MedPath

Safety Study of a Long-Acting Injectable Steroid to Treat Knee Osteoarthritis

Phase 1
Completed
Conditions
Osteoarthritis, Knee
Interventions
Drug: Vehicle
Registration Number
NCT02609126
Lead Sponsor
Eupraxia Pharmaceuticals Inc.
Brief Summary

The main purpose of this study is to understand the pharmacokinetics of EP-104IAR and to determine whether it is safe to use in patients with osteoarthritis (OA) of the knee. The study will also provide some preliminary insights into whether the experimental treatment reduces pain in the knee.

Osteoarthritis is the most common joint disease, affecting over 20 million people in the US alone. Currently, pain treatments that are injected directly into the knee often work for only a short time and may also have side effects within the rest of the body. The experimental treatment is a steroid that is in the same family of drugs as the most common current injectable treatments for knee osteoarthritis. For this study, the drug is coated with a polymer intended to prolong the time it stays inside the knee and lessen potential side effects.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
32
Inclusion Criteria
  • OA of Index Knee
  • Kellgren Lawrence Grade 2 or 3
  • Patient-reported pain (PtPain) of Index Knee ≥4 but ≤9
  • PtPain of non-Index Knee <6
  • BMI ≦ 40 kg/m2
Exclusion Criteria
  • Intra-articular joint injection in the Index Knee within the past 8 weeks for glucocorticoids and 6 months for hyaluronic acid
  • Insulin-dependent diabetes
  • Active infection
  • Pregnant or breast feeding

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
EP-104IAREP-104IAR15mg EP-104IAR in 4 mL carrier fluid
VehicleVehicle4 mL carrier fluid
Primary Outcome Measures
NameTimeMethod
Peak Plasma Concentration (Cmax) of fluticasone propionateUp to 42 weeks
Fluticasone propionate concentrations in synovial fluidUp to 30 weeks
Area under the plasma concentration versus time curve (AUC) of fluticasone propionate12 weeks
Incidence of treatment-emergent adverse eventsUp to 42 weeks
Change from baseline in clinical laboratory parameters: hematology, chemistry (including cortisol) and urinalysisUp to 42 weeks
Secondary Outcome Measures
NameTimeMethod
Change from baseline in patient-reported Short Form - 36 quality of life scoresUp to 42 weeks
Change from baseline in Physician's Global Assessment of ArthritisUp to 42 weeks
Change from baseline in patient-reported Western Ontario and McMaster Universities Arthritis Index (WOMAC)Up to 42 weeks
Time to baseline pain in patient-reported Pain Numerical Rating Scale for Index kneeWeekly up to 42 weeks
Change from baseline in patient-reported Pain Numerical Rating Scale for Index kneeWeekly up to 42 weeks
Change from baseline in patient-reported Global Assessment of ArthritisUp to 42 weeks

Trial Locations

Locations (3)

Centre for Studies in Family Medicine

🇨🇦

London, Ontario, Canada

Fowler Kennedy Sports Medicine Clinic

🇨🇦

London, Ontario, Canada

Rebalance MD

🇨🇦

Victoria, British Columbia, Canada

© Copyright 2025. All Rights Reserved by MedPath