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Efficacy and Safety of Insulin Glargine/Lixisenatide Fixed Combination Versus Insulin Glargine Alone on Top of Metformin in Type 2 Diabetic Patients

Phase 2
Completed
Conditions
Type 2 Diabetes Mellitus
Interventions
Drug: Insulin glargine /lixisenatide Fixed Ratio Combination
Drug: Insulin glargine
Drug: Metformin (Background drug)
Registration Number
NCT01476475
Lead Sponsor
Sanofi
Brief Summary

Primary Objective:

* The purpose of this study was to compare insulin glargine/ lixisenatide fixed ratio combination (FRC) versus insulin glargine on glycemic control over 24 weeks, as evaluated by glycosylated hemoglobin (HbA1c) reduction in type 2 diabetic participants treated with metformin.

Secondary Objectives:

* To compare insulin glargine/lixisenatide FRC versus insulin glargine over 24 weeks on:

* Glycemic control in relation to a meal as evaluated by post-prandial plasma glucose and glucose excursions during a standardized meal test;

* Percentage of participants reaching HbA1c \<7% or ≤6.5%;

* 7-point Self-Monitored Plasma Glucose (SMPG) profile;

* Body weight;

* Insulin glargine dose

* Fasting Plasma Glucose (FPG);

* Percentage of participants requiring rescue therapy during the 24-week open label treatment period;

* To assess safety and tolerability of insulin glargine/lixisenatide FRC.

Detailed Description

Approximately 27 weeks including a 24-week treatment period.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
323
Inclusion Criteria

Not provided

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Exclusion Criteria

Not provided

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Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Insulin glargine/Lixisenatide Fixed Ratio Combination (FRC)Insulin glargine /lixisenatide Fixed Ratio CombinationFRC injected once daily (QD) for 24 weeks. Dose individually adjusted.
Insulin glargine/Lixisenatide Fixed Ratio Combination (FRC)Metformin (Background drug)FRC injected once daily (QD) for 24 weeks. Dose individually adjusted.
Insulin glargineMetformin (Background drug)Insulin glargine QD for 24 weeks. Dose individually adjusted.
Insulin glargineInsulin glargineInsulin glargine QD for 24 weeks. Dose individually adjusted.
Primary Outcome Measures
NameTimeMethod
Change in HbA1c From Baseline to Week 24Baseline, Week 24

Change in HbA1c was calculated by subtracting baseline value from Week 24 value. Missing data was imputed using last observation carried forward (LOCF). On-treatment period for this efficacy variable was defined as the time from the first dose of study drug till before the introduction of rescue medication and up to 14 days after the last injection of investigational medicinal product (IMP).

Secondary Outcome Measures
NameTimeMethod
Change in 2-hour Postprandial Plasma Glucose (PPG) From Baseline to Week 24Baseline, Week 24

The 2-hour PPG test measured blood glucose 2 hours after eating a standardized meal. Change in PPG was calculated by subtracting baseline value from Week 24 value. Missing data was imputed using LOCF. On-treatment period for this efficacy variable was defined as the time from the first dose of study drug till before the introduction of rescue medication and up to the date of last injection of IMP.

Change in 2-hour Plasma Glucose Excursion From Baseline to Week 24Baseline, Week 24

2-hour plasma glucose excursion = 2-hour PPG minus plasma glucose value obtained 30 minutes prior to the start of the meal and before IMP administration. Change in plasma glucose excursion was calculated by subtracting baseline value from Week 24 value. Missing data was imputed using LOCF. On-treatment period for this efficacy variable was defined as the time from the first dose of study drug till before the introduction of rescue medication and up to the date of last injection of IMP.

Change in Average 7-Point Self-Monitored Plasma Glucose (SMPG) Profiles From Baseline to Week 24Baseline, Week 24

Participants recorded a 7-point plasma glucose profile measured before and 2-hours after each meal and at bedtime, over a single day, once in a week before baseline, before visit Week 12 and before visit Week 24 and the average value across the profiles performed in the week before a visit for the 7-time points was calculated. Change in average 7-point SMPG was calculated by subtracting baseline value from Week 24 value. Missing data was imputed using LOCF. On-treatment period for this efficacy variable was defined as the time from the first dose of study drug till before the introduction of rescue medication and up to the date of last injection of IMP.

Change in Body Weight From Baseline to Week 24Baseline, Week 24

Change in body weight was calculated by subtracting baseline value from Week 24 value. Missing data was imputed using LOCF. On-treatment period for this efficacy variable was defined as the time from the first dose of study drug till before the introduction of rescue medication and up to 3 days after the last injection of IMP.

Average Daily Insulin Glargine Dose at Week 24Week 24

Missing data was imputed using LOCF. On-treatment period for this efficacy variable was defined as the time from the first dose of study drug till before the introduction of rescue medication and up to the date of last injection of IMP.

Change in FPG From Baseline to Week 24Baseline, Week 24

Change in FPG was calculated by subtracting baseline value from Week 24 value. Missing data was imputed using LOCF. On-treatment period for this efficacy variable was defined as the time from the first dose of study drug till before the introduction of rescue medication and up to 1 day after the last injection of IMP.

Percentage of Participants Requiring Rescue Therapy During 24-week Treatment PeriodBaseline up to Week 24

Routine fasting SMPG and central laboratory FPG (and HbA1c after Week 12) values were used to determine the requirement of rescue medication. If fasting SMPG value exceed the specified limit for 3 consecutive days, the central laboratory FPG (and HbA1c after Week 12) were performed. Threshold values from Week 8 to Week 12: fasting SMPG/FPG \>240 mg/dL (13.3 mmol/L), and from Week 12 to Week 30: fasting SMPG/FPG \>200 mg/dL (11.1 mmol/L) or HbA1c \>8%.

Percentage of Participants With HbA1c ≤6.5 % or <7.0 % at Week 24Week 24

On-treatment period for this efficacy variable was defined as the time from the first dose of study drug till before the introduction of rescue medication and up to 14 days after the last injection of IMP.

Change in 30-minute and 1-hour PPG From Baseline to Week 24Baseline, Week 24

The 30 minute and 1-hour PPG test measured blood glucose 30 minutes and 1-hour after eating a standardized meal. Change in PPG was calculated by subtracting baseline value from Week 24 value. Missing data was imputed using LOCF. On-treatment period for this efficacy variable was defined as the time from the first dose of study drug till before the introduction of rescue medication and up to the date of last injection of IMP.

Change in 30 Minute and 1-hour Plasma Glucose Excursion From Baseline to Week 24Baseline, Week 24

30-minute and 1-hour plasma glucose excursion = 30-minute and 1-hour PPG minus plasma glucose value obtained 30 minutes prior to the start of the meal and before IMP administration. Change in plasma glucose excursion was calculated by subtracting baseline value from Week 24 value. Missing data was imputed using LOCF. On-treatment period for this efficacy variable was defined as the time from the first dose of study drug till before the introduction of rescue medication and up to the date of last injection of IMP.

Percentage of Participants Reaching HbA1c <7% at Week 24 With no Documented Symptomatic Hypoglycemia During 24-week Treatment PeriodBaseline up to Week 24

Documented symptomatic hypoglycemia was an event during which typical symptoms of hypoglycemia were accompanied by a measured plasma glucose concentration of ≤70 mg/dL (3.9 mmol/L). Participants without any post-baseline on-treatment value for HbA1c were counted as non-responders if they experienced at least one documented symptomatic hypoglycemia before the introduction of rescue medication and up to 1 day after the last injection of IMP. Otherwise, they were counted as missing data. On-treatment period for this efficacy variable was defined as the time from the first dose of study drug till before the introduction of rescue medication and up to 14 days after the last injection of IMP.

Percentage of Participants Reaching HbA1c <7% With no Body Weight Gain at Week 24Week 24

Participants without any post-baseline on-treatment values (for HbA1c and body weight) that were no more than 30 days apart were counted as non-responders if at least one of the components (for HbA1c and body weight) was available and showed non-response. Otherwise, they were counted as missing data.

Percentage of Participants With Documented Symptomatic and Severe Symptomatic HypoglycemiaFirst dose of study drug up to 3 days after the last dose administration (maximum of 219 days)

Documented symptomatic hypoglycemia was an event during which typical symptoms of hypoglycemia were accompanied by a measured plasma glucose concentration of ≤70 mg/dL (3.9 mmol/L).Severe symptomatic hypoglycemia was an event requiring assistance of another person to actively administer carbohydrate, glucagon, or other resuscitative actions. These episodes were associated with sufficient neuroglycopenia to induce seizure, unconsciousness or coma. All episodes in which neurological impairment was severe enough to prevent self-treatment and which were thought to place participants at risk for injury to themselves or others.

Trial Locations

Locations (70)

Investigational Site Number 152403

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Santiago, Chile

Investigational Site Number 203401

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Plzen, Czech Republic

Investigational Site Number 203405

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Praha 8, Czech Republic

Investigational Site Number 348404

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Debrecen, Hungary

Investigational Site Number 703403

🇸🇰

Kosice, Slovakia

Investigational Site Number 703404

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Moldava Nad Bodvou, Slovakia

Investigational Site Number 152401

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Santiago, Chile

Investigational Site Number 642403

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Bucuresti, Romania

Investigational Site Number 703405

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Nitra, Slovakia

Investigational Site Number 840411

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Las Vegas, Nevada, United States

Investigational Site Number 208401

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København Nv, Denmark

Investigational Site Number 208404

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Køge, Denmark

Investigational Site Number 208402

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Slagelse, Denmark

Investigational Site Number 208403

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Svendborg, Denmark

Investigational Site Number 840401

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Larenceville, Georgia, United States

Investigational Site Number 840403

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Lexington, Kentucky, United States

Investigational Site Number 840407

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Medford, Oregon, United States

Investigational Site Number 840410

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Dallas, Texas, United States

Investigational Site Number 152405

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Santiago, Chile

Investigational Site Number 250402

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Narbonne, France

Investigational Site Number 250404

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Poitiers Cedex, France

Investigational Site Number 250401

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Vandoeuvre Les Nancy, France

Investigational Site Number 276403

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Oberhausen, Germany

Investigational Site Number 348405

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Budapest, Hungary

Investigational Site Number 348406

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Budapest, Hungary

Investigational Site Number 440402

🇱🇹

Kaunas, Lithuania

Investigational Site Number 484405

🇲🇽

Durango, Mexico

Investigational Site Number 616406

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Gdansk, Poland

Investigational Site Number 616403

🇵🇱

Krakow, Poland

Investigational Site Number 616404

🇵🇱

Pulawy, Poland

Investigational Site Number 616402

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Szczecin, Poland

Investigational Site Number 642404

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Timisoara, Romania

Investigational Site Number 752402

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Skellefteå, Sweden

Investigational Site Number 752403

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Växjö, Sweden

Investigational Site Number 840417

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Roswell, Georgia, United States

Investigational Site Number 840412

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Paramount, California, United States

Investigational Site Number 840404

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Hyattsville, Maryland, United States

Investigational Site Number 840405

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Rockville, Maryland, United States

Investigational Site Number 840408

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Little Rock, Arkansas, United States

Investigational Site Number 840415

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West Seneca, New York, United States

Investigational Site Number 840413

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Durham, Pennsylvania, United States

Investigational Site Number 840414

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Renton, Washington, United States

Investigational Site Number 152404

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Santiago, Chile

Investigational Site Number 203403

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Novy Jicin, Czech Republic

Investigational Site Number 152402

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Santiago, Chile

Investigational Site Number 203402

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Praha 2, Czech Republic

Investigational Site Number 440403

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Kedainiai, Lithuania

Investigational Site Number 276401

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Dresden, Germany

Investigational Site Number 276402

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Ludwigshafen, Germany

Investigational Site Number 348401

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Balatonfüred, Hungary

Investigational Site Number 484403

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Guadalajara, Mexico

Investigational Site Number 440401

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Kaunas, Lithuania

Investigational Site Number 440404

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Klaipeda, Lithuania

Investigational Site Number 616405

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Bialystok, Poland

Investigational Site Number 484401

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Cuernavaca, Mexico

Investigational Site Number 484402

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Guadalajara, Mexico

Investigational Site Number 616407

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Lodz, Poland

Investigational Site Number 642402

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Brasov, Romania

Investigational Site Number 616401

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Warszawa, Poland

Investigational Site Number 642405

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Iasi, Romania

Investigational Site Number 642406

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Targu Mures, Romania

Investigational Site Number 642401

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Oradea, Romania

Investigational Site Number 703402

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Bratislava, Slovakia

Investigational Site Number 703406

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Kosice, Slovakia

Investigational Site Number 752401

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Stockholm, Sweden

Investigational Site Number 703401

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Zilina, Slovakia

Investigational Site Number 840402

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Norman, Oklahoma, United States

Investigational Site Number 348402

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Szeged, Hungary

Investigational Site Number 348403

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Szeged, Hungary

Investigational Site Number 484404

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Acapulco, Mexico

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