MedPath

TBTC Study 29: Rifapentine During Intensive Phase Tuberculosis (TB) Treatment

Phase 2
Completed
Conditions
Pulmonary Tuberculosis
Interventions
Registration Number
NCT00694629
Lead Sponsor
Centers for Disease Control and Prevention
Brief Summary

Protocol Synopsis The goal of this Phase 2 clinical trial is to evaluate the antimicrobial activity and safety of an experimental intensive phase (first 8 weeks of treatment) tuberculosis treatment regimen in which rifapentine is substituted for rifampin.

Primary Objective

* To compare the antimicrobial activity and safety of standard daily regimen comprised of rifampin (approximately 10 mg/kg/dose) + isoniazid + pyrazinamide + ethambutol (RHZE) to that of an experimental regimen comprised of rifapentine (approximately 10 mg/kg/dose) + isoniazid + pyrazinamide + ethambutol (PHZE).

Secondary Objectives

* To determine and compare for each regimen the time to culture-conversion, using data from 2-, 4-, 6-, and 8-week cultures (10, 20, 30, 40 doses).

* To determine and compare for each regimen the proportion of patients with any Grade 3 or 4 adverse reactions

* To determine the correlation of the MGIT/BACTEC liquid culture growth index and other mycobacterial and clinical biomarkers with time to culture conversion and treatment failure

* To store serum for future assessment of biomarkers of TB treatment response and hypersensitivity to study drugs.

* To compare adverse events and 2-month culture conversion rates among HIV-infected patients vs. HIV-uninfected patients

* To determine the tolerability and safety, and estimate the antimicrobial activity, of experimental regimens that include isoniazid + pyrazinamide + ethambutol plus either rifapentine 15 mg/kg/dose or rifapentine 20 mg/kg/dose, all administered daily. Assessment of these doses of rifapentine will be performed as an extension to the main study after enrollment in the main study has been completed.

Design

This will be a prospective, multicenter, open-label clinical study. Adults suspected of having pulmonary tuberculosis who meet eligibility criteria will be randomized to receive either the experimental intensive phase tuberculosis treatment regimen or the standard intensive phase tuberculosis treatment regimen. Randomization will be stratified by presence/absence of cavitation on baseline chest radiograph, and by geographic continent. All doses of study drugs will be given under direct observation and administered 5 days per week. After a subject completes intensive phase therapy, he/she then will be treated with a non-experimental continuation phase tuberculosis treatment regimen.

The study extension will be a prospective, multicenter clinical trial. Eligibility criteria will be the same as for the main study. Participants will be randomized to one of four regimens: the standard intensive phase treatment regimen, an investigational regimen in which rifapentine 10 mg/kg/dose is substituted for rifampin, an investigational regimen in which rifapentine 15 mg/kg/dose is substituted for rifampin, or an investigational regimen in which rifapentine 20 mg/kg is substituted for rifampin. Randomization will be stratified by the presence/absence of cavitation on baseline chest radiograph, and by study site. Study drugs will be administered 7 days per week. After a subject completes intensive phase therapy, he/she then will be treated with a non-experimental continuation phase tuberculosis treatment regimen. Subjects will have blood drawn for one pharmacokinetic determination of rifapentine concentration at or after the week 2 visit during intensive phase therapy.

This study is being conducted in 2 phases.

1. The main study compares a 10 mg/kg dose of rifapentine, open label, against 10 mg/kg rifampin in an otherwise standard intensive phase regimen of treatment for pulmonary tuberculosis. The projected sample size was 480 enrollments; 530 patients were actually enrolled.

2. The study extension evaluates higher doses of rifapentine, with the specific rifapentine doses (10 mg/kg, 15 mg/kg, and 20 mg/kg) blinded to patients and clinicians, with data collection and endpoints otherwise similar to the main study. The projected sample size for the study extension is 320 enrollments.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
865
Inclusion Criteria
  1. Suspected pulmonary tuberculosis with acid-fast bacilli in a stained smear of expectorated or induced sputum.

  2. Willingness to have HIV testing performed, if HIV serostatus is not known or if the last documented negative HIV test was more than 3 months prior to enrollment.

  3. 5 (five) or fewer days of multidrug therapy for tuberculosis disease in the 6 months preceding initiation of study drugs.

  4. 7 (seven) or fewer days of fluoroquinolone therapy in the 30 days preceding initiation of study drugs.

  5. Age >= 18 years

  6. Karnofsky score of at least 60 (requires occasional assistance but is able to care for most of his/her needs; see Appendix B)

  7. Signed informed consent

  8. Women of child-bearing potential must agree to practice an adequate (barrier) method of birth control or to abstain from heterosexual intercourse during study therapy.

  9. Laboratory parameters done within 14 days prior to, enrollment:

    • Serum or plasma alanine aminotransferase (ALT) activity ≤ 3 times the upper limit of normal
    • Serum or plasma total bilirubin level ≤ 2.5 times the upper limit of normal
    • Serum or plasma creatinine level ≤ 2 times the upper limit of normal
    • Complete blood count with hemoglobin level of at least 7.0 g/dL
    • Complete blood count with platelet count of at least 100,000/mm3
    • Negative pregnancy test (women of childbearing potential)
Exclusion Criteria
  1. Pregnant or breast-feeding
  2. Known intolerance or allergy to any of the study drugs
  3. Concomitant disorders or conditions for which isoniazid (INH), rifamycins, pyrazinamide (PZA), or ethambutol (EMB) are contraindicated. These include severe hepatic damage, acute liver disease of any cause, and acute uncontrolled gouty arthritis.
  4. Current or planned therapy, during the intensive phase of TB therapy, with combination antiretroviral therapy for HIV, or with cyclosporine or tacrolimus. Cyclosporine and tacrolimus have unacceptable interactions with rifamycins.
  5. Pulmonary silicosis
  6. Central nervous system TB
  7. Weight < 40 kg or > 85 kg

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
4rifapentinerifapentine 20 mg/kg, isoniazid, pyrazinamide, ethambutol
1rifampinrifampin, isoniazid, pyrazinamide, ethambutol
2rifapentinerifapentine 10 mg/kg, isoniazid, pyrazinamide, ethambutol
3rifapentinerifapentine 15 mg/kg, isoniazid, pyrazinamide, ethambutol
Primary Outcome Measures
NameTimeMethod
The proportion of patients, by regimen, having negative sputum cultures at completion of eight weeks (40 doses) of treatmentcompletion of eight weeks (40 doses) of treatment
The proportion of patients, by regimen, who permanently discontinue the assigned study treatment for any reason during the first eight weeksduring the first eight weeks of treatment
Secondary Outcome Measures
NameTimeMethod
compare adverse events and 2-month culture conversion rates among HIV-infected patients vs. HIV-uninfected patients8 weeks
correlation of the MGIT/BACTEC liquid culture growth index and other mycobacterial and clinical biomarkers with time to culture conversion and treatment failureduration of TB treatment
time to culture-conversion2-, 4-, 6-, and 8-week cultures (10, 20, 30, 40 doses)
proportion of patients with any Grade 3 or 4 adverse reactions8 weeks
• To determine the tolerability and safety, and estimate the antimicrobial activity, of experimental regimens that include higher doses of rifapentine.8 weeks.

• To determine the tolerability and safety, and estimate the antimicrobial activity, of experimental regimens that include isoniazid + pyrazinamide + ethambutol plus either rifapentine 15 mg/kg/dose or rifapentine 20 mg/kg/dose, all administered daily. Assessment of these doses of rifapentine will be performed as an extension to the main study after enrollment in the main study has been completed.

Trial Locations

Locations (29)

Washington DC Veterans Administration Medical Center

🇺🇸

Washington DC, District of Columbia, United States

Agencia de Salut Publica

🇪🇸

Barcelona, Spain

University of North Texas Health Science Center

🇺🇸

Fort Worth, Texas, United States

LA County/USC Medical Center

🇺🇸

Los Angeles, California, United States

University of Southern California Medical Center

🇺🇸

Los Angeles, California, United States

Emory University School of Medicine

🇺🇸

Atlanta, Georgia, United States

Duke University Medical Center

🇺🇸

Durham, North Carolina, United States

Veterans Administration Tennessee Valley Health Care System

🇺🇸

Nashville, Tennessee, United States

Houston Veterans Administration Medical Center

🇺🇸

Houston, Texas, United States

Audi L. Murphy VA Hospital

🇺🇸

San Antonio, Texas, United States

Seattle King County Health Department

🇺🇸

Seattle, Washington, United States

Makerere University Medical School

🇺🇬

Kampala, Uganda

University of Manitoba

🇨🇦

Winnepeg, Manitoba, Canada

Denver Department of Public Health and Hospitals

🇺🇸

Denver, Colorado, United States

Boston Medical Center

🇺🇸

Boston, Massachusetts, United States

Central Arkansas Veterans Health System

🇺🇸

Little Rock, Arkansas, United States

University of California, San Francincisco

🇺🇸

San Francisco, California, United States

University of California at San Diego

🇺🇸

San Diego, California, United States

Chicago VA Medical Center (Lakeside)

🇺🇸

Chicago, Illinois, United States

Northwestern University

🇺🇸

Chicago, Illinois, United States

Hines VA Medical Center

🇺🇸

Hines, Illinois, United States

Johns Hopkins University School of Medicine

🇺🇸

Baltimore, Maryland, United States

New Jersey Medical School

🇺🇸

Newark, New Jersey, United States

Columbia University/Presbyterian Medical Center

🇺🇸

New York, New York, United States

Harlem Hospital, Columbia University

🇺🇸

New York, New York, United States

Nashville VA Medical Center

🇺🇸

Nashville, Tennessee, United States

Hopital Universitario Clementino Fraga Filho

🇧🇷

Rio de Janeiro, Brazil

Montreal Chest Institute McGill University

🇨🇦

Montreal, Quebec, Canada

Nelson R Mandela School of Medicine

🇿🇦

Durban, KwaZulu Natal, South Africa

© Copyright 2025. All Rights Reserved by MedPath