MedPath

Body Weight, Sleep, and Heart Health

Early Phase 1
Completed
Conditions
Obesity
Circadian Dysregulation
Cardiovascular Risk Factor
Interventions
Radiation: PET Imaging
Behavioral: Circadian Study Protocol
Drug: 11C-Meta-Hydroxyephedrine (mHED)
Drug: 11C-CGP12177
Drug: O15-water
Registration Number
NCT03388788
Lead Sponsor
Oregon Health and Science University
Brief Summary

A multidisciplinary investigation examining the circadian mechanisms regulating cardiovascular (CV) risk in obesity. Specifically, in a valid circadian protocol, the investigators aim to study resting cardiovascular risk markers and the reactivity of circadian rhythms in these risk markers to standardized stressors in obesity. Furthermore, using an ingenious approach, the investigators propose to explore impairment in pre/post synaptic function in the cardiac left ventricle.

Detailed Description

Overall, these studies will help us answer whether CV rhythms predispose obese individuals to increased CV disease risk - particularly around the vulnerable morning period. The results will serve as a foundation for clinical trials of appropriately timed dosing of medications targeting aspects of the CV system in obesity that increase effectiveness while decreasing side-effects.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
16
Inclusion Criteria
  • Ages 25-65
  • Lean and overweight (BMI 18.5-40kg/m2)
  • Habitually sedentary
Exclusion Criteria
  • History of smoking/tobacco use
  • Insomnia
  • Moderate to severe obstructive sleep apnea.
  • Prior shift work within 6 months prior to the study.
  • Prescription medications
  • Drugs of abuse
  • Acute, chronic, or debilitating medical condition (including diabetes, hypertension, and metabolic syndrome)

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Normal WeightPET ImagingHealthy lean controls \[18.5\<BMI\<25 kg/m2 and WC \<94/80 (men and women respectively)\] will participate in a 5-day circadian study protocol with PET imaging using radiopharmaceuticals (11C-meta-hydroxyephedrine, 11C-CGP12177, and O15-water).
Normal Weight11C-Meta-Hydroxyephedrine (mHED)Healthy lean controls \[18.5\<BMI\<25 kg/m2 and WC \<94/80 (men and women respectively)\] will participate in a 5-day circadian study protocol with PET imaging using radiopharmaceuticals (11C-meta-hydroxyephedrine, 11C-CGP12177, and O15-water).
OverweightCircadian Study ProtocolHealthy obese \[30≤BMI\<40 and waist circumference (WC) ≥94/80 (men and women respectively)\] will participate in a 5-day circadian study protocol with PET imaging using radiopharmaceuticals (11C-meta-hydroxyephedrine, 11C-CGP12177, and O15-water).
OverweightO15-waterHealthy obese \[30≤BMI\<40 and waist circumference (WC) ≥94/80 (men and women respectively)\] will participate in a 5-day circadian study protocol with PET imaging using radiopharmaceuticals (11C-meta-hydroxyephedrine, 11C-CGP12177, and O15-water).
Normal WeightO15-waterHealthy lean controls \[18.5\<BMI\<25 kg/m2 and WC \<94/80 (men and women respectively)\] will participate in a 5-day circadian study protocol with PET imaging using radiopharmaceuticals (11C-meta-hydroxyephedrine, 11C-CGP12177, and O15-water).
Overweight11C-Meta-Hydroxyephedrine (mHED)Healthy obese \[30≤BMI\<40 and waist circumference (WC) ≥94/80 (men and women respectively)\] will participate in a 5-day circadian study protocol with PET imaging using radiopharmaceuticals (11C-meta-hydroxyephedrine, 11C-CGP12177, and O15-water).
OverweightPET ImagingHealthy obese \[30≤BMI\<40 and waist circumference (WC) ≥94/80 (men and women respectively)\] will participate in a 5-day circadian study protocol with PET imaging using radiopharmaceuticals (11C-meta-hydroxyephedrine, 11C-CGP12177, and O15-water).
Normal WeightCircadian Study ProtocolHealthy lean controls \[18.5\<BMI\<25 kg/m2 and WC \<94/80 (men and women respectively)\] will participate in a 5-day circadian study protocol with PET imaging using radiopharmaceuticals (11C-meta-hydroxyephedrine, 11C-CGP12177, and O15-water).
Normal Weight11C-CGP12177Healthy lean controls \[18.5\<BMI\<25 kg/m2 and WC \<94/80 (men and women respectively)\] will participate in a 5-day circadian study protocol with PET imaging using radiopharmaceuticals (11C-meta-hydroxyephedrine, 11C-CGP12177, and O15-water).
Overweight11C-CGP12177Healthy obese \[30≤BMI\<40 and waist circumference (WC) ≥94/80 (men and women respectively)\] will participate in a 5-day circadian study protocol with PET imaging using radiopharmaceuticals (11C-meta-hydroxyephedrine, 11C-CGP12177, and O15-water).
Primary Outcome Measures
NameTimeMethod
Blood Pressure5 Days

Beat-by-beat and ambulatory blood pressure measurements.

Secondary Outcome Measures
NameTimeMethod
Heart Rate5 Days

Heart rate via 2-channel echocardiogram (ECG)

Norepinephrine5 days

Venous Norepinephrine to estimate sympathetic output

Heart Rate Variability (HRV)5 days

Analysis of HRV from 12-lead ECG to assess parasympathetic activity

Aldosterone5 days

Venous Aldosterone to estimate sympathetic output

Norepinephrine reuptake transport5 days.

Radiolabeled meta-hydroxyephedrine (11C-mHED) to measure norepinephrine reuptake during PET Imaging.

Beta-adrenergic receptor density5 days.

Radiolabeled agonist (11C-CGP12177) to measure beta-adrenergic receptors during PET Imaging.

Dual Emission X-ray Absorbance (DEXA) Body composition1 day

DEXA imaging to assess body composition.

Coronary Artery Calcium Score1 scan.

Coronary Calcium Computed Tomography (CT) Scan

Tumor Necrosis Factor alpha (TNF-alpha)5 days

TNF-alpha to assess inflammation.

Coronary blood flow5 days.

Radiolabeled water (O15-water) to measure coronary blood flow during PET Imaging.

Epinephrine5 days

Venous Epinephrine to estimate sympathetic output

Cortisol5 days

Saliva cortisol to estimate sympathetic output

malondialdehyde (MDA) adducts5 days

Plasma MDA to measure oxidative stress and inflammation.

Flow Mediated Dilation (FMD)5 days

FMD to measure endothelial function.

Coronary Microvascular Blood Flux3 days

1. Determine in lean healthy humans if coronary microvascular function, measured as coronary microvascular blood flux, has an endogenous circadian rhythm with lowest function in the morning. 2. Test the hypothesis that people with obesity have impaired coronary microvascular blood flux compared to lean individuals, with the exaggerated impairment during the morning. Measured using myocardial contrast echocardiography.

Endocannabinoid5 days

Plasma endocannabinoid to estimate sympathetic regulation

Trial Locations

Locations (1)

Oregon Health & Science University

🇺🇸

Portland, Oregon, United States

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