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Study to determine if the investigational drug obeticholic acid (also known as OCA) in combination with the investigational drug bezafibrate (BZF), has an effect on Primary Biliary Cholangitis (also known as Primary Biliary Cirrhosis or PBC).

Phase 1
Conditions
Primary Biliary Cholangitis (PBC) in patients with Inadequate Response or who were Unable to Tolerate Ursodeoxycholic Acid
MedDRA version: 20.1Level: LLTClassification code 10036680Term: Primary biliary cirrhosisSystem Organ Class: 100000004871
Therapeutic area: Diseases [C] - Digestive System Diseases [C06]
Registration Number
EUCTR2018-002575-17-FR
Lead Sponsor
Intercept Pharmaceuticals, Inc.
Brief Summary

Not available

Detailed Description

Not available

Recruitment & Eligibility

Status
ot Recruiting
Sex
All
Target Recruitment
54
Inclusion Criteria

- A definite or probable diagnosis of PBC (consistent with the European Association for the Study of the Liver [EASL] Practice Guidelines and the American Association for the Study of Liver Diseases; [Lindor 2009a, EASL 2017])
- Qualifying ALP and bilirubin liver biochemistry values
- Age =18 years
- Taking UDCA for at least 12 months (stable dose for =3 months) before Day 1 or unable to tolerate or unresponsive to UDCA (no UDCA for =3 months) before Day 1
Are the trial subjects under 18? no
Number of subjects for this age range:
F.1.2 Adults (18-64 years) yes
F.1.2.1 Number of subjects for this age range 50
F.1.3 Elderly (>=65 years) yes
F.1.3.1 Number of subjects for this age range 4

Exclusion Criteria

- History or presence of other concomitant liver diseases
- Presence of clinical complications of PBC or clinically significant (CS) hepatic decompensation
- Current or history of gallbladder disease with or without cholelithiasis
- Severe renal failure (serum creatinine >1.5 mg/100 mL (>135 µmol/L); creatinine clearance <60 mL/min) or undergoing dialysis
- Severe pruritus, or required systemic treatment for pruritus (eg, with bile acid sequestrants or rifampicin) within 2 months of Day 1
- History of known or suspected CS hypersensitivity to OCA, BZF, or other fibrates or any of their components
- Was treated with commercially available OCA or participated in a previous study involving OCA within 1 year before Screening or plans to use commercially available OCA during the study
- Is unable to tolerate BZF or other fibrates, was treated with commercially available fibrates or participated in a previous study involving fibrates within 3 months before Screening, or plans to use commercially available fibrates during the study

Note: Other protocol defined Inclusion/Exclusion criteria may apply

Study & Design

Study Type
Interventional clinical trial of medicinal product
Study Design
Not specified
Primary Outcome Measures
NameTimeMethod
Main Objective: The primary objective is to assess the effects of the combination of OCA and BZF on alkaline phosphatase (ALP) in comparison to OCA alone in subjects with PBC who had an inadequate response or who were unable to tolerate ursodeoxycholic acid (UDCA).;Secondary Objective: The secondary objectives are to assess the effects of the combination of OCA and BZF in comparison to OCA alone in subjects with PBC who had an inadequate response or who were unable to tolerate UDCA on the following:<br>- Safety and tolerability<br>- Response and normalization rates of biochemical disease markers<br>- Disease-specific symptoms as assessed by health-related quality of life questionnaires <br>- Biomarkers of bile acid synthesis and homeostasis;Primary end point(s): Absolute change in ALP from baseline to Week 12 in the DB Treatment Period;Timepoint(s) of evaluation of this end point: week 12
Secondary Outcome Measures
NameTimeMethod
Secondary end point(s): - Safety and tolerability<br>- Response and normalization rates of biochemical disease markers<br>- Disease-specific symptoms as assessed by health-related quality of life questionnaires <br>- Biomarkers of bile acid synthesis and homeostasis;Timepoint(s) of evaluation of this end point: Baseline to End of study
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