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Pivotal Efficacy and Safety Registration Trial of FP187 in Moderate to Severe Plaque Psoriasis

Phase 2
Completed
Conditions
Plaque Psoriasis
Interventions
Drug: FP187
Drug: Placebo
Registration Number
NCT01230138
Lead Sponsor
Forward-Pharma GmbH
Brief Summary

The purpose of this trial is to investigate the efficacy and safety of different doses and dose administrations of FP187 compared to a placebo treatment in patients with moderate to severe plaque psoriasis.

Detailed Description

The trial tests two different dose levels and two different daily dosing schedules (twice daily (BID) and three times daily (TID))over 20 weeks of treatment. Key is effect as measured by achievement of a 75% reduction in PASI after 20 weeks and safety monitored by adverse events and safety lab.

There are 3 active arms:

1. FP-187 at a daily dose of 750mg divided in three doses (250mg TID)

2. FP-187 at a daily dose of 750mg divided in two doses (375mg BID)

3. FP-187 at a daily dose of 500mg divided in two doses (250mg BID)

and 1 placebo arm.

An additional open (flexible dosing) treatment arm has been amended to the trial

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
252
Inclusion Criteria
  • Patients of either sex at least 18 years of age

  • A clinical diagnosis of plaque psoriasis defined as skin areas with erythema, induration and scaling, with a body surface area of no less than 10% and in total to be scoring at least 10 on the PASI scale

  • The psoriasis disease have been stable for at least 6 months at randomization

  • Signed and dated informed consent

  • Sexually active females of childbearing potential must be either surgically sterile (hysterectomy or tubal ligation) or use a highly effective (failure rate < 1%) medically accepted contraceptive method during the trial as well as one month after trial is finished such as:

    • Systemic contraceptive (oral, implant, injection),
    • Intrauterine device (IUD) inserted for at least one month prior to study entrance
  • Willingness and ability to comply with the trial procedures

  • Patient is beside the psoriasis disease in good general health in the opinion of the Investigator, as determined by medical history, physical examination, vital signs and clinical laboratory parameters (hematology, biochemistry and urinalysis).

Exclusion Criteria
  • Female patients who are pregnant or breast-feeding or planning to become pregnant up to 7 months from treatment start as well as male patients plan-ning pregnancy with their partner up to 7 months from treatment start or practise unprotected sexual relationship up to 7 months from treatment start
  • Known allergy to any of the constituents of the product being tested
  • Pustular forms of psoriasis, erythrodermic or guttate psoriasis
  • Known immunosuppressive diseases (e.g., AIDS/HIV)
  • Presence of another serious or progressive disease which, according to the Investigator may interfere with treatment outcome
  • Active skin disease such as atopic dermatitis, rosacea, lupus erythematosus, or other inflammatory or infectious skin disease which, according to the Investigator may interfere with treatment outcome
  • Use of topical medical treatment or UVB treatment - Use of systemic anti-psoriatic treatment preceding the baseline visit Methotrexate, cyclosporine, steroids or PUVA treatment within x weeks; Biological treatment (efalizumab, adalimumab, infliximab, etanercept) within xx weeks; Acitretin within x months; Treatment with Fumaderm® or other DMF containing products during past xx weeks prior to baseline visit; Discontinuation of previous treatment with Fumaderm® or other DMF containing products due to lack of efficacy or side effects;
  • Has within the past x weeks prior to baseline visit been treated with drugs influencing the course of the psoriasis such as antimalarial drugs, beta-blockers or lithium
  • Has a relevant clinical history of stomach or intestinal problems (eg gastritis or peptic ulcer within the last 10 years )
  • Has liver enzyme measures (AST, ALT, Gamma-GT) higher than 2x UNL)
  • Has an estimated Creatinine Clearance: < xx ml/min
  • Has leucopenia (leukocyte count < x/mm3) or eosinophilia (count >x/µl) or lymphopenia (count < x/nl).
  • Has protein in the urine test at screening or baseline visit
  • Participation in another clinical trial during the last month preceding the baseline visit or participation in a trial with treatment of biologicals within x months prior to baseline visit
  • Patients who are involved in the organisation of the clinical investigation or are in any way dependant on the investigator or sponsor

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
FP187 - TIDFP187FP187 250mg TID (total daily dose of 750mg)
FP187- BIDFP187FP187 375mg BID (total daily dose of 750mg)of 750mg administered as 375mg BID
FP187-LD-BIDFP187FP187 250mg BID (total daily dose of 500mg)
PlaceboPlaceboPlacebo treatment
Open, flexible dosing treatment armFP187Open treatment using a flexible dosing schedule for 8 weeks with maximum dose of 750mg FP187 and with a total dosing of 20 weeks. All investigations following same schedule.
Primary Outcome Measures
NameTimeMethod
Proportion of patients achieving PASI 75 compared to placeboAfter 20 weeks of treatment

Proportion of patients achieving PASI75 (a reduction in the PASI score of 75% or more)

Secondary Outcome Measures
NameTimeMethod
PASI 75At week 4, 8, 12 and 16

Proportion of patients achieving PASI75 (a reduction of the PASI score of 75% or more compared to baseline)

PASI 50At week 4, 8, 12, 16 and 20

Proportion of patients who achieves PASI 50 (a reduction of the PASI score of 50% or more compared to baseline)

PASI 90At week 4, 8, 12, 16 and 20

Proportion of patients achieving PASI90 (a reduction of the PASI score of 90% or more compared to baseline

PGA (Physicians Global Assessment)At week 4, 8, 12, 16 and 20

On a 5-point scale from 0 (abscence or very mild disease) to 4 (very severe disease) proportion of patients being responders - defined as patients achieving either a score of 0 or 1 or a two point improvement

PaGA (Patients Global AssessmentAt week 4,8,12,16 and 20

Patients evaluation on a 5-point Likert scale 1 (very good) - 5 (very poor)based on the evaluation of: "Considering all the ways your psoriasis affects you, how have you been doing in the last 24 hours?"

PruritusAt week 4, 8, 12, 16 and 20

Patient evaluation of pruritus measured on a VAS (Visual Analog Scale) from 0mm (no pruritus) to 100mm (worst possible pruritus)

Patient rated QoL (Quality of Life)At week 4, 8, 12, 16 and 20

Patient filling in 10 questions on the DLQI QoL system with a calculated summary score and analysis of the improvement from baseline

Adverse events (AEs)At week 4, 8, 12, 16 and 20

Summary of incidense and severity of AEs and ADRs (Adverse Drug Reactions)/SAEs (Serious Adverse Events)/SUSARs (Suspected Unexpected Serious Adverse Reactions)

Safety lab testAt week 20

Summary of lab parameters and clinically relevant changes over the treatment period in standard clinical chemistry tests, standard haematology tests and urin dip stick test

Trial Locations

Locations (2)

Dermatological Dept., Uniklinikum, TU-Dresden

🇩🇪

Dresden, Germany

SCIderm

🇩🇪

Hamburg, Germany

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