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Study of SAR447537 (INBRX-101) Compared to Plasma-derived A1PI Therapy in Adults With AATD Emphysema

Phase 2
Active, not recruiting
Conditions
Alpha 1-Antitrypsin Deficiency
Emphysema
Interventions
Registration Number
NCT05856331
Lead Sponsor
Sanofi
Brief Summary

Phase 2 study to compare SAR447537 (INBRX-101) to plasma derived A1PI therapy in adults with AATD emphysema

Detailed Description

This is a Phase 2, Double-Blind, Randomized, Active-Control, Parallel Group Study to Assess the Pharmacokinetics, Pharmacodynamics, Immunogenicity, and Safety of SAR447537 (INBRX-101) Compared to Plasma-Derived Alpha1-Proteinase Inhibitor (A1PI) Augmentation Therapy in Adults With Alpha-1 Antitrypsin Deficiency (AATD) Emphysema.

Recruitment & Eligibility

Status
ACTIVE_NOT_RECRUITING
Sex
All
Target Recruitment
99
Inclusion Criteria
  1. Males or females 18-80 years of age, inclusive, at the time of screening
  2. Diagnosis of AATD
  3. Evidence of emphysema secondary to AATD
  4. FEV1 of ≥ 30% and ≤ 80% predicted at screening
  5. Current non-smoking status.
Exclusion Criteria
  1. Receipt of A1PI augmentation therapy within 5 weeks prior to the first dose of study drug
  2. Known or suspected allergy to components of SAR447537 (INBRX-101), A1PI or human IgG
  3. Known selective or severe Immunoglobulin A (IgA) deficiency
  4. Known or suspected diagnosis of type 1 diabetes or diagnosed with uncontrolled type 2 diabetes
  5. Received IV immunoglobulins, monoclonal antibodies and/or other biologic therapies within 30 days
  6. On waiting list for lung or liver transplant
  7. Acute respiratory tract infection or COPD exacerbation within 4 weeks prior to or during screening
  8. Evidence of decompensated cirrhosis
  9. Active cancers or has a history of malignancy within 5 years prior to screening
  10. History of unstable cor pulmonale
  11. Clinically significant congestive heart failure

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
SAR447537 (INBRX-101) Q3WSAR447537IV every 3-weeks (Q3W) and placebo (normal saline)
Zemaira (A1PI)Zemaira60 mg/kg IV once weekly (QW) and placebo (normal saline)
SAR447537 (INBRX-101) Q4WSAR447537IV every 4-weeks (Q4W) and placebo (normal saline)
Primary Outcome Measures
NameTimeMethod
Serum functional AAT (fAAT) levels at steady-state32 Weeks

To assess the mean change in average fAAT concentration as measured by anti-neutrophil elastase capacity \[ANEC\] from baseline to average serum trough fAAT concentration at steady-state (Ctrough,ss) in participants treated with SAR447537 compared to A1PI

Secondary Outcome Measures
NameTimeMethod
fAAT Concentration changes32 Weeks

Mean change in serum fAAT concentration from baseline to fAAT average concentration at steady-state (Cavg, ss) in participants treated with SAR447537 compared to A1PI.

Days with fAAT above the lower limit of the normal range32 weeks

Percentage of days with fAAT above the lower limit of the normal range during steady-state dosing in participants treated with SAR447537 compared to A1PI.

Incidence of TEAEs32 Weeks

Incidence of all treatment-emergent adverse events (TEAEs), TEAEs ≥ Grade 3, serious adverse events (SAEs), TEAEs leading to IMP discontinuation, adverse events of special interest (AESI) (including infusion- related reactions).

Anti-drug antibodies32 Weeks

Frequency of anti-drug antibodies (ADA) against SAR447537 and endogenous AAT, as well as neutralizing ADA (NAb) against SAR447537 and endogenous AAT.

Population Pharmacokinetics: Clearance32 Weeks

Modeling by means of appropriate software to characterize the pharmacokinetic profile of SAR447537 via estimation of the parameter clearance

Population Pharmacokinetics: Volume of Distribution32 Weeks

Modeling by means of appropriate software to characterize the pharmacokinetic profile of SAR447537 via estimation of the parameter volume of distribution

Covariate Analysis: Biometric Values: Weight32 Weeks

Assessment of the impact of participant's weight \[in kg\] on the pharmacokinetic profile of SAR447537

Covariate Analysis: Biometric Values: Height32 Weeks

Assessment of the impact of participant's height \[in cm\] on the pharmacokinetic profile of SAR447537

Covariate Analysis: Biometric Values: Age32 Weeks

Assessment of the impact of participant's age \[in years\] on the pharmacokinetic profile of SAR447537

Covariate Analysis: Biometric Values: Sex32 Weeks

Assessment of the impact of participant's sex \[male or female\] on the pharmacokinetic profile of SAR447537

Trial Locations

Locations (81)

University of Alabama at Birmingham- Site Number : 105

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Birmingham, Alabama, United States

University of Alabama at Birmingham

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Birmingham, Alabama, United States

St Joseph's Hospital and Medical Center- Site Number : 126

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Phoenix, Arizona, United States

St Joseph's Hospital and Medical Center

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Phoenix, Arizona, United States

David Geffen School of Medicine- Site Number : 124

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Los Angeles, California, United States

David Geffen School of Medicine

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Los Angeles, California, United States

UC Davis Comprehensive Cancer Center- Site Number : 110

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Sacramento, California, United States

UC Davis Medical Center

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Sacramento, California, United States

National Jewish Medical and Research Center- Site Number : 123

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Denver, Colorado, United States

National Jewish Medical and Research Center

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Denver, Colorado, United States

Western Connecticut Medical Group- Site Number : 119

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Danbury, Connecticut, United States

Western Connecticut Medical Group

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Danbury, Connecticut, United States

GW Medical Faculty Associates - GW Cancer& Blood Disorders- Site Number : 107

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Washington, District of Columbia, United States

University of Florida College of Medicine- Site Number : 101

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Gainesville, Florida, United States

University of Florida

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Gainesville, Florida, United States

Bruce W. Carter Miami VA Medical Center - NAVREF - PPDS- Site Number : 114

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Miami, Florida, United States

University of Miami

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Miami, Florida, United States

Pulmonary and Sleep of Tampa Bay- Site Number : 115

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Tampa, Florida, United States

Pulmonary and Sleep of Tampa Bay

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Tampa, Florida, United States

Cleveland Clinic Florida

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Weston, Florida, United States

University of Chicago

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Chicago, Illinois, United States

Loyola University Medical Center- Site Number : 112

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Maywood, Illinois, United States

Loyola University Medical Center

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Maywood, Illinois, United States

Indiana University

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Indianapolis, Indiana, United States

Indiana University Health University Hospital- Site Number : 127

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Indianapolis, Indiana, United States

Brigham and Women's Hospital - Lung Center

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Boston, Massachusetts, United States

M Health Fairview Clinics and Surgery Center - Minneapolis- Site Number : 125

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Minneapolis, Minnesota, United States

M Health Fairview Clinics and Surgery Center - Minneapolis

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Minneapolis, Minnesota, United States

Hannibal Regional Healthcare System-HRMG-Hannibal- Site Number : 111

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Hannibal, Missouri, United States

Hannibal Clinic

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Hannibal, Missouri, United States

Columbia University Irving Medical Center- Site Number : 104

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New York, New York, United States

Columbia University

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New York, New York, United States

Pulmonary Health Physicians

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Syracuse, New York, United States

Oregon Health and Science University- Site Number : 117

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Portland, Oregon, United States

Oregon Health and Science University

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Portland, Oregon, United States

Clinical Research Associates Of Central PA , LLC- Site Number : 128

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DuBois, Pennsylvania, United States

Clinical Research Associates Of Central PA , LLC

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DuBois, Pennsylvania, United States

Penn State Health Milton S. Hershey Medical Center- Site Number : 122

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Hershey, Pennsylvania, United States

Penn State Health Milton S. Hershey Medical Center

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Hershey, Pennsylvania, United States

Temple University Hospital- Site Number : 130

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Philadelphia, Pennsylvania, United States

Temple University Hospital

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Philadelphia, Pennsylvania, United States

Velocity Clinical Research - Spartanburg - PPDS- Site Number : 120

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Spartanburg, South Carolina, United States

Velocity Clinical Research - Spartanburg - PPDS

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Spartanburg, South Carolina, United States

Houston Methodist Hospital- Site Number : 113

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Houston, Texas, United States

Houston Methodist Hospital

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Houston, Texas, United States

University of Utah Health

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Salt Lake City, Utah, United States

University of Utah Health Care- Site Number : 106

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Salt Lake City, Utah, United States

Donna McIntyre

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Brisbane, Queensland, Australia

Queensland Centre for Pulmonary Transplantation

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Chermside, Queensland, Australia

Investigational Site Number : 204

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South Brisbane, Queensland, Australia

Royal Adelaide Hospital

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North Adelaide, South Australia, Australia

Eastern Health Clinical School

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Box Hill, Victoria, Australia

Investigational Site Number : 207

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Box Hill, Victoria, Australia

Investigational Site Number : 203

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Fitzroy, Victoria, Australia

St Vincent Hospital Melbourne

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Fitzroy, Victoria, Australia

Frankston Hospital

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Frankston, Victoria, Australia

Institute for Respiratory Health

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Nedlands, Western Australia, Australia

Investigational Site Number : 206

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Nedlands, Western Australia, Australia

Investigational Site Number : 201

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Adelaide, Australia

Investigational Site Number : 202

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Chermside, Australia

Investigational Site Number : 205

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Frankston, Australia

Investigational Site Number : 701

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Hellerup, Denmark

Investigational Site Number : 702

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Vejle, Denmark

NZRSI

🇳🇿

Greenlane, Auckland, New Zealand

Investigational Site Number : 403

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Auckland, New Zealand

Investigational Site Number : 404

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Wellington, New Zealand

P3 Research

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Wellington, New Zealand

Investigational Site Number : 801

🇵🇱

Warszawa, Mazowieckie, Poland

Investigational Site Number : 802

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Kraków, Poland

Investigational Site Number : 901

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Santander, Cantabria, Spain

Investigational Site Number : 903

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Santiago de Compostela, Spain

Investigational Site Number : 601

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Göteborg, Sweden

Ninewells Hospital - PPDS

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Dundee, Angus, United Kingdom

Investigational Site Number : 306

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Wythenshawe, Cheshire West And Chester, United Kingdom

Medicines Evaluation Unit

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Manchester, Cheshire, United Kingdom

Royal Devon and Exeter Hospital (Wonford) - Barrack Rd

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Exeter, Devon, United Kingdom

Investigational Site Number : 304

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Southampton, Hampshire, United Kingdom

Southampton General Hospital

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Southampton, Hampshire, United Kingdom

Investigational Site Number : 302

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Birmingham, Warwickshire, United Kingdom

Queen Elizabeth Hospital Birmingham

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Birmingham, Warwickshire, United Kingdom

Investigational Site Number : 307

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Exeter, United Kingdom

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