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A clinical trial of Capeciatabine to compare the bioequivalence of test and reference products

Not Applicable
Completed
Conditions
Health Condition 1: C509- Malignant neoplasm of breast of unspecified site
Registration Number
CTRI/2011/10/002069
Lead Sponsor
Dr Reddys Laboratories
Brief Summary

Not available

Detailed Description

Not available

Recruitment & Eligibility

Status
Completed
Sex
Not specified
Target Recruitment
110
Inclusion Criteria

1.Male or Female18 to 79 years of age (both inclusive) and having a Body Mass Index (BMI) at least 17 calculated as weight in kg / height in m2

2.Patients must have/have had histopathologically /cytologically confirmed breast cancer or

colorectal cancer.

3.Patients with Dukesâ?? C colon cancer who have undergone complete resection of the primary tumor when treatment with fluoropyrimidine therapy alone is preferred.

Or

Patients with metastatic colorectal carcinoma when treatment with fluoropyrimidine therapy alone is preferred

Or

Patients with metastatic breast cancer resistant to both Paclitaxel and an anthracycline containing chemotherapy regimen or resistant to Paclitaxel and for whom further anthracycline therapy is not indicated

4.Patients who require a daily dose of Capecitabine monotherapy, who are stabilized on twice daily dosing at a dose of 1250 mg/m2 and who have completed at least one cycle of chemotherapy

5.Patients should have their BSA (as per the DuBois formula) between 1.26-1.91 m2 (Both inclusive).

Note : Dosage and administration of Capecitabine will be as per instructions given in section 1.7 Dosage and administration.

6.Eastern Cooperative Oncology Group (ECOG) performance status <= 2.

7.Patient with adequate bone marrow, renal and hepatic function

Exclusion Criteria

1.Prior unanticipated severe reaction to fluoropyrimidine therapy, or known sensitivity to 5-fluorouracil, or known DPD (Dihydropyrimidine Dehydrogenase) deficiency.

2.Pregnant or breast-feeding female

3.Any of the following cardiac conditions:

a.Unstable angina

b.Myocardial infarction within the past 6 months

c.NYHA (New York State Heart Association) class II-IV heart failure

d.Severe uncontrolled ventricular arrhythmias

e.Clinically significant pericardial disease

f.Electrocardiographic evidence of acute ischemic or active conduction system abnormalities

g.Any other cardiac illness that could lead to a safety risk to the patient in case of enrolment in the study

4.History of drug/alcohol addiction

5.Known brain metastasis

6.Patient having abnormal serum calcium level at screening visit which as judged by Investigator could lead to safety risk to the patient upon participation in the trial or could interfere with the conduct of the trial.

7.Pre-existing motor or sensory neurotoxicity of a severity >= grade 2 by NCI CTCAE criteria.

8.A positive hepatitis screen including hepatitis B surface antigen, HCV or HAV (IgM) antibodies

Study & Design

Study Type
BA/BE
Study Design
Not specified
Primary Outcome Measures
NameTimeMethod
To characterise the pharmacokinetic profile of the sponsorâ??s test formulation (Capecitabine Tablets 500 mg, Manufactured by Dr. Reddyâ??s Laboratories, India) relative to that of reference formulation (XELODA® 500 mg tablets, Distributed by Roche Laboratories Inc., USA) in patients of Metastatic Breast Cancer or Colorectal Cancer under fed condition and to assess the bioequivalence.Timepoint: NI
Secondary Outcome Measures
NameTimeMethod
To monitor the safety of the patients, who are exposed to the Investigational Medicinal Product. <br/ ><br> <br/ ><br>Timepoint: NI
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