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A study to determine the safety, tolerability and process by which ibuprofen is absorbed, distributed, metabolized, and eliminated by the body over a 5-7 minute infusion.

Phase 1
Completed
Conditions
Thrombophlebitis
Inflammatory and Immune System - Other inflammatory or immune system disorders
Registration Number
ACTRN12609000309280
Lead Sponsor
Cumberland Pharmaceuticals Incorparated
Brief Summary

Not available

Detailed Description

Not available

Recruitment & Eligibility

Status
Completed
Sex
All
Target Recruitment
12
Inclusion Criteria

Healthy volunteers between the ages of 18 and 65 years (at the time of consent).

Exclusion Criteria

Participants lacking good venous access in both arms.

History of allergy or hypersensitivity to Non-Steroidal Anti-Inflammatory Drugs (NSAIDs) or any component of intravenous ibuprofen.

Have never taken aspirin or ibuprofen

History of abuse of alcohol or other drugs in the 2 months before CTM administration.

Have used prescription drugs (not including oral contraceptives) within 14 days before CTM administration or have used aspirin within one week before CTM administration or over-the-counter pain relievers (NSAIDs or acetaminophen) within 3 days before CTM administration.

Have taken investigational drugs within 30 days before CTM administration.

Have donated blood or blood products within 30 days before CTM administration.

Be pregnant or nursing.

Have had breast cancer.

Have a clinically significant laboratory test

Presence or history of the following conditions: asthma, bleeding tendency, hypertension, heart failure, peptic ulcer disease, inflammatory bowel disease, or any other gastrointestinal disorder, renal or hepatic disease..

Have a calculated creatinine clearance(estimated by means of the
Cockcroft-Gault equation) of < 75mL/min

Inability to understand the requirements of the study. Participants must
be willing to provide written informed consent (as evidenced by
signature on an informed consent document approved by an Institutional Review Board [IRB]), and agree to abide by the study restrictions.

Refusal to provide written authorization for use and disclosure of protected health information

Be otherwise unsuitable for the study, in the opinion of the Investigator.

Study & Design

Study Type
Interventional
Study Design
Not specified
Primary Outcome Measures
NameTimeMethod
To evaluate the pharmacokinetic profile of a single dose of IVIb administered over 5-7 minutes by doing blood analysis.[Predose, Immediately after<br>completion of the intravenous Clinical Trial Material (CTM) administration then at Hours 0.25,<br>0.5, 0.75, 1, 1.5, 2, 2.5, 3, 4, 5, 6, 8, 10 and 12 hours after treatment.]
Secondary Outcome Measures
NameTimeMethod
To evaluate the safety and tolerability of a single dose of IVIb by assessing the<br>frequency, severity and duration of treatment-emergent adverse events,<br>including those related to the infusion site, in healthy adult participants who received a single dose of IVIb and oral placebo administration given concurrently as compared to a crossover oral ibuprofen and intravenous placebo administration. This will be done by frequently asking the volunteer non leading questions regarding there well-being, also visual observation looking for volunteer deteriation.<br>Adevrse Events iexamples: swelling and redness at infusion site, nausea and headache.[Predose, Immediately after<br>completion of the intravenous CTM administration then at Hours 0.5, 1, 2, 3, 4, 5, 6, 8, 10 and 12 hours after treatment.]
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