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A Study to Investigate the Pharmacodynamic Effect of Single Doses of MT-8554 in Healthy Subjects

Phase 1
Completed
Conditions
Healthy
Interventions
Drug: MT-8554 low dose
Drug: MT-8554 high dose
Drug: Placebo
Registration Number
NCT02536209
Lead Sponsor
Mitsubishi Tanabe Pharma Corporation
Brief Summary

The purpose of this study is to investigate the pharmacodynamic effect of single doses of MT-8554 in healthy subjects.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
Male
Target Recruitment
20
Inclusion Criteria
  • Healthy and free from clinically significant illness or disease
  • Male Caucasian subjects aged 18 to 55
  • A body weight of ≥60 kg
Exclusion Criteria
  • Participation in more than three clinical studies involving administration of an Investigational Medicinal Product (IMP) in the previous year, or any study within 12 weeks.
  • Clinically significant endocrine, thyroid, hepatic, respiratory, gastro-intestinal, renal, cardiovascular disease, or history of any significant psychiatric/psychotic illness disorder.
  • Clinically relevant abnormal medical history, physical findings or laboratory values

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
Regimen 1MT-8554 low dosePeriod 1: MT-8554 low dose, Period 2: MT-8554 high dose, Period 3: Placebo and Period 4: Oxycodone hydrochloride, respectively single dosing
Regimen 1MT-8554 high dosePeriod 1: MT-8554 low dose, Period 2: MT-8554 high dose, Period 3: Placebo and Period 4: Oxycodone hydrochloride, respectively single dosing
Regimen 3MT-8554 high dosePeriod 1: Placebo, Period 2: MT-8554 low dose, Period 3: Oxycodone hydrochloride and Period 4: MT-8554 high dose, respectively single dosing
Regimen 1Oxycodone hydrochloridePeriod 1: MT-8554 low dose, Period 2: MT-8554 high dose, Period 3: Placebo and Period 4: Oxycodone hydrochloride, respectively single dosing
Regimen 2MT-8554 low dosePeriod 1: MT-8554 high dose, Period 2: Oxycodone hydrochloride, Period 3: MT-8554 low dose and Period 4: Placebo, respectively single dosing
Regimen 4MT-8554 low dosePeriod 1: Oxycodone hydrochloride, Period 2: Placebo, Period 3: MT-8554 high dose and Period 4: MT-8554 low dose, respectively single dosing
Regimen 4MT-8554 high dosePeriod 1: Oxycodone hydrochloride, Period 2: Placebo, Period 3: MT-8554 high dose and Period 4: MT-8554 low dose, respectively single dosing
Regimen 1PlaceboPeriod 1: MT-8554 low dose, Period 2: MT-8554 high dose, Period 3: Placebo and Period 4: Oxycodone hydrochloride, respectively single dosing
Regimen 2MT-8554 high dosePeriod 1: MT-8554 high dose, Period 2: Oxycodone hydrochloride, Period 3: MT-8554 low dose and Period 4: Placebo, respectively single dosing
Regimen 3PlaceboPeriod 1: Placebo, Period 2: MT-8554 low dose, Period 3: Oxycodone hydrochloride and Period 4: MT-8554 high dose, respectively single dosing
Regimen 2Oxycodone hydrochloridePeriod 1: MT-8554 high dose, Period 2: Oxycodone hydrochloride, Period 3: MT-8554 low dose and Period 4: Placebo, respectively single dosing
Regimen 2PlaceboPeriod 1: MT-8554 high dose, Period 2: Oxycodone hydrochloride, Period 3: MT-8554 low dose and Period 4: Placebo, respectively single dosing
Regimen 3MT-8554 low dosePeriod 1: Placebo, Period 2: MT-8554 low dose, Period 3: Oxycodone hydrochloride and Period 4: MT-8554 high dose, respectively single dosing
Regimen 4PlaceboPeriod 1: Oxycodone hydrochloride, Period 2: Placebo, Period 3: MT-8554 high dose and Period 4: MT-8554 low dose, respectively single dosing
Regimen 3Oxycodone hydrochloridePeriod 1: Placebo, Period 2: MT-8554 low dose, Period 3: Oxycodone hydrochloride and Period 4: MT-8554 high dose, respectively single dosing
Regimen 4Oxycodone hydrochloridePeriod 1: Oxycodone hydrochloride, Period 2: Placebo, Period 3: MT-8554 high dose and Period 4: MT-8554 low dose, respectively single dosing
Primary Outcome Measures
NameTimeMethod
Pharmacodynamic effect as measured by Visual Analogue Scale for Cold Pressor Testup to 10 hours post dosing
Secondary Outcome Measures
NameTimeMethod
Safety and Tolerability as measured by physical examinationup to Day6 of treatment period 4
Safety and Tolerability as measured by ECGup to Day6 of treatment period 4
Safety and Tolerability as measured by vital signsup to Day6 of treatment period 4
Safety and Tolerability as measured by laboratory safety assessmentsup to Day6 of treatment period 4
Plasma concentration of Oxycodone hydrochloride at the time of Pharmacodynamic assessmentsup to 10 hours post dosing
Safety and Tolerability as measured by number of participants with adverse eventsup to Day6 of treatment period 4
Plasma concentration of MT-8554 at the time of Pharmacodynamic assessmentsup to 10 hours post dosing

Trial Locations

Locations (1)

Investigational center

🇬🇧

City name, United Kingdom

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