Beach, California, United States

UCSD - Altman Clinical and Translational Research Institute (ACTRI)

🇺🇸

La Jolla, California, United States

Advanced Medical Research - La Palma

🇺🇸

La Palma, California, United States

Local Institution - 0202

🇺🇸

Los Angeles, California, United States

Rheumatology Center of San Diego

🇺🇸

San Diego, California, United States

Private Practice - Dr. Nazanin Firooz

🇺🇸

West Hills, California, United States

Local Institution - 0164

🇺🇸

Woodland Hills, California, United States

Colorado Arthritis Associates

🇺🇸

Denver, Colorado, United States

UConn Health

🇺🇸

Farmington, Connecticut, United States

Bay Area Arthritis and Osteoporosis

🇺🇸

Brandon, Florida, United States

Clinical Research of West Florida, Inc. (Clearwater)

🇺🇸

Clearwater, Florida, United States

University Of Florida

🇺🇸

Gainesville, Florida, United States

Vida Clinical Research

🇺🇸

Kissimmee, Florida, United States

Omega Research MetroWest

🇺🇸

Orlando, Florida, United States

Millennium Research

🇺🇸

Ormond Beach, Florida, United States

IRIS Research and Development, LLC

🇺🇸

Plantation, Florida, United States

Local Institution - 0137

🇺🇸

South Miami, Florida, United States

West Broward Rheumatology Associates

🇺🇸

Tamarac, Florida, United States

Piedmont West

🇺🇸

Atlanta, Georgia, United States

North Georgia Rheumatology

🇺🇸

Suwanee, Georgia, United States

Greater Chicago Specialty Physicians - Orland Park

🇺🇸

Orland Park, Illinois, United States

Western KY Rheumatology

🇺🇸

Hopkinsville, Kentucky, United States

Local Institution - 0171

🇺🇸

Baton Rouge, Louisiana, United States

Local Institution - 0134

🇺🇸

Wheaton, Maryland, United States

Local Institution - 0221

🇺🇸

Rochester Hills, Michigan, United States

Saint Paul Rheumatology

🇺🇸

Eagan, Minnesota, United States

Washington University/ Barnes Jewish Hospital

🇺🇸

Saint Louis, Missouri, United States

Local Institution - 0165

🇺🇸

Saint Louis, Missouri, United States

Local Institution - 0091

🇺🇸

Las Vegas, Nevada, United States

Sahni Rheumatology & Therapy

🇺🇸

West Long Branch, New Jersey, United States

Local Institution - 0132

🇺🇸

Bronx, New York, United States

The Feinstein Institute for Medical Research

🇺🇸

Manhasset, New York, United States

Local Institution - 0203

🇺🇸

Charlotte, North Carolina, United States

DJL Clinical Research, PLLC

🇺🇸

Charlotte, North Carolina, United States

The Ohio State University Wexner Medical Center (OSUWMC) - CarePoint East-Rheumatology and Immunolog

🇺🇸

Columbus, Ohio, United States

Paramount Medical Research and Consulting, Llc

🇺🇸

Middleburg Heights, Ohio, United States

Oklahoma Medical Research Foundation-Multiple Sclerosis Center of Excellence

🇺🇸

Oklahoma City, Oklahoma, United States

Oklahoma Medical Research Foundation

🇺🇸

Oklahoma City, Oklahoma, United States

Shelby Research LLC

🇺🇸

Memphis, Tennessee, United States

Arthritis and Rheumatology Research Institute

🇺🇸

Allen, Texas, United States

Local Institution - 0152

🇺🇸

Allen, Texas, United States

Amarillo Center for Clinical Research-Research

🇺🇸

Amarillo, Texas, United States

Local Institution - 0029

🇺🇸

Mesquite, Texas, United States

Overlake Arthritis and Osteoporosis Center

🇺🇸

Bellevue, Washington, United States

Sun Research Institute

🇺🇸

San Antonio, Texas, United States

Local Institution - 0130

🇦🇷

Quilmes, Buenos Aires, Argentina

Local Institution - 0195

🇦🇷

San Fernando, Buenos Aires, Argentina

Local Institution - 0024

🇦🇷

San Isidro, Buenos Aires, Argentina

Local Institution - 0025

🇦🇷

Córdoba, Cordoba, Argentina

Local Institution - 0074

🇦🇷

Buenos Aires, Distrito Federal, Argentina

Local Institution - 0145

🇦🇷

Caba, Distrito Federal, Argentina

Local Institution - 0041

🇦🇷

San Juan, Argentina

Local Institution - 0040

🇦🇷

Caba, Distrito Federal, Argentina

Local Institution - 0027

🇦🇷

San Miguel de Tucumán, Tucuman, Argentina

Local Institution - 0207

🇦🇷

Buenos Aires, Argentina

Local Institution - 0128

🇦🇷

Buenos Aires, Argentina

Local Institution - 0063

🇦🇺

Botany, New South Wales, Australia

Local Institution - 0072

🇦🇺

Westmead, New South Wales, Australia

Local Institution - 0066

🇦🇺

Maroochydore, Queensland, Australia

Local Institution - 0065

🇦🇺

Woodville, South Australia, Australia

Local Institution - 0062

🇦🇺

Camberwell, Victoria, Australia

Local Institution - 0064

🇦🇺

Ivanhoe, Victoria, Australia

Serviços Especializados em Reumatologia

🇧🇷

Salvador, Bahia, Brazil

Centro de Pesquisas da Clínica IBIS

🇧🇷

Salvador, Bahia, Brazil

IPC-MT Instituto de Pesquisas Clínicas de Mato Grosso

🇧🇷

Cuiabá, Mato Grosso, Brazil

Cmip-Centro Mineiro de Pesquisa

🇧🇷

Juiz de Fora, Minas Gerais, Brazil

Centro de Estudos em Terapias Inovadoras-Rheumatology

🇧🇷

Curitiba, Parana, Brazil

LMK Serviços Médicos S/S-Reumacenter

🇧🇷

Porto Alegre, RIO Grande DO SUL, Brazil

Centro Multidisciplinar de Estudos Clinicos

🇧🇷

São Bernardo do Campo, SAO Paulo, Brazil

Local Institution - 0013

🇧🇷

São Paulo, SAO Paulo, Brazil

Fundação Faculdade Regional de Medicina de São José do Rio Preto

🇧🇷

São José do Rio Preto, São Paulo, Brazil

CEPIC - Centro Paulista de Investigação Clínica

🇧🇷

São Paulo, Brazil

Local Institution - 0127

🇨🇱

Osorno, LOS Lagos, Chile

Local Institution - 0143

🇨🇱

Valdivia, Los Rios, Chile

Local Institution - 0073

🇨🇱

Santiago, Metropolitana, Chile

Local Institution - 0043

🇨🇱

Santiago, Metropolitana, Chile

Local Institution - 0075

🇨🇱

Providencia, Región Metropolitana De Santiago, Chile

China-Japan Friendship Hospital

🇨🇳

Beijing, Beijing, China

Peking University Shougang Hospital

🇨🇳

Beijing, Beijing, China

The Seventh Affiliated Hospital, Sun Yat-sen University

🇨🇳

Shenzhen, Guangdong, China

Nanjing Drum Tower Hospital The Affiliated Hospital of Nanjing University Medical School

🇨🇳

Nanjing, Jiangsu, China

Jiangsu Province Hospital

🇨🇳

Nanjing, Jiangsu, China

The First Affiliated Hospital of Soochow University

🇨🇳

Suzhou, Jiangsu, China

The First Hospital of Jilin University

🇨🇳

Changchun, Jilin, China

The 2nd Affiliated Hospital of Dalian Medical University

🇨🇳

Dalian, Liaoning, China

Qilu Hospital of Shandong University (Qingdao)

🇨🇳

Jinan, Shandong, China

Jining No.1 People's Hospital

🇨🇳

Jining, Shandong, China

Local Institution - 0194

🇨🇳

Changzhi, Shanxi, China

Local Institution - 0181

🇨🇳

Kunming, Yunnan, China

Local Institution - 0191

🇨🇳

Beijing, China

Salud SURA Industriales

🇨🇴

Medellín, Antioquia, Colombia

Local Institution - 0185

🇨🇴

Cali, Valle Del Cauca, Colombia

Centro de Reumatologia y Ortopedia

🇨🇴

Barranquilla, Colombia

Centro de Investigacion en Reumatologia y Especialidades Medicas S.A.S

🇨🇴

Bogotá, Colombia

Centro de Estudios de Reumatología y Dermatología SAS

🇨🇴

Cali, Colombia

Preventive Care

🇨🇴

Chía, Colombia

Healthy Medical Center S.A.S

🇨🇴

Zipaquira, Colombia

CHU Bordeaux Haut-Leveque

🇫🇷

Pessac, Aquitaine, France

CHRU de Brest

🇫🇷

Brest, Finistère, France

Bordeaux University Hospital - Pellegrin-Rhumatologie

🇫🇷

Bordeaux, France

Centre Hospitalier Universitaire de Caen Normandie

🇫🇷

Caen, France

Chru De Lille

🇫🇷

Lille Cedex, France

Hôpital Européen Marseille-Service de recherche clinique

🇫🇷

Marseille, France

CHU Strasbourg-Hautepierre-Service de Rhumatologie

🇫🇷

Strasbourg, France

Local Institution - 0087

🇩🇪

Köln, Nordrhein-Westfalen, Germany

Charité Research Organisation

🇩🇪

Berlin, Germany

Local Institution - 0086

🇩🇪

Essen, Germany

Klinikum Der Albrecht-Ludwigs-Universitat

🇩🇪

Freiburg, Germany

All India Institute of Medical Sciences

🇮🇳

New Delhi, Delhi, India

Amber Clinic

🇮🇳

Ahmedabad, Gujarat, India

Medanta The Medicity

🇮🇳

Gurugram, Haryana, India

ChanRe Rheumatology And Immunology Center And Research

🇮🇳

Bengaluru, Karnataka, India

Krishna Institute of Medical Science

🇮🇳

Secunderabad, Telangana, India

Local Institution - 0119

🇮🇪

Manorhamilton, Leitrim, Ireland

Local Institution - 0106

🇮🇪

Dublin, Ireland

Local Institution - 0107

🇮🇪

Galway, Ireland

University of Fukui Hospital

🇯🇵

Eiheiji-cho,Yoshida-gun, Fukui, Japan

University of Occupational and Enviromental Health

🇯🇵

Kitakyushu, Fukuoka, Japan

Hokkaido University Hospital

🇯🇵

Sapporo, Hokkaido, Japan

Kanazawa University Hospital

🇯🇵

Kanazawa, Ishikawa, Japan

Tohoku University Hospital-Department of Rheumatology

🇯🇵

Sendai-shi, Miyagi, Japan

Juntendo University Hospital

🇯🇵

Bunkyo-ku, Tokyo, Japan

Tokyo Metropolitan Tama Medical Center

🇯🇵

Fuchu, Tokyo, Japan

Nihon University Itabashi Hospital

🇯🇵

Itabashiku, Tokyo, Japan

Toho University Ohashi Medical Center

🇯🇵

Meguro-ku, Tokyo, Japan

Keio university hospital-Division of Rheumatology, Department of Internal Medicine

🇯🇵

Shinjuku-ku, Tokyo, Japan

National Center for Global Health and Medicine

🇯🇵

Shinjuku-ku, Tokyo, Japan

Koujunkai Daido Clinic

🇯🇵

Aichi, Japan

National Hospital Organization Chibahigashi National Hospital

🇯🇵

Chiba, Japan

Fukushima Medical University

🇯🇵

Fukushima, Japan

St. Luke's International Hospital

🇯🇵

Tokyo, Japan

The University Of Tokyo Hospital

🇯🇵

Tokyo, Japan

Local Institution - 0060

🇲🇽

Mexico City, Distrito Federal, Mexico

Local Institution - 0018

🇲🇽

Mexico City, Distrito Federal, Mexico

Local Institution - 0182

🇲🇽

Mexico City, Distrito Federal, Mexico

Local Institution - 0020

🇲🇽

Leon, Guanajuato, Mexico

Local Institution - 0017

🇲🇽

Guadalajara, Jalisco, Mexico

Local Institution - 0022

🇲🇽

Zapopan, Jalisco, Mexico

Local Institution - 0071

🇲🇽

Monterrey, Nuevo LEON, Mexico

Local Institution - 0021

🇲🇽

Chihuahua, Mexico

Local Institution - 0061

🇲🇽

Merida, Mexico

Local Institution - 0158

🇲🇽

Mexico City, Mexico

Centrum Medyczne Reuma Park

🇵🇱

Warszawa, Mazowieckie, Poland

Local Institution - 0161

🇵🇱

Łomża, Podlaskie, Poland

Local Institution - 0051

🇵🇱

Bydgoszcz, Poland

Medyczne Centrum Hetmańska

🇵🇱

Poznan, Poland

Local Institution - 0142

🇵🇱

Rzeszów, Poland

Local Institution - 0050

🇵🇱

Sosnowiec, Poland

MICS Centrum Medyczne Warszawa

🇵🇱

Warszawa, Poland

Uniwersytecki Szpital Kliniczny-Klinika Reumatologii i Chorób Wewnętrznych

🇵🇱

Wrocław, Poland

GCM Medical Group, PSC - Hato Rey Site-Hato Rey

🇵🇷

San Juan, Puerto Rico

Local Institution - 0131

🇵🇷

San Juan, Puerto Rico

Sc Medaudio-Optica Srl

🇷🇴

Râmnicu Vâlcea, Vâlcea, Romania

Hightech Medical Services SRL-Centrul pentru Studiul Metabolismului

🇷🇴

Bucharest, Romania

Spital Clinic Sf. Maria

🇷🇴

Bucharest, Romania

Centrul de Kinetoterapie si Masaj Banat SRL

🇷🇴

Giroc, Romania

Local Institution - 0206

🇪🇸

Santander, Cantabria, Spain

CHUAC-Complejo Hospitalario Universitario A Coruña-Reumatologia

🇪🇸

A Coruña, Spain

Hospital Universitari Vall d'Hebron-Rheumatology

🇪🇸

Barcelona, Spain

HOSPITAL GENERAL UNIVERSITARIO GREGORIO MARAÑON-Reumatología

🇪🇸

Madrid, Spain

Hospital Universitario Virgen de Valme-RHEUMATOLOGY

🇪🇸

Sevilla, Spain

Chang Gung Memorial Hospital at Kaohsiung-Rheumatology

🇨🇳

Kaohsiung Niao Sung Dist, Taiwan

China Medical University Hospital

🇨🇳

Taichung, Taiwan

Taichung Veterans General Hospital

🇨🇳

Taichung, Taiwan

National Taiwan University Hospital-Immunology

🇨🇳

Taipei, Taiwan

Taipei Veterans General Hospital

🇨🇳

Taipei, Taiwan

Addenbrooke's Hospital

🇬🇧

Cambridge, Cambridgeshire, United Kingdom

Local Institution - 0110

🇬🇧

Bradford, United Kingdom

Local Institution - 0120

🇬🇧

Edinburgh, United Kingdom

Local Institution - 0125

🇬🇧

Manchester, United Kingdom

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