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Single Ascending Dose Study of BMS-820132 in Patients With Type 2 Diabetes

Phase 1
Completed
Conditions
Diabetes Mellitus, Non-Insulin-Dependent
Interventions
Drug: BMS-820132
Drug: Placebo
Registration Number
NCT01105429
Lead Sponsor
Bristol-Myers Squibb
Brief Summary

BMS-820132 is an investigational new drug being developed by BMS for treating Type 2 diabetes. The purpose of this study is to test the safety/tolerability (potential side effects) of single doses of the investigational new drug, as well as the amount of study drug in the blood, in subjects with type 2 diabetes.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
56
Inclusion Criteria
  • Males and females of childbearing potential (willing to use an acceptable method of contraception), or females of non-childbearing potential (i.e., post-menopausal or surgically sterile)
  • Diagnosis of type 2 diabetes treated with metformin monotherapy on a stable regimen for at least 2 months
  • Body Mass Index (BMI) of 18 to 40 kg/m2
  • Fasting glucose in the range of 100-250 mg/dL
  • Hemoglobin A1c (HbA1c) in the range of 6.5% -9.5%
Read More
Exclusion Criteria
  • Clinically significant deviation from normal in medical history, physical examination, ECGs, and clinical laboratory determinations
  • Any significant acute or chronic medical illness other than stable and well controlled hypertension, microalbuminuria, dyslipidemia, or depression
  • Past history of diabetic ketoacidosis and/or C-peptide < 1.0 ng/mL, hyperosmolar nonketotic syndrome, lactic acidosis, or recurrent hypoglycemia
  • Any major surgery within 4 weeks of study drug administration
  • Any gastrointestinal surgery that could impact upon the absorption of study drug
  • Smoking more than 10 cigarettes per day
  • Recent drug or alcohol abuse
  • Women who are pregnant or breastfeeding
  • Positive urine screen for drugs of abuse
  • Positive blood screen for hepatitis C antibody, hepatitis B surface antigen, or HIV-1, -2 antibody
Read More

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
BMS-820132 (1.0 mg) or PlaceboBMS-820132-
BMS-820132 (0.3 mg) or PlaceboBMS-820132-
BMS-820132 (0.3 mg) or PlaceboPlacebo-
BMS-820132 (1.0 mg) or PlaceboPlacebo-
BMS-820132 (3 mg) or PlaceboBMS-820132-
BMS-820132 (3 mg) or PlaceboPlacebo-
BMS-820132 (10 mg) or PlaceboBMS-820132-
BMS-820132 (10 mg) or PlaceboPlacebo-
BMS-820132 (30 mg) or PlaceboBMS-820132-
BMS-820132 (30 mg) or PlaceboPlacebo-
BMS-820132 (75 mg) or PlaceboBMS-820132-
BMS-820132 (75 mg) or PlaceboPlacebo-
BMS-820132 (150 mg) or PlaceboBMS-820132-
BMS-820132 (150 mg) or PlaceboPlacebo-
BMS-820132 (300 mg) or PlaceboBMS-820132-
BMS-820132 (300 mg) or PlaceboPlacebo-
BMS-820132 (TBD) or PlaceboBMS-820132-
BMS-820132 (TBD) or PlaceboPlacebo-
Primary Outcome Measures
NameTimeMethod
Safety and Tolerability of the investigational drug, as assessed by adverse event monitoring, physical examinations, clinical laboratory determinations, electrocardiograms (ECG), and vital sign assessmentsWithin 5 days of study drug administration
Secondary Outcome Measures
NameTimeMethod
Exposure to the investigational drug and its metabolitesWithin 2 days after study drug administration
Pharmacodynamic activity of the investigational drug on biomarkersWithin 2 days after study drug administration
Excretion of the investigational drug and metabolites from the bodyWithin 2 days after study drug administration

Trial Locations

Locations (3)

Profil Institute For Clinical Research, Inc. (Picr)

🇺🇸

Chula Vista, California, United States

Elite Research Institute

🇺🇸

Miami, Florida, United States

Clinical Pharmacology Of Miami Inc.

🇺🇸

Miami, Florida, United States

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