MedPath

A Study to Evaluate Safety and Efficacy of BIIB091 in Participants With Relapsing Forms of Multiple Sclerosis

Phase 2
Recruiting
Conditions
Relapsing Forms of Multiple Sclerosis
Interventions
Drug: DRF
Drug: Placebo
Registration Number
NCT05798520
Lead Sponsor
Biogen
Brief Summary

The primary objectives are to investigate the safety and tolerability of BIIB091 monotherapy in participants with relapsing multiple sclerosis (RMS) (Part 1), and to evaluate the effects of BIIB091 combination therapy with Diroximel Fumarate (DRF) compared with the DRF monotherapy arm, on the key Magnetic Resonance Imaging (MRI) measure of active Central Nervous System (CNS) inflammation (Part 2). The secondary objectives are to evaluate the effects of BIIB091 monotherapy on the MRI measures of active CNS inflammation, to evaluate the effects of BIIB091 combination therapy with DRF compared with the DRF monotherapy arm on additional MRI measures of active CNS inflammation, to investigate the safety and tolerability of BIIB091 combination therapy with DRF in participants with RMS.

Detailed Description

Not available

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
275
Inclusion Criteria
  1. Diagnosis of RMS [relapsing-remitting multiple sclerosis (RRMS) or active secondary progressive multiple sclerosis (SPMS)] in accordance with the 2017 Revised McDonald criteria.

  2. Time since MS symptom onset is <20 years.

  3. Must have expanded disability status scale (EDSS) score of 0 through 5.0 at screening and baseline.

  4. Must have at least 1 of the following occurring prior to Baseline (Day 1):

    • ≥2 clinical relapses in the last 24 months (but not within 30 days prior to Baseline [Day 1]) with at least 1 relapse during the last 12 months prior to randomization.
    • ≥1 clinical relapse within the past 24 months (but not within 30 days prior to Baseline [Day 1]) and ≥1 new brain MRI lesion (Gd-positive and/or new or enlarging T2 hyperintense lesion) within the past 12 months prior to randomization. The screening MRI could be used to satisfy this criterion (if needed for inclusion, local reading is required). For new or enlarging T2 hyperintense lesions, the reference scan cannot be >12 months prior to randomization.
    • ≥1 GdE lesion on brain MRI within 6 months prior to randomization.

Key

Exclusion Criteria
  1. Diagnosis of primary progressive multiple sclerosis (PPMS) in accordance with the 2017 Revised McDonald criteria.

  2. An MS relapse that has occurred within 30 days prior to Baseline (Day 1) or the participant has not stabilized from a previous relapse at the time of screening.

  3. History of severe allergic, anaphylactic reactions or hypersensitivity reaction to BIIB091 or DRF, the excipients contained in the formulation, and if appropriate, any diagnostic agents to be administered during the study, including the following:

    • Known hypersensitivity to any components of the study treatment
    • Known hypersensitivity to previous fumarate or bruton's tyrosine kinase (BTK) inhibitor treatments
    • History of hypersensitivity to parenteral administration of Gd-based contrast agents
  4. Evidence of severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2) infection within the past 4 weeks prior to Baseline.

  5. History or positive test result at screening for human immunodeficiency virus (HIV).

  6. Current or history of hepatitis C infection regardless of viral load.

  7. Current or possible hepatitis B.

  8. Current enrollment or plan to enroll in any other drug, biological, device, clinical study, or treatment with an investigational drug or approved therapy for investigational use within 90 days prior to randomization or 5 half-lives of the drug or therapy, whichever is longer.

NOTE: Other protocol defined Inclusion/Exclusion criteria may apply.

Study & Design

Study Type
INTERVENTIONAL
Study Design
SEQUENTIAL
Arm && Interventions
GroupInterventionDescription
Part 1: BIIB091 Low Dose + Matching Placebo for DRFPlaceboParticipants will receive BIIB091 low dose and matching placebo for DRF, orally, for up to 48 weeks.
Part 1: BIIB091 High Dose + Matching Placebo for DRFPlaceboParticipants will receive BIIB091 high dose and matching placebo for DRF, orally, for up to 48 weeks.
Part 1: DRF + Matching Placebo for BIIB091DRFParticipants will receive DRF standard dose and matching placebo for BIIB091, orally, for up to 48 weeks.
Part 2: DRF + Matching Placebo for BIIB091DRFParticipants will receive DRF standard dose and matching placebo for BIIB091, orally, for up to 48 weeks.
Part 1: BIIB091 Low Dose + Matching Placebo for DRFBIIB091Participants will receive BIIB091 low dose and matching placebo for DRF, orally, for up to 48 weeks.
Part 2: BIIB091 + DRF Standard DoseDRFParticipants will receive selected dose of BIIB091 (based on Part 1 data) and DRF standard dose, orally, for up to 48 weeks.
Part 1: BIIB091 High Dose + Matching Placebo for DRFBIIB091Participants will receive BIIB091 high dose and matching placebo for DRF, orally, for up to 48 weeks.
Part 1: DRF + Matching Placebo for BIIB091PlaceboParticipants will receive DRF standard dose and matching placebo for BIIB091, orally, for up to 48 weeks.
Part 2: DRF + Matching Placebo for BIIB091PlaceboParticipants will receive DRF standard dose and matching placebo for BIIB091, orally, for up to 48 weeks.
Part 2: BIIB091 + DRF Low DoseDRFParticipants will receive selected dose of BIIB091 (based on Part 1 data) and DRF low dose, orally, for up to 48 weeks.
Part 2: BIIB091 + DRF Standard DoseBIIB091Participants will receive selected dose of BIIB091 (based on Part 1 data) and DRF standard dose, orally, for up to 48 weeks.
Part 2: BIIB091 + DRF Low DoseBIIB091Participants will receive selected dose of BIIB091 (based on Part 1 data) and DRF low dose, orally, for up to 48 weeks.
Primary Outcome Measures
NameTimeMethod
Part 2: Cumulative Number of New T1 Gadolinium-Enhancing (GdE) LesionsWeek 8 to Week 16
Part 1: Number of Participants With Adverse Events (AEs)Day 1 up to Week 50

An AE is any untoward medical occurrence in a participant or clinical investigation participant administered a pharmaceutical product and that does not necessarily have a causal relationship with this treatment. An AE can therefore be any unfavorable and unintended sign (including an abnormal laboratory finding), symptom, or disease temporally associated with the use of a medicinal (investigational) product or auxiliary medicinal product, whether or not related to the medicinal (investigational) product or auxiliary medicinal product.

Part 1: Number of Participants With Serious Adverse Events (SAEs)From signing the informed consent form (ICF) to Week 50

SAE is any untoward medical occurrence that at any dose results in death, in the view of the investigator, places the participant at immediate risk of death (a life-threatening event), requires inpatient hospitalization or prolongation of existing hospitalization, results in persistent or significant disability/incapacity, results in a congenital anomaly/birth defect or is a medically important event.

Secondary Outcome Measures
NameTimeMethod
Part 1: Cumulative Number of New T1 Gadolinium-Enhancing (GdE) LesionsWeek 8 to Week 16
Part 1: Number of Participants With Change From Baseline in Heart RateUp to Week 50
Part 2: Number of Participants With AEsDay 1 up to Week 50

An AE is any untoward medical occurrence in a participant or clinical investigation participant administered a pharmaceutical product and that does not necessarily have a causal relationship with this treatment. An AE can therefore be any unfavorable and unintended sign (including an abnormal laboratory finding), symptom, or disease temporally associated with the use of a medicinal (investigational) product or auxiliary medicinal product, whether or not related to the medicinal (investigational) product or auxiliary medicinal product.

Part 1: Cumulative Number of New or Enlarging T2 Hyperintense LesionsWeek 8 to Week 16
Part 1: Cumulative Volume of New or Enlarging T2 Hyperintense LesionsWeek 8 to Week 16
Part 1: Mean Change From Baseline in QT Interval Corrected for Heart Rate Using Fridericia's Formula (QTcF), RR, PR, QRS, and QT IntervalsUp to Week 50
Part 2: Cumulative Volume of New or Enlarging T2 Hyperintense LesionsWeek 8 to Week 16
Part 2: Number of Participants With SAEsFrom signing of ICF up to Week 50

SAE is any untoward medical occurrence that at any dose results in death, in the view of the investigator, places the participant at immediate risk of death (a life-threatening event), requires inpatient hospitalization or prolongation of existing hospitalization, results in persistent or significant disability/incapacity, results in a congenital anomaly/birth defect or is a medically important event.

Part 2: Number of Participants With Change From Baseline in QTcF, RR, PR, QRS, and QT intervalsUp to Week 50
Part 2: Number of Participants With Change From Baseline in Heart RateUp to Week 50
Part 2: Number of Participants With ECG Abnormalities as Assessed by 12-Lead ECG MeasurementsUp to Week 50
Part 1: Number of Participants With Clinically Significant Electrocardiogram (ECG) AbnormalitiesUp to Week 50
Part 2: Cumulative Number of New or Enlarging T2 Hyperintense LesionsWeek 8 to Week 16

Trial Locations

Locations (77)

Vanderbilt MS Center

🇺🇸

Nashville, Tennessee, United States

HonorHealth Neurology

🇺🇸

Scottsdale, Arizona, United States

Alta Bates Summit Medical Center

🇺🇸

Berkeley, California, United States

University of California at Irvine Medical Center

🇺🇸

Orange, California, United States

University of Colorado School of Medic

🇺🇸

Aurora, Colorado, United States

University of Miami Miller School of Medicine

🇺🇸

Miami, Florida, United States

University of South Florida

🇺🇸

Tampa, Florida, United States

Vero Beach Neurology and Research Institute

🇺🇸

Vero Beach, Florida, United States

Fort Wayne Neurological Center

🇺🇸

Fort Wayne, Indiana, United States

University of Kansas Medical Center Research Institute, Inc.

🇺🇸

Kansas City, Kansas, United States

International Neurorehabilitation Institute

🇺🇸

Lutherville, Maryland, United States

Washington University

🇺🇸

Saint Louis, Missouri, United States

Holy Name

🇺🇸

Teaneck, New Jersey, United States

University of New Mexico

🇺🇸

Albuquerque, New Mexico, United States

South Shore Neurologic Associates, P.C.

🇺🇸

Patchogue, New York, United States

Wake Forest University - School of Medicine - Central

🇺🇸

Winston-Salem, North Carolina, United States

University of Cincinnati Physicians Company

🇺🇸

Cincinnati, Ohio, United States

The Cleveland Clinic Foundation

🇺🇸

Cleveland, Ohio, United States

The Boster Center for Multiple Sclerosis

🇺🇸

Columbus, Ohio, United States

Neurology Clinic, PC

🇺🇸

Cordova, Tennessee, United States

The University of Texas Health Science Center San Antonio

🇺🇸

San Antonio, Texas, United States

University of Wisconsin Hospital and Clinics

🇺🇸

Madison, Wisconsin, United States

The Medical College of Wisconsin

🇺🇸

Milwaukee, Wisconsin, United States

'MHAT Avis - Medica' OOD

🇧🇬

Pleven, Bulgaria

UMHAT 'Dr. Georgi Stranski', EAD

🇧🇬

Pleven, Bulgaria

UMHAT 'Sv. Georgi', EAD

🇧🇬

Plovdiv, Bulgaria

MHATNP 'Sv.Naum', EAD

🇧🇬

Sofia, Bulgaria

University First MHAT-Sofia, 'St. Joan Krastitel' EAD

🇧🇬

Sofia, Bulgaria

Acibadem City Clinic Tokuda University Hospital Ead

🇧🇬

Sofia, Bulgaria

DCC Neoclinic EAD

🇧🇬

Sofia, Bulgaria

UMHAT "Sv. Ivan Rilski", EAD

🇧🇬

Sofia, Bulgaria

Diagnostic Consultation Center CONVEX EOOD

🇧🇬

Sofia, Bulgaria

Fakultni nemocnice u sv. Anny v Brne

🇨🇿

Brno, Czechia

Fakultni nemocnice Hradec Kralove

🇨🇿

Hradec Kralove, Czechia

Nemocnice Jihlava p.o.

🇨🇿

Jihlava, Czechia

Fakultni Thomayerova nemocnice

🇨🇿

Praha 4-Krc, Czechia

Krajska zdravotni a.s. - Nemocnice Teplice o.z.

🇨🇿

Teplice, Czechia

Studienzentrum fur Neurologie und Psychiatrie

🇩🇪

Boeblingen, Baden Wuerttemberg, Germany

Klinikum Bayreuth GmbH- Hohe Warte

🇩🇪

Bayreuth, Bayern, Germany

Neuropraxis Muenchen Sued

🇩🇪

Unterhaching, Bayern, Germany

Universitaetsklinikum Duesseldorf AoeR

🇩🇪

Duesseldorf, Nordrhein Westfalen, Germany

ZNS - Zentrum fuer Neurologisch-Psychiatrische Studien

🇩🇪

Siegen, Nordrhein Westfalen, Germany

Universitaetsklinikum Carl Gustav Carus TU Dresden

🇩🇪

Dresden, Germany

I.R.C.C.S. Neuromed-Istituto Neurologico Mediterraneo

🇮🇹

Pozzilli, Isernia, Italy

Fondazione Istituto G.Giglio di Cefalù

🇮🇹

Cefalù, Palermo, Italy

IRCCS Ospedale Policlinico San Martino

🇮🇹

Genova, Italy

Azienda Ospedaliera Universitaria- Università degli Studi della Campania "Luigi Vanvitelli"

🇮🇹

Napoli, Italy

Fondazione Istituto Neurologico Casimiro Mondino

🇮🇹

Pavia, Italy

Azienda Ospedaliera Universitaria Policlinico Tor Vergata

🇮🇹

Roma, Italy

Azienda Ospedaliera Universitaria Policlinico Umberto I - Università di Roma La Sapienza

🇮🇹

Roma, Italy

COPERNICUS Podmiot Leczniczy Sp. z o. o.,

🇵🇱

Gdansk, Poland

Samodzielny Publiczny Specjalistyczny Szpital Zachodni im. Jana Pawla II

🇵🇱

Grodzisk Mazowiecki, Poland

Centrum Medyczne Pratia Katowice

🇵🇱

Katowice, Poland

M.A. - LEK A.M.Maciejowscy SC.

🇵🇱

Katowice, Poland

Nzoz Novo-Med

🇵🇱

Katowice, Poland

Resmedica Sp.z o.o

🇵🇱

Kielce, Poland

Szpital Uniwersytecki w Krakowie

🇵🇱

Krakow, Poland

Centrum Neurologii K. Selmaj

🇵🇱

Lodz, Poland

Instytut Zdrowia dr Boczarska-Jedynak sp.z.o.o, Sp.K

🇵🇱

Oswiecim, Poland

Med-Polonia Sp. z o.o.

🇵🇱

Poznan, Poland

NZOZ 'NEURO-KARD', 'Ilkowski i Partnerzy' Sp. Partn. Lek.

🇵🇱

Poznan, Poland

Nzoz Palomed

🇵🇱

Rzeszów, Poland

NeuroProtect Sp. z o.o.

🇵🇱

Warszawa, Poland

Wielospecjalistyczne Centrum Medyczne Ibismed

🇵🇱

Zabrze, Poland

Caribbean Center for Clinical Research

🇵🇷

Guaynabo, Puerto Rico

Spitalul Universitar de Urgenta Elias

🇷🇴

Bucuresti, Romania

S.C Neurocity S.R.L

🇷🇴

București, Romania

S.C Clubul Sanatatii SRL

🇷🇴

Campulung Muscel, Romania

Hospital Universitario Quironsalud Madrid

🇪🇸

Pozuelo de Alarcon, Madrid, Spain

Hospital Universitario Virgen de la Arrixaca

🇪🇸

El Palmar, Murcia, Spain

Hospital del Mar

🇪🇸

Barcelona, Spain

Hospital Universitario Reina Sofia

🇪🇸

Cordoba, Spain

Hospital Universitario Ramon y Cajal

🇪🇸

Madrid, Spain

Hospital Regional Universitario de Malaga

🇪🇸

Malaga, Spain

Ospedale Regionale di Lugano

🇨🇭

Lugano, Ticino, Switzerland

Inselspital - Universitaetsspital Bern

🇨🇭

Bern, Switzerland

Universitaetsspital Zuerich

🇨🇭

Zuerich, Switzerland

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