MedPath

Efficacy and Safety of Sotagliflozin Versus Placebo in Patients With Type 2 Diabetes Mellitus Not Currently Treated With Antidiabetic Therapy

Phase 3
Completed
Conditions
Type 2 Diabetes Mellitus
Interventions
Registration Number
NCT02926937
Lead Sponsor
Lexicon Pharmaceuticals
Brief Summary

Primary Objective:

To demonstrate the superiority of Sotagliflozin 400 milligrams (mg) versus placebo on hemoglobin A1c (HbA1c) reduction in participants with type 2 diabetes (T2D) who have inadequate glycemic control on diet and exercise.

Secondary Objectives:

* To compare Sotagliflozin 400 mg versus placebo based on:

* Change from baseline in 2-hour postprandial glucose (PPG) following a mixed meal.

* Change from baseline in fasting plasma glucose (FPG).

* Change from baseline in systolic blood pressure (SBP) for participants with baseline SBP ≥130 millimeter per mercury (mmHg).

* Change from baseline in SBP for all participants.

* Change from baseline in body weight.

* Proportion of participants with HbA1c \<6.5%, \<7.0%.

* To compare Sotagliflozin 200 mg versus placebo based on:

* Change from baseline in HbA1c.

* Change from baseline in 2-hour postprandial glucose (PPG) following a mixed meal.

* Change from baseline in body weight.

* Change from baseline in SBP for all participants.

* To evaluate the safety of Sotagliflozin 400 and 200 mg versus placebo.

Detailed Description

Up to 34 weeks, including a Screening Period consisting of a Screening Phase of up to 2 weeks and a 2-week single-blind placebo Run-in Phase, a 26-week double-blind Treatment Period, and a 4-week post-treatment Follow-up visit to collect safety information.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
399
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Sotagliflozin 200 mgPlaceboFollowing a 2-week run-in period, participants were randomized to Sotagliflozin 200 mg administered as 1 Sotagliflozin tablet and 1 matching placebo tablet, QD, before the first meal of the day in the double-blind treatment period for up to 26 weeks.
PlaceboPlaceboFollowing a 2-week run-in period, participants were randomized to matching placebo to sotagliflozin administered as 2 tablets, QD, before the first meal of the day in the double-blind treatment period for up to 26 weeks.
Sotagliflozin 400 mgSotagliflozin (SAR439954)Following a 2-week run-in period, participants were randomized to Sotagliflozin 400 milligrams (mg) administered as two 200 mg tablets, once daily (QD), before the first meal of the day in the double-blind treatment period for up to 26 weeks.
Sotagliflozin 200 mgSotagliflozin (SAR439954)Following a 2-week run-in period, participants were randomized to Sotagliflozin 200 mg administered as 1 Sotagliflozin tablet and 1 matching placebo tablet, QD, before the first meal of the day in the double-blind treatment period for up to 26 weeks.
Primary Outcome Measures
NameTimeMethod
Change From Baseline in Hemoglobin A1c (HbA1c) at Week 26 (Sotagliflozin 400 mg Versus Placebo)Baseline to Week 26

An analysis of covariance (ANCOVA) model was used for the analysis.

Secondary Outcome Measures
NameTimeMethod
Change From Baseline in 2-hour Postprandial Plasma Glucose (PPG) Following a Mixed Meal at Week 26 (Sotagliflozin 400 mg Versus Placebo)Baseline to Week 26

An ANCOVA model was used for the analysis.

Change From Baseline in 2-hour Postprandial Plasma Glucose (PPG) Following a Mixed Meal at Week 26 (Sotagliflozin 200 mg Versus Placebo)Baseline to Week 26

An ANCOVA model was used for the analysis.

Change From Baseline in Fasting Plasma Glucose (FPG) at Week 26 (Sotagliflozin 400 mg Versus Placebo)Baseline to Week 26

An ANCOVA model was used for the analysis.

Change From Baseline in Systolic Blood Pressure (SBP) at Week 12 in Participants With Baseline SBP ≥130 Millimeter of Mercury (mmHg) (Sotagliflozin 400 mg Versus Placebo)Baseline to Week 12

An ANCOVA model was used for the analysis.

Change From Baseline in SBP at Week 12 for All Participants (Sotagliflozin 400 mg Versus Placebo)Baseline to Week 12

An ANCOVA model was used for the analysis.

Change From Baseline in SBP at Week 12 for All Participants (Sotagliflozin 200 mg Versus Placebo)Baseline to Week 12

An ANCOVA model was used for the analysis.

Change From Baseline in Body Weight at Week 26 (Sotagliflozin 400 mg Versus Placebo)Baseline to Week 26

An ANCOVA model was used for the analysis.

Change From Baseline in Body Weight at Week 26 (Sotagliflozin 200 mg Versus Placebo)Baseline to Week 26

An ANCOVA model was used for the analysis.

Percentage of Participants With HbA1c <6.5% at Week 26 (Sotagliflozin 400 mg Versus Placebo)Week 26
Percentage of Participants With HbA1c <7.0% at Week 26 (Sotagliflozin 400 mg Versus Placebo)Week 26
Change From Baseline in HbA1c at Week 26 (Sotagliflozin 200 mg Versus Placebo)Baseline to Week 26

An ANCOVA model was used for the analysis.

Trial Locations

Locations (70)

Investigational Site Number 4841010

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Aguascalientes, Mexico

Investigational Site Number 4841001

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Culiacan, Mexico

Investigational Site Number 4841005

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Durango, Durango, Mexico

Investigational Site Number 4841002

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Monterrey, Nuevo León, Mexico

Investigational Site Number 8401011

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Los Angeles, California, United States

Investigational Site Number 8401035

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San Dimas, California, United States

Investigational Site Number 8401024

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Bradenton, Florida, United States

Investigational Site Number 8401007

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Hialeah, Florida, United States

Investigational Site Number 8401051

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Anderson, South Carolina, United States

Investigational Site Number 8401033

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Atlanta, Georgia, United States

Investigational Site Number 8401048

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Akron, Ohio, United States

Investigational Site Number 8401023

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Sugar Land, Texas, United States

Investigational Site Number 8401049

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Tucson, Arizona, United States

Investigational Site Number 8401058

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Garden Grove, California, United States

Investigational Site Number 8401017

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Huntington Park, California, United States

Investigational Site Number 8401044

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Chicago, Illinois, United States

Investigational Site Number 4841004

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Chihuahua, Mexico

Investigational Site Number 8401057

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Canoga Park, California, United States

Investigational Site Number 8401014

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Daytona Beach, Florida, United States

Investigational Site Number 8401038

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Lake Charles, Louisiana, United States

Investigational Site Number 8401028

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Anaheim, California, United States

Investigational Site Number 8401022

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Montclair, California, United States

Investigational Site Number 8401039

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Norwalk, California, United States

Investigational Site Number 8401026

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Tucson, Arizona, United States

Investigational Site Number 8401029

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Hawaiian Gardens, California, United States

Investigational Site Number 8401056

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Long Beach, California, United States

Investigational Site Number 8401013

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Long Beach, California, United States

Investigational Site Number 8401063

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Los Angeles, California, United States

Investigational Site Number 8401025

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Tustin, California, United States

Investigational Site Number 4841006

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Aguascalientes, Mexico

Investigational Site Number 8401003

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Marion, Ohio, United States

Investigational Site Number 4841003

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Cd. México, México, Mexico

Investigational Site Number 4841009

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Guadalajara, Mexico

Investigational Site Number 4841007

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Mexico, Mexico

Investigational Site Number 4841008

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Monterrey, Mexico

Investigational Site Number 8401050

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Houston, Texas, United States

Investigational Site Number 8401008

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Miami, Florida, United States

Investigational Site Number 8401001

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San Antonio, Texas, United States

Investigational Site Number 8401015

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Van Nuys, California, United States

Investigational Site Number 8401062

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Palm Harbor, Florida, United States

Investigational Site Number 8401031

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Denver, Colorado, United States

Investigational Site Number 8401002

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Greer, South Carolina, United States

Investigational Site Number 8401060

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Northglenn, Colorado, United States

Investigational Site Number 8401040

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Clearwater, Florida, United States

Investigational Site Number 8401046

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Homestead, Florida, United States

Investigational Site Number 8401018

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Miami, Florida, United States

Investigational Site Number 8401061

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West Palm Beach, Florida, United States

Investigational Site Number 8401016

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West Des Moines, Iowa, United States

Investigational Site Number 8401042

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Fayetteville, North Carolina, United States

Investigational Site Number 1241006

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Vancouver, Canada

Investigational Site Number 8401012

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Greensboro, North Carolina, United States

Investigational Site Number 8401052

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Newton, Iowa, United States

Investigational Site Number 8401034

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Wichita, Kansas, United States

Investigational Site Number 8401041

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Levittown, Pennsylvania, United States

Investigational Site Number 8401020

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Corvallis, Oregon, United States

Investigational Site Number 8401006

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Eugene, Oregon, United States

Investigational Site Number 8401010

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Suffolk, Virginia, United States

Investigational Site Number 8401055

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Schertz, Texas, United States

Investigational Site Number 8401005

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Fort Worth, Texas, United States

Investigational Site Number 1241005

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Toronto, Canada

Investigational Site Number 1241001

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Toronto, Canada

Investigational Site Number 8401019

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Houston, Texas, United States

Investigational Site Number 8401059

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North Richland Hills, Texas, United States

Investigational Site Number 8401004

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San Antonio, Texas, United States

Investigational Site Number 8401037

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Katy, Texas, United States

Investigational Site Number 8401043

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McAllen, Texas, United States

Investigational Site Number 8401054

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San Antonio, Texas, United States

Investigational Site Number 8401032

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Chesapeake, Virginia, United States

Investigational Site Number 1241002

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Sherbrooke, Canada

Investigational Site Number 8401053

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Orlando, Florida, United States

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