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A Study to Compare the Pharmacokinetics of YM150 Formulation-A and Formulation-B

Phase 1
Completed
Conditions
Healthy Volunteer
Pharmacokinetics of YM150
Interventions
Registration Number
NCT01125657
Lead Sponsor
Astellas Pharma Inc
Brief Summary

This study is to compare its pharmacokinetics profile of two YM150 formulations by 2x2 crossover method.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
Male
Target Recruitment
44
Inclusion Criteria
  • Body weight: ≥50.0 kg, <80.0 kg
  • BMI: ≥17.6, <26.4
  • Healthy, as judged by the investigator or sub-investigator based on the results of physical examinations and lab tests
Exclusion Criteria
  • Received any investigational drugs within 120 days before the study
  • Donated 400 mL of whole blood within 90 days, 200 mL of whole blood within 30 days, or blood components within 14 days before the study
  • Received medication within 7 days before the study
  • A deviation from the assessment criteria of physical examinations or laboratory tests
  • A deviation from the normal reference range of coagulation test [PT (INR) or aPTT]
  • History of drug allergies
  • Upper gastrointestinal disease within 7 days before the study
  • Concurrent or previous hepatic, gastrointestinal, heart, cerebrovascular or respiratory diseases
  • Concurrent or previous malignant tumor
  • Previous treatment with YM150

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
formualation-A to -B sequence groupYM150-
formulation-B to -A sequence groupYM150-
Primary Outcome Measures
NameTimeMethod
Plasma concentration of YM150 and its metabolites measured by blood samplefor 3 days after drug administration
Secondary Outcome Measures
NameTimeMethod
Safety assessed by AEs, vital signs, 12-lead ECG and lab testsor 3 days after drug administration
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