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Measurement of Insulin Levels in the Cerebrospinal Fluid of Healthy Adults After a Single Intranasal Dose - Middle Age

Phase 1
Not yet recruiting
Conditions
Healthy
Interventions
Drug: Low Dose Regular insulin
Drug: High Dose Regular insulin
Other: 0.9% Saline
Registration Number
NCT06434038
Lead Sponsor
HealthPartners Institute
Brief Summary

The purpose of this study is to find out whether insulin, a drug approved by the FDA for the treatment of diabetes mellitus, reaches the brain and spinal cord when delivered as a nasal spray (intranasally). Intranasal insulin has been shown to improve memory and mood in patients with neurological diseases such as mild cognitive impairment and dementia, but more evidence is needed to support the ability to effectively target the brain through intranasal routes.

18 healthy middle-aged adults will be randomly assigned to receive a single intranasal dose of 40 units insulin ("low dose" group), 80 units insulin ("high dose" group), or saline (placebo, or control group). Participants will undergo an image-guided lumbar puncture (spinal tap) performed by a study clinician. Samples of cerebrospinal fluid (a fluid surrounding the brain and spinal cord) and blood will be collected at 5 timepoints during the lumbar puncture: once prior to the administration of intranasal insulin, and again at 10, 20, 30, and 40 minutes after the dose is given. Samples will be tested to determine the level of insulin detected in the cerebrospinal fluid and blood at each time point. Results of this study will provide essential information about the ability of insulin to reach the brain after intranasal administration.

Detailed Description

Not available

Recruitment & Eligibility

Status
NOT_YET_RECRUITING
Sex
All
Target Recruitment
18
Inclusion Criteria
  1. Subject is between ≥36 and ≤ 55 years of age
  2. Subject's BMI is between >=18.5 and <=24.9, or can safely undergo a lumbar puncture at the discretion of the radiologist
  3. MOCA score ≥26
  4. Subject must be proficient in speaking English to comply with instructions and measures for the study
  5. Subject can provide written informed consent
  6. Female subjects must have either: (1) a negative pregnancy test at the screening visit and treatment visit OR (2) be at least 2 years post-menopausal / surgically sterile.
Exclusion Criteria
  1. Subject has medical history and/or clinically determined disorders: chronic sinusitis, previous nasal and/or oto-pharyngeal surgery and severe deviated septum and/or other anomalies.
  2. Subject has history of any of the following: active and significant central nervous system, psychiatric illness, pulmonary, or cardiovascular disorders or any other clinically relevant abnormality that inclusion would pose a safety risk to the subject as determined by investigator
  3. Subject has participated in a clinical trial investigation within 3 months of this study.
  4. Subject has an insulin allergy
  5. Subject has Insulin-dependent diabetes
  6. Subject is pregnant or breast feeding
  7. Contraindication to spinal tap or other safety factors that preclude lumbar puncture in the investigator's opinion
  8. Any other clinically relevant finding that would pose a safety risk to the subject as determined by the investigator

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Low dose intranasal insulinLow Dose Regular insulinOne dose of 40 international units of regular insulin administered intranasally.
High dose Intranasal InsulinHigh Dose Regular insulinOne dose of 80 international units of regular insulin administered intranasally.
Placebo Control0.9% SalineOne dose of 0.9% saline administered intranasally.
Primary Outcome Measures
NameTimeMethod
Tmax of insulin concentration-Cerebrospinal FLuid0-40 minutes post-intranasal administration

CSF insulin concentration will also be reported by Tmax (time of peak concentration)

Concentration of insulin over Time - Cerebrospinal fluid0-40 minutes post-intranasal administration

Insulin concentration detected in cerebrospinal fluid at 5 time points (pre-insulin dose; and 10, 20, 30, 40 minutes after dose). Values will be reported as μIU/mL. Higher values indicate a greater concentration of insulin in the cerebrospinal fluid. Concentrations for each time point (overall and by dose) will be reported as a mean +/- standard error.

AUC (area under the curve) of insulin concentration-Cerebrospinal Fluid0-40 minutes post-intranasal administration

CSF insulin concentration will also be reported by AUC (area under the curve, measured as time x concentration)

Cmax of insulin concentration- Cerebrospinal Fluid0-40 minutes post- intranasal administration

CSF insulin concentration will also be reported by Cmax (peak concentration)

Secondary Outcome Measures
NameTimeMethod
AUC (area under the curve) of insulin concentration - Serum0-40 minutes post-intranasal administration

Serum insulin concentration will also be reported by AUC (area under the curve, measured as time x concentration).

Tmax of insulin - Serum0-40 minutes post-intranasal administration

Serum insulin concentration will also be reported by Tmax (time to peak concentration)

Insulin Concentration Over Time- Serum0-40 minutes post-intranasal administration

Insulin concentration detected in blood at 5 time points (pre-insulin dose; and 10, 20, 30, 40 minutes after dose). Values will be reported at μIU/mL. Higher values indicate a greater concentration of insulin in the blood. Concentrations for each time point (overall and by dose) will be reported as a mean +/- standard error.

Cmax of insulin concentration - Serum0-40 minutes post-intranasal adminitration

Serum insulin concentration will also be reported by Cmax (peak concentration)

Trial Locations

Locations (1)

HealthPartners Neuroscience Center

🇺🇸

Saint Paul, Minnesota, United States

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