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A Study of Evacetrapib (LY2484595) in Participants With High Cholesterol

Phase 3
Terminated
Conditions
Hyperlipidemia
Interventions
Registration Number
NCT02227784
Lead Sponsor
Eli Lilly and Company
Brief Summary

The purpose of the ACCENTUATE study is to evaluate whether the study drug known as evacetrapib is effective in treating participants with high cholesterol and atherosclerotic cardiovascular disease (ASCVD) and/or diabetes.

Detailed Description

Not available

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
366
Inclusion Criteria
  • Must be treated with atorvastatin 40 mg/day for at least 30 days prior to screening
  • Have an LDL-C >70 mg/deciliter(dL) or non-HDL-C >100 mg/dL
  • Have screening triglycerides ≤400 mg/dL (≤4.5 millimoles/Liter)
  • Individuals with ASCVD and/or individuals with type 1 or type 2 diabetes
Exclusion Criteria
  • Have a hemoglobin A1c (HbA1c) >9.5%
  • New York Heart Association (NYHA) class III or IV congestive heart failure
  • History of either a transient ischemic stroke or ischemic stroke <30 days
  • History of acute coronary syndrome (ACS) <30 days

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Atorvastatin + EvacetrapibEvacetrapibAtorvastatin 40 milligrams (mg) orally once daily for 28 days during lead in period. Atorvastatin 40 mg plus evacetrapib 130 mg with placebo for blinding orally once daily for 90 days. Open label extension (atorvastatin 40 mg plus evacetrapib 130 mg) is available for compliant participants.
Atorvastatin + EvacetrapibPlaceboAtorvastatin 40 milligrams (mg) orally once daily for 28 days during lead in period. Atorvastatin 40 mg plus evacetrapib 130 mg with placebo for blinding orally once daily for 90 days. Open label extension (atorvastatin 40 mg plus evacetrapib 130 mg) is available for compliant participants.
Atorvastatin 80 mgAtorvastatinAtorvastatin 40 mg orally once daily for 28 days during lead in period. Atorvastatin 80 mg orally with placebo for blinding once daily for 90 days. Open label extension (atorvastatin 40 mg plus evacetrapib 130 mg) is available for compliant participants.
Atorvastatin 80 mgPlaceboAtorvastatin 40 mg orally once daily for 28 days during lead in period. Atorvastatin 80 mg orally with placebo for blinding once daily for 90 days. Open label extension (atorvastatin 40 mg plus evacetrapib 130 mg) is available for compliant participants.
Atorvastatin + EzetimibeAtorvastatinAtorvastatin 40 mg orally once daily for 28 days during lead in period. Atorvastatin 40 mg plus ezetimibe 10 mg with placebo for blinding orally once daily for 90 days. Open label extension (atorvastatin 40 mg plus evacetrapib 130 mg) is available for compliant participants.
Atorvastatin + EzetimibePlaceboAtorvastatin 40 mg orally once daily for 28 days during lead in period. Atorvastatin 40 mg plus ezetimibe 10 mg with placebo for blinding orally once daily for 90 days. Open label extension (atorvastatin 40 mg plus evacetrapib 130 mg) is available for compliant participants.
Atorvastatin 40 mgPlaceboAtorvastatin 40 mg orally once daily for 28 days during lead in period. Atorvastatin 40 mg with placebo for blinding orally once daily for 90 days. Open label extension (atorvastatin 40 mg plus evacetrapib 130 mg) is available for compliant participants.
Atorvastatin + EvacetrapibAtorvastatinAtorvastatin 40 milligrams (mg) orally once daily for 28 days during lead in period. Atorvastatin 40 mg plus evacetrapib 130 mg with placebo for blinding orally once daily for 90 days. Open label extension (atorvastatin 40 mg plus evacetrapib 130 mg) is available for compliant participants.
Atorvastatin + EzetimibeEzetimibeAtorvastatin 40 mg orally once daily for 28 days during lead in period. Atorvastatin 40 mg plus ezetimibe 10 mg with placebo for blinding orally once daily for 90 days. Open label extension (atorvastatin 40 mg plus evacetrapib 130 mg) is available for compliant participants.
Atorvastatin 40 mgAtorvastatinAtorvastatin 40 mg orally once daily for 28 days during lead in period. Atorvastatin 40 mg with placebo for blinding orally once daily for 90 days. Open label extension (atorvastatin 40 mg plus evacetrapib 130 mg) is available for compliant participants.
Primary Outcome Measures
NameTimeMethod
Percent Change From Baseline to 3 Months in Low-Density Lipoprotein Cholesterol (LDL-C)Baseline, 3 Months

Change in LDL-C levels from baseline to the 3-month visit expressed as a percentage of the baseline levels. LDL-C was measured by beta quantification. Statistics are from analysis of covariance with log baseline measurement and treatment is included in the model. Least Square Means (LS means) and median differences were analyzed in log units and converted to standard units. Log Percent change from baseline response is the dependent variable.

Secondary Outcome Measures
NameTimeMethod
Percent Change From Baseline to 3 Months in High-Density Lipoprotein Cholesterol (HDL-C)Baseline, 3 Months

Change in HDL-C levels from baseline to the 3-month visit expressed as a percentage of the baseline levels. LS medians and median differences were analyzed in log units and converted to standard units. Statistics are from mixed model repeated measures analysis with log baseline measurement, treatment, visit, and treatment by visit interaction included in the model. Log percent change from baseline response is the dependent variable. Within-participant repeated measures at multiple visits are modeled by a compound symmetry covariance structure.

Percent Change From Baseline to 3 Months in Apolipoprotein AI (apoAI)Baseline, 3 Months

Change in apoAI levels from baseline to the 3-month visit expressed as a percentage of the baseline levels. Statistics are from analysis of covariance with log baseline measurement and treatment is included in the model. LS means and median differences were analyzed in log units and converted to standard units. Log Percent change from baseline response is the dependent variable.

Percent Change From Baseline to 3 Months in Non-HDL-CBaseline, 3 Months

Change in Non-HDL-C levels from baseline to the 3-month visit expressed as a percentage of the baseline levels. LS medians and median differences were analyzed in log units and converted to standard units. Statistics are from mixed model repeated measures analysis with log baseline measurement, treatment, visit, and treatment by visit interaction included in the model. Log percent change from baseline response is the dependent variable. Within-participant repeated measures at multiple visits are modeled by a compound symmetry covariance structure.

Percent Change From Baseline to 3 Months in Apolipoprotein B (apoB)Baseline, 3 Months

Change in apoB levels from baseline to the 3-month visit expressed as a percentage of the baseline levels. Statistics are from analysis of covariance with log baseline measurement and treatment is included in the model. LS means and median differences were analyzed in log units and converted to standard units. Log Percent change from baseline response is the dependent variable.

Percent Change From Baseline to 3 Months in Cholesterol Efflux CapacityBaseline, 3 Months

Change in cholesterol efflux capacity from baseline to the 3-month visit expressed as a percentage of the baseline levels. Statistics are from analysis of covariance with log baseline measurement and treatment is included in the model. LS means and median differences were analyzed in log units and converted to standard units. Log Percent change from baseline response is the dependent variable.

Percent Change From Baseline to 3 Months in Lipoprotein(a) (Lp[a])Baseline, 3 Months

Change in Lp(a) levels from baseline to the 3-month visit expressed as a percentage of the baseline levels. Statistics are from analysis of covariance with log baseline measurement and treatment is included in the model. LS means and median differences were analyzed in log units and converted to standard units. Log Percent change from baseline response is the dependent variable.

Trial Locations

Locations (63)

Alan Graff, MD, PA

🇺🇸

Fort Lauderdale, Florida, United States

Northwest Heart Clinical Research, LLC

🇺🇸

Arlington Heights, Illinois, United States

Maryland Cardiovascular Specialists

🇺🇸

Baltimore, Maryland, United States

Northwest Houston Heart Center

🇺🇸

Tomball, Texas, United States

Overlea Personal Physicians

🇺🇸

Baltimore, Maryland, United States

Holston Medical Group Clinical Research

🇺🇸

Kingsport, Tennessee, United States

Clinical Investigation Specialists Inc

🇺🇸

Kenosha, Wisconsin, United States

Palm Research Center

🇺🇸

Las Vegas, Nevada, United States

University Clinical Investigators, Inc.

🇺🇸

Tustin, California, United States

Midwest Institute for Clinical Research

🇺🇸

Indianapolis, Indiana, United States

Cedar-Crosse Research Center

🇺🇸

Chicago, Illinois, United States

Aventiv Research

🇺🇸

Columbus, Ohio, United States

Suncoast Research Group, LLC

🇺🇸

Miami, Florida, United States

Indiana Heart Physicians Inc

🇺🇸

Indianapolis, Indiana, United States

Nature Coast Clinical Research, LLC

🇺🇸

Inverness, Florida, United States

Georgia Heart Specialists

🇺🇸

Covington, Georgia, United States

Heart and Vascular Center of New Brunswick LLC

🇺🇸

Somerset, New Jersey, United States

Encompass Clinical Research

🇺🇸

Spring Valley, California, United States

Advanced Clinical Research

🇺🇸

Carmichael, California, United States

Tooraj Joseph Raoof M.D., Inc.

🇺🇸

Encino, California, United States

Diablo Clinical Research

🇺🇸

Walnut Creek, California, United States

United Osteoporosis Center

🇺🇸

Gainesville, Georgia, United States

Cardiac Research

🇺🇸

Colorado Springs, Colorado, United States

Desert Clinical Research

🇺🇸

Mesa, Arizona, United States

Progressive Medical Research

🇺🇸

Port Orange, Florida, United States

Cape Cod Research Institute

🇺🇸

Hyannis, Massachusetts, United States

Metrolina Internal Medicine, P.A.

🇺🇸

Charlotte, North Carolina, United States

High Point Clinical Trials Center

🇺🇸

High Point, North Carolina, United States

Midwest CRC

🇺🇸

Crystal Lake, Illinois, United States

Grace Research

🇺🇸

Bossier City, Louisiana, United States

GCM Medical Group PSC

🇵🇷

San Juan, Puerto Rico

Buffalo Cardiology and Pulmonary Associates, P.C.

🇺🇸

Williamsville, New York, United States

Lillestol Research LLC

🇺🇸

Fargo, North Dakota, United States

Solaris Clinical Research

🇺🇸

Meridian, Idaho, United States

Hutchinson Clinic

🇺🇸

Hutchinson, Kansas, United States

ActivMed Practices & Research, Inc

🇺🇸

Methuen, Massachusetts, United States

PMG Research of Wilmington, LLC

🇺🇸

Wilmington, North Carolina, United States

Partners in Clinical Research

🇺🇸

Cumberland, Rhode Island, United States

Clinical Research Puerto Rico, Inc.

🇵🇷

San Juan, Puerto Rico

Boice Willis Clinic, PA

🇺🇸

Rocky Mount, North Carolina, United States

Black Hills Cardiovascular Research Group

🇺🇸

Rapid City, South Dakota, United States

Research and Cardiovascular Corp.

🇵🇷

Ponce, Puerto Rico

PMG Research of Charleston, LLC

🇺🇸

Mount Pleasant, South Carolina, United States

Kootenai Heart Clinics, LLC

🇺🇸

Spokane, Washington, United States

Saratoga Clinical Research LLC

🇺🇸

Saratoga Springs, New York, United States

Irvine Clinical Research Center

🇺🇸

Irvine, California, United States

Rancho Cucamonga Clinical

🇺🇸

Rancho Cucamonga, California, United States

Central Phoenix Med Clinic LLC

🇺🇸

Phoenix, Arizona, United States

University of Colorado Health Sciences Center

🇺🇸

Aurora, Colorado, United States

South Oklahoma Heart Research, LLC

🇺🇸

Oklahoma City, Oklahoma, United States

Portland Preventive Cardiology, LLC

🇺🇸

Portland, Oregon, United States

Cardiology Research Assoc.

🇺🇸

Daytona Beach, Florida, United States

Heart Center Research, LLC

🇺🇸

Huntsville, Alabama, United States

VA Long Beach Healthcare System

🇺🇸

Long Beach, California, United States

Avail Clinical Research LLC

🇺🇸

DeLand, Florida, United States

Cardiology Partners Clinical Research Institute, LLC

🇺🇸

Wellington, Florida, United States

ZASA Clinical Research

🇺🇸

Boynton Beach, Florida, United States

Medex Healthcare Research, Inc.

🇺🇸

New York, New York, United States

Asheville Cardiology Associates

🇺🇸

Asheville, North Carolina, United States

Northwest Clinical Research Center

🇺🇸

Bellevue, Washington, United States

Community Medical Associates

🇺🇸

Louisville, Kentucky, United States

National Clinical Research - Richmond

🇺🇸

Richmond, Virginia, United States

East West Medical Institute

🇺🇸

Honolulu, Hawaii, United States

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