MedPath

A Study of Disitamab Vedotin With Other Anticancer Drugs in Solid Tumors

Phase 2
Recruiting
Conditions
Breast Neoplasms
Gastroesophageal Junction Adenocarcinoma
HER2 Low Breast Neoplasms
HER2 Positive Breast Neoplasms
Stomach Neoplasms
Triple Negative Breast Neoplasms
Metastatic Breast Cancer
Metastatic Gastric Cancer
Advanced Breast Cancer
Advanced Gastric Cancer
Interventions
Registration Number
NCT06157892
Lead Sponsor
Seagen, a wholly owned subsidiary of Pfizer
Brief Summary

This clinical trial is studying solid tumor cancers. A solid tumor is one that starts in part of your body like your lungs or liver instead of your blood. Once they've grown bigger in one spot or spread to other parts of the body, they're harder to treat. This is called advanced or metastatic cancer.

Participants in this study must have breast cancer or gastric cancer. Participants must have tumors that have HER2 on them. This allows the cancer to grow more quickly or spread faster. There are few treatment options for patients with advanced or metastatic solid tumors that express HER2.

This clinical trial uses an experimental drug called disitamab vedotin (DV). Disitamab vedotin is a type of antibody drug conjugate or ADC. ADCs are designed to stick to cancer cells and kill them.

This clinical trial uses a drug called tucatinib, which has been approved to treat cancer in the United States and some other countries. This drug is sold under the brand name TUKYSA®.

This study will test how safe and how well DV with tucatinib works for participants with solid tumors. This study will also test what side effects happen when participants take these drugs. A side effect is anything a drug does to the body besides treating the disease.

Detailed Description

This clinical trial is to evaluate disitamab vedotin in combination with tucatinib in subjects with LA/metastatic breast cancer or gastric cancer/GEJC that express HER2. The study has a dose escalation phase evaluating disitamab vedotin plus tucatinib followed by a dose optimization phase. The 2 dose levels identified in the dose escalation phase will be assessed in the optimization phase for both safety and efficacy in HER2-expressing LA/mBC and LA/mGC/GEJC. Once the safety and efficacy profile of disitamab vedotin plus tucatinib has been established and a disitamab vedotin dose with the optimum benefit/risk ratio has been determined the disitamab vedotin plus tucatinib combination therapy will be evaluated in an expansion phase with 4 expansion cohorts in subjects with HER2-low LA/mGC/GEJC, HER2+ LA/mGC/GEJC, HER2-low LA/mBC, and HER2+ LA/mBC.

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
172
Inclusion Criteria

General Inclusion Criteria

  • Measurable disease according to RECIST v1.1
  • Eastern Cooperative Oncology Group (ECOG) Performance Status score of 0 or 1

Dose Escalation and Optimization Phase Inclusion Criteria

  • Histologically or cytologically confirmed diagnosis of gastric or gastroesophageal junction adenocarcinoma or breast carcinoma
  • Locally-advanced, unresectable, or metastatic stage
  • Must have experienced disease progression on or after standard of care therapies or be intolerant of standard of care therapies.

Cohort A (HER2-Low Breast Cancer) Inclusion Criteria

  • Histologically or cytologically confirmed diagnosis of breast carcinoma

  • Locally-advanced, unresectable, or metastatic stage

  • HER2-low status determined by most recent local assessment (IHC 1+ or IHC 2+/ISH-negative)

  • Prior therapies requirements

    • No more than 3 prior systemic cytotoxic chemotherapy regimens (including ADCs) for LA/mBC.

    • Participants with known BRCA mutation must have received a PARP-inhibitor where available and not medically contraindicated

    • Have progression on or after, or intolerant to, T-DXd, sacituzumab govitecan, or other topoisomerase I inhibitor therapies, if available as local standard of care therapy

    • Participants with HR+ tumors must have intolerance to endocrine therapy or endocrine therapy refractory disease:

      • Progressed on ≥2 lines of endocrine therapy for LA/mBC AND had received a CDK4/6 inhibitor in the adjuvant or metastatic setting OR
      • Progressed on 1 line of endocrine therapy for LA/mBC AND had a relapse while on adjuvant endocrine therapy after definitive surgery for primary tumor AND had received a CDK4/6 inhibitor in the adjuvant or advanced setting
    • Participants with HR negative, HER2-low and PD-L1-positive (CPS 10 or greater) tumors must have received pembrolizumab with chemotherapy if available as local standard of care therapy.

    • Participants with HR negative, HER2-low and PD-L1-positive (CPS 10 or greater) tumors must have received pembrolizumab (or other PD-(L)1 inhibitor) with chemotherapy if available as local standard of care therapy and not medically contraindicated.

Cohort B (HER2+ Breast Cancer) Inclusion Criteria

  • Histologically or cytologically confirmed diagnosis breast carcinoma

  • Locally-advanced, unresectable, or metastatic stage

  • HER2+ status determined by most recent local assessment (IHC 3+ or IHC 2+/ISH+)

  • Participants must have:

    • Received prior trastuzumab, pertuzumab and a taxane if available as local standard of care therapy for advanced disease.
    • Have progression on or after, or intolerant to, T-DXd or other topoisomerase I inhibitor therapies
    • No more than 3 prior systemic cytotoxic chemotherapy regimens (including ADCs) for LA/mBC

Cohort C (HER2-Low Gastric or Gastroesophageal Junction Adenocarcinoma) Inclusion Criteria

  • Histologically or cytologically confirmed diagnosis of gastric or gastroesophageal junction adenocarcinoma

  • Locally-advanced, unresectable, or metastatic stage

  • HER2-low expression defined as IHC 1+ or IHC 2+/ISH-negative determined by most recent local assessment

  • Willing and able to provide archival or newly obtained formalin-fixed paraffin-embedded (FFPE) tumor tissue blocks

  • Participants must have received:

    • Prior systemic therapy with platinum, fluorouracil, or taxane for locally advanced unresectable or metastatic disease
    • Progression within 6 months of last dose of (neo)adjuvant cytotoxic chemotherapy is considered as 1 line of systemic therapy for LA/mGC/GEJC
    • Prior anti-PD-(L)1 therapy is allowed
    • No more than 2 prior systemic cytotoxic chemotherapy regimens (including ADC) for LA/mGC/GEJC
  • Must not have received prior treatment with HER2 directed therapy

Cohort D (HER2+ LA/mGC/GEJC) Inclusion Criteria

  • Histologically or cytologically confirmed diagnosis of gastric or gastroesophageal junction adenocarcinoma

  • Locally-advanced, unresectable, or metastatic stage

  • HER2+ status determined by most recent local assessment (IHC 3+ or IHC 2+/ISH+)

  • Participants must have:

    • Received prior trastuzumab plus fluoropyrimidine and platinum containing chemotherapy if no contraindication.
    • Prior T-DXd treatment is allowed
    • Prior PD1 inhibitor therapy is allowed
    • No more than 2 prior systemic cytotoxic chemotherapy regimens (including ADCs) for LA/mGC/GEJC
Exclusion Criteria
  • Known hypersensitivity to any excipient contained in the drug formulation of disitamab vedotin or tucatinib
  • Prior therapy with ADCs with MMAE payload
  • Prior therapy with tucatinib
  • Active CNS and/or leptomeningeal metastasis.
  • Participants who have received prior systemic anticancer treatment including investigational agents within 4 weeks prior to first dose of study treatment
  • History of other invasive malignancy within 3 years before the first dose of study intervention, or any evidence of residual disease from a previously diagnosed malignancy.
  • Unable to swallow oral tablets or capsules or any significant GI disease which would preclude the adequate oral absorption of medications

Study & Design

Study Type
INTERVENTIONAL
Study Design
SEQUENTIAL
Arm && Interventions
GroupInterventionDescription
Dose Escalation - Previously treated advanced GC/GEJC or breast cancerdisitamab vedotindisitamab vedotin + tucatinib
Dose Escalation - Previously treated advanced GC/GEJC or breast cancertucatinibdisitamab vedotin + tucatinib
Dose Optimization - HER2-low and HER2+ LA/mBCdisitamab vedotindisitamab vedotin + tucatinib
Dose Optimization - HER2-low and HER2+ LA/mBCtucatinibdisitamab vedotin + tucatinib
Dose Optimization - HER2-low and HER2+ LA/mGC/GEJCdisitamab vedotindisitamab vedotin + tucatinib
Dose Optimization - HER2-low and HER2+ LA/mGC/GEJCtucatinibdisitamab vedotin + tucatinib
Dose Expansion - HER2-low LA/mBCdisitamab vedotindisitamab vedotin + tucatinib
Dose Expansion - HER2-low LA/mBCtucatinibdisitamab vedotin + tucatinib
Dose Expansion - HER2+ LA/mBCdisitamab vedotindisitamab vedotin + tucatinib
Dose Expansion - HER2+ LA/mBCtucatinibdisitamab vedotin + tucatinib
Dose Expansion - HER2-low LA/mGC/GEJCdisitamab vedotindisitamab vedotin + tucatinib
Dose Expansion - HER2-low LA/mGC/GEJCtucatinibdisitamab vedotin + tucatinib
Dose Expansion - HER2+ LA/mGC/GEJCdisitamab vedotindisitamab vedotin + tucatinib
Dose Expansion - HER2+ LA/mGC/GEJCtucatinibdisitamab vedotin + tucatinib
Primary Outcome Measures
NameTimeMethod
Number of participants with dose limiting toxicities (DLTs) in dose escalation phaseUp to 28 days
Number of participants with adverse events (AEs)Through 30 days after the last study treatment; approximately 5 years

Any untoward medical occurrence in a clinical study participant, temporally associated with the use of study intervention, whether or not considered related to the study intervention

Number of participants with laboratory abnormalitiesThrough 30-37 days after the last study treatment: approximately 5 years
Number of participants with dose alterationsThrough 30-37 days after the last study treatment: approximately 5 years
Objective response rate (ORR) per Response Evaluation Criteria in Solid Tumors version 1.1 (RECIST v1.1) by investigator assessmentApproximately 3 years

The proportion of participants with confirmed response (CR) or partial response (PR) according to RECIST v1.1.

Secondary Outcome Measures
NameTimeMethod
Duration of response (DOR) per RECIST v1.1 by investigator assessmentApproximately 5 years

The time from start of the first documentation of objective tumor response of CR or PR (that is subsequently confirmed) to the first documentation of progressive disease (PD) per RECIST v1.1, or to death due to any cause

Disease control rate (DCR) per RECIST v1.1 by investigator assessmentApproximately 5 years

The proportion of participants with stable disease (SD) or confirmed CR or PR according to RECIST v1.1.

Progression free survival (PFS) per RECIST v1.1 by investigator assessmentApproximately 5 years

The time from the start of any study treatment (or randomization date for participants in dose optimization phase) to the first documentation of disease progression per RECIST v1.1 or death due to any cause.

Overall survival (OS)Approximately 5 years

The time from the start of any study treatment (or randomization date for participants in dose optimization phase) to the date of death due to any cause.

Pharmacokinetic (PK) parameter - Maximum concentration (Cmax)Through 30-37 days after the last study treatment; approximately 5 years
PK parameter - Area under the concentration-time curve to the time of the last quantifiable concentration (AUClast)Approximately 1 month
Incidence of anti-drug antibodies (ADAs) against disitamab vedotinThrough 30-37 days after the last study treatment; approximately 5 years

Trial Locations

Locations (118)

Ecg Medica Sl

🇪🇸

Valencia, Spain

Arizona Cancer Center / University of Arizona

🇺🇸

Tucson, Arizona, United States

Banner-University Medical Center Tucson Campus

🇺🇸

Tucson, Arizona, United States

The University of Arizona Cancer Center-North Campus Pharmacy, Attn: Kelly Myrdal

🇺🇸

Tucson, Arizona, United States

The University of Arizona Cancer Center-Main

🇺🇸

Tucson, Arizona, United States

Chao Family Comprehensive Cancer Center University of California Irvine

🇺🇸

Orange, California, United States

UC Irvine Medical Center

🇺🇸

Orange, California, United States

University of California, San Francisco | HDFCCC - Hematopoietic Malignancies

🇺🇸

San Francisco, California, United States

UCLA Department of Medicine - Hematology & Oncology

🇺🇸

Santa Monica, California, United States

Colorado West Healthcare System, dba Community Hospital

🇺🇸

Grand Junction, Colorado, United States

Colorado West Healthcare, dba Grand Valley Oncology

🇺🇸

Grand Junction, Colorado, United States

Danbury Hospital

🇺🇸

Danbury, Connecticut, United States

The Whittingham Cancer Center / Norwalk Hospital

🇺🇸

Norwalk, Connecticut, United States

Georgetown University Medical Center

🇺🇸

Washington, District of Columbia, United States

MedStar Georgetown University Hospital

🇺🇸

Washington, District of Columbia, United States

Moffitt Cancer Center - International Plaza

🇺🇸

Tampa, Florida, United States

H. Lee Moffitt Cancer Center and Research Institute

🇺🇸

Tampa, Florida, United States

Moffitt Cancer Center - McKinley Campus

🇺🇸

Tampa, Florida, United States

Moffitt McKinley Hospital

🇺🇸

Tampa, Florida, United States

Moffitt Cancer Center at Wesley Chapel

🇺🇸

Wesley Chapel, Florida, United States

Georgia Cancer Specialists - Athens

🇺🇸

Athens, Georgia, United States

Georgia Cancer Specialists - Annex

🇺🇸

Atlanta, Georgia, United States

Atlanta Cancer Care - Atlanta

🇺🇸

Atlanta, Georgia, United States

Georgia Cancer Specialists-Northside

🇺🇸

Atlanta, Georgia, United States

Northside Hospital, Inc.- Central Research Department

🇺🇸

Atlanta, Georgia, United States

Northside Hospital

🇺🇸

Atlanta, Georgia, United States

Georgia Cancer Specialists - Blairsville

🇺🇸

Blairsville, Georgia, United States

Georgia Cancer Specialists - Canton

🇺🇸

Canton, Georgia, United States

Atlanta Cancer Care - Cumming

🇺🇸

Cumming, Georgia, United States

Georgia Cancer Specialists - Cumming

🇺🇸

Cumming, Georgia, United States

Georgia Cancer Specialists - Decatur

🇺🇸

Decatur, Georgia, United States

Suburban Hematology-Oncology Associates - Duluth

🇺🇸

Duluth, Georgia, United States

Suburban Hematology-Oncology Associates- Lawrenceville

🇺🇸

Lawrenceville, Georgia, United States

Georgia Cancer Specialists - Macon

🇺🇸

Macon, Georgia, United States

Georgia Cancer Specialists - Marietta

🇺🇸

Marietta, Georgia, United States

Memorial Hospital

🇺🇸

Shiloh, Illinois, United States

Siteman Cancer Center - Shiloh

🇺🇸

Shiloh, Illinois, United States

Massachusetts General Hospital Cancer Center

🇺🇸

Boston, Massachusetts, United States

Massachusetts General Hospital.

🇺🇸

Boston, Massachusetts, United States

University of Texas Southwestern Medical Center - Simmons Cancer Center

🇺🇸

Dallas, Texas, United States

Brigham and Women's Hospital

🇺🇸

Boston, Massachusetts, United States

Dana Farber Cancer Institute

🇺🇸

Boston, Massachusetts, United States

Dana Farber Cancer Institute- Chestnut Hill

🇺🇸

Newton, Massachusetts, United States

Siteman Cancer Center - West County

🇺🇸

Creve Coeur, Missouri, United States

Siteman Cancer Center - North County

🇺🇸

Florissant, Missouri, United States

Saint Luke's Cancer Institute LLC

🇺🇸

Kansas City, Missouri, United States

St Lukes Hospital

🇺🇸

Kansas City, Missouri, United States

Barnes-Jewish Hospital

🇺🇸

Saint Louis, Missouri, United States

Washington University in St Louis.

🇺🇸

Saint Louis, Missouri, United States

Washington University School of Medicine - Siteman Cancer Center

🇺🇸

Saint Louis, Missouri, United States

Siteman Cancer Center - South County

🇺🇸

Saint Louis, Missouri, United States

Siteman Cancer Center - St Peters

🇺🇸

Saint Peters, Missouri, United States

Renown Oncology

🇺🇸

Reno, Nevada, United States

Renown Regional Medical Center

🇺🇸

Reno, Nevada, United States

San Juan Oncology Associates

🇺🇸

Farmington, New Mexico, United States

Memorial Sloan Kettering Cancer Center - Main Hospital

🇺🇸

New York, New York, United States

Zangmeister Cancer Center

🇺🇸

Columbus, Ohio, United States

Saint Francis Hospital / Bon Secours - South Carolina

🇺🇸

Greenville, South Carolina, United States

Sarah Cannon Research Institute - Pharmacy

🇺🇸

Nashville, Tennessee, United States

SCRI Oncology Partners

🇺🇸

Nashville, Tennessee, United States

Tennessee Oncology-Nashville/Sarah Cannon Research Institute

🇺🇸

Nashville, Tennessee, United States

Parkland Health and Hospital System

🇺🇸

Dallas, Texas, United States

University of Texas Southwestern Medical Center Simmons Cancer Center - Redbird

🇺🇸

Dallas, Texas, United States

University of Texas Southwestern Medical Center Clinical Lab-Zale Lipshy University Hospital

🇺🇸

Dallas, Texas, United States

University of Texas Southwestern Medical Center-Simmons Cancer Center Pharmacy

🇺🇸

Dallas, Texas, United States

University of Texas Southwestern Medical Center-William P. Clements Jr. University Hospital

🇺🇸

Dallas, Texas, United States

University of Texas Southwestern Medical Center

🇺🇸

Dallas, Texas, United States

University of Texas Southwestern Simmons Cancer Center - Fort Worth

🇺🇸

Fort Worth, Texas, United States

University of Texas Southwestern Medical Center Clinical Laboratory - Richardson/Plano

🇺🇸

Richardson, Texas, United States

Harborview Medical Center

🇺🇸

Seattle, Washington, United States

Fred Hutchinson Cancer Center / Seattle Cancer Care Alliance / University of Washington

🇺🇸

Seattle, Washington, United States

University of Washington Medical Center

🇺🇸

Seattle, Washington, United States

University of Wisconsin Carbone Cancer Center - Eastpark Medical Center

🇺🇸

Madison, Wisconsin, United States

Carbone Cancer Center / University of Wisconsin

🇺🇸

Madison, Wisconsin, United States

Peninsula & South Eastern Hematology and Oncology Group (PASO)

🇦🇺

Frankston, Victoria, Australia

Slade Pharmacy Frankston

🇦🇺

Frankston, Victoria, Australia

Slade Health

🇦🇺

Mount Waverley, Victoria, Australia

BC Cancer Kelowna.

🇨🇦

Kelowna, British Columbia, Canada

Ottawa Hospital Cancer Centre

🇨🇦

Ottawa, Ontario, Canada

University of Ottawa / Ottawa General Hospital

🇨🇦

Ottawa, Ontario, Canada

Sunnybrook Health Sciences Centre

🇨🇦

Toronto, Ontario, Canada

University Health Network, Princess Margaret Hospital

🇨🇦

Toronto, Ontario, Canada

A.O.U. Federico II

🇮🇹

Napoli, Campania, Italy

Azienda Ospedaliera Universitaria (AOU) Federico II

🇮🇹

Napoli, Campania, Italy

Istituto Nazionale Tumori IRCCS Fondazione G. Pascale

🇮🇹

Napoli, Campania, Italy

Istituto Europeo di Oncologia

🇮🇹

Milano, Lombardia, Italy

Niguarda Ca' Granda Hospital

🇮🇹

Milano, Lombardia, Italy

Humanitas Istituto Clinico Catanese

🇮🇹

Misterbianco (CT), Sicilia, Italy

Azienda Ospedaliera Universitaria Integrata di Verona.

🇮🇹

Verona, Veneto, Italy

Centro Ricerche Cliniche Di Verona Srl

🇮🇹

Verona, Veneto, Italy

UOC Diagnostica per lmmagini e Radioterapia

🇮🇹

Napoli, Italy

Dong-A University Hospital

🇰🇷

Busan, Other, Korea, Republic of

National Cancer Center

🇰🇷

Goyang-si, Other, Korea, Republic of

Chungbuk National University Hospital

🇰🇷

Cheongju-si, Korea, Republic of

Gachon University Gil Medical Center

🇰🇷

Incheon, Korea, Republic of

Seoul National University Bundang Hospital

🇰🇷

Seongnam-si, Korea, Republic of

Korea University Anam Hospital

🇰🇷

Seoul, Korea, Republic of

Samsung Medical Center

🇰🇷

Seoul, Korea, Republic of

Seoul National University Hospital

🇰🇷

Seoul, Korea, Republic of

Severance Hospital Yonsei University Health System

🇰🇷

Seoul, Korea, Republic of

St. Vincent's Hospital, The Catholic University of Korea

🇰🇷

Suwon-si, Korea, Republic of

Quirén Salud Barcelona

🇪🇸

Barcelona, Spain

Hospital Universitari Vall d´Hebron

🇪🇸

Barcelona, Spain

CETIR Grup Medic

🇪🇸

Barcelona, Spain

Hospital Universitario de Basurto

🇪🇸

Bilbao, Spain

Grupo Hospitalario QuironSalud

🇪🇸

Erandio Bizkaia, Spain

L'Institut Catala d'Oncologia.

🇪🇸

L'Hospitalet de Llobregat, Spain

Farmacia-Ensayos. Planta S - Hospital Universitario HM Sanchinarro-CIOCC-START Madrid

🇪🇸

Madrid, Spain

START Madrid-CIOCC_Hospital HM Sanchinarro

🇪🇸

Madrid, Spain

Hospital Clinico Universitario de Valencia

🇪🇸

Valencia, Spain

National Cheng Kung University Hospital

🇨🇳

Tainan, Taiwan

National Taiwan University Hospital

🇨🇳

Taipei, Taiwan

National Taiwan University Cancer Center

🇨🇳

Taipei, Taiwan

The Royal Marsden Hospital

🇬🇧

London, United Kingdom

St Bartholomew's Hospital

🇬🇧

London, United Kingdom

The Royal Marsden NHS Foundation Trust (RM)

🇬🇧

London, United Kingdom

The Christie NHS Foundation Trust

🇬🇧

Manchester, United Kingdom

The Royal Marsden NHS Foundation Trust

🇬🇧

Sutton, United Kingdom

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