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Masitinib in First Line Treatment of Gastro-Intestinal Stromal Tumor (GIST)

Phase 3
Terminated
Conditions
Gastrointestinal Stromal Tumors
Interventions
Registration Number
NCT00812240
Lead Sponsor
AB Science
Brief Summary

Masitinib in First Line Treatment of Gastro-Intestinal Stromal Tumor (GIST)

Detailed Description

Masitinib is a selective tyrosine kinase inhibitor with potent activity against wild-type c-Kit, the juxta membrane domain of c-Kit, and PDGFR. In addition to its direct inhibitory action against these kinase targets, masitinib is also thought to promote survival via modulation of immunostimulation-mediated anticancer effects and modulation of the tumor microenvironment. The objective of this prospective, multicenter, randomized, open-label, active-controlled study is to compare the efficacy and safety of masitinib with respect to imatinib in the first line treatment of gastro-intestinal stromal tumor (GIST). Treatment will be given until disease progression, limiting toxicity or patient consent withdrawal.

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
335
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Active Comparator (7.5)ImatinibParticipants receive imatinib at 400 or 600 mg per day
Masitinib (7.5)MasitinibParticipants receive masitinib (7.5 mg/kg/day), given orally twice daily.
Masitinib (6.0)MasitinibParticipants receive masitinib (6.0 mg/kg/day), given orally twice daily
Active Comparator (6.0)ImatinibParticipants receive imatinib at 400 or 600 mg per day
Primary Outcome Measures
NameTimeMethod
Progression Free Survival (PFS)From day of randomization to disease progression or death, assessed for a maximum of 96 months]

Progression Free Survival is defined as the time from randomization to first documentation of objective tumor progression (date of tumor assessment documenting progressive disease assessed by CT Scan according to RECIST 1.1 and based on central review) or to death due to any cause (whichever comes first).

Secondary Outcome Measures
NameTimeMethod
Overall Survival (OS)From day of randomization to death, assessed for a maximum of 96 months

Overall survival is defined as time in months from the randomization date to the date of death due to any cause

Trial Locations

Locations (41)

Centre Val d'Aurèle

🇫🇷

Montpellier, France

Makassed General Hospital Tarik Jadide

🇱🇧

Beirut, Lebanon

Hôpital Saint-Georges

🇱🇧

Beirut, Lebanon

Hôpital Européen Georges Pompidou

🇫🇷

Paris, France

Hôpital de la Source

🇫🇷

Orléans, France

Cancer Centers of the Carolinas

🇺🇸

Greenville, South Carolina, United States

CHD de Vendée

🇫🇷

La Roche sur Yon, France

Institut Paoli Calmette

🇫🇷

Marseille, France

Centre Hsopitalier de La Rochelle

🇫🇷

La Rochelle, France

Beth Israel Medical Center

🇺🇸

New York, New York, United States

Institut Sainte Catherine

🇫🇷

Avignon, France

Centre René Gauducheau

🇫🇷

Nantes, France

Centre Léon Bérard

🇫🇷

Lyon, France

Hopital Bocage

🇫🇷

Dijon, France

Centre Hospitalier Victor Jousselin

🇫🇷

Dreux, France

Centre Oscar Lambret

🇫🇷

Lille, France

Centre Hospitalier d'Abbeville

🇫🇷

Abbeville, France

Hôpital Jean Minjoz

🇫🇷

Besançon, France

Hôpitalo Henri Mondor

🇫🇷

Créteil, France

Rafik Hariri University Hospital

🇱🇧

Beirut, Lebanon

Groupe Hospitalier Diaconesse Croix Saint Simon

🇫🇷

Paris, France

Hotel Dieu de France

🇱🇧

Beirut, Lebanon

Institut Bergonié

🇫🇷

Bordeaux, France

Hôpital Morvan

🇫🇷

Brest, France

Centre Georges François Leclerc

🇫🇷

Dijon, France

Clinique Pasteur

🇫🇷

Evreux, France

Centre Hospitalier de Gap

🇫🇷

Gap, France

Clinique Armoricaine de Radiologie

🇫🇷

Saint Brieuc, France

Hôpital Tenon

🇫🇷

Paris, France

Centre René Huguenin

🇫🇷

Saint-Cloud, France

Institut de Cancérologie de la Loire

🇫🇷

Saint-Priest-en-Jarez, France

Hôpital Saint-Joseph

🇱🇧

Jdeïdé, Lebanon

Centre Hospitalier Robert Boulin

🇫🇷

Libourne, France

Hôpital Bichat Claude Bernard

🇫🇷

Paris, France

Hôpital Charles Nicolle

🇫🇷

Rouen, France

Hôpital Robert Debré

🇫🇷

Reims, France

MD Anderson Cancer Center

🇺🇸

Orlando, Florida, United States

Ohio State University

🇺🇸

Columbus, Ohio, United States

The Emory Clinic

🇺🇸

Atlanta, Georgia, United States

Henry Ford Health System

🇺🇸

Detroit, Michigan, United States

Medical College of Wisconsin

🇺🇸

Milwaukee, Wisconsin, United States

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