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A Study of LY3372689 to Assess the Safety, Tolerability, and Efficacy in Participants With Alzheimer's Disease

Phase 2
Active, not recruiting
Conditions
Alzheimer Disease
Interventions
Drug: Placebo
Registration Number
NCT05063539
Lead Sponsor
Eli Lilly and Company
Brief Summary

The purpose of this study is to assess the safety, tolerability and effect of study drug LY3372689 in participants with early symptomatic Alzheimer's Disease

Detailed Description

Not available

Recruitment & Eligibility

Status
ACTIVE_NOT_RECRUITING
Sex
All
Target Recruitment
330
Inclusion Criteria
  • Gradual and progressive change in memory function reported by participants or informants for ≥ 6 months
  • MMSE score of 22 to 30 (inclusive) at baseline
  • CDR global score of 0.5 to 1.0 (inclusive), with a memory box score ≥0.5.
  • Meet 18F flortaucipir positron emission tomography (PET) scan (central analysis) criteria
  • Have a study partner who will provide written informed consent to participate
Exclusion Criteria
  • Contraindication to MRI or PET scans
  • Have known allergies to LY3372689, related compounds, or any components of the formulations

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
PlaceboPlaceboPlacebo given orally
LY3372689 Low DoseLY3372689LY3372689 given orally
LY3372689 High DoseLY3372689LY3372689 given orally
Primary Outcome Measures
NameTimeMethod
Change from Baseline to End Time Point in Integrated Alzheimer's Disease Rating Scale (iADRS)Baseline, 76 to 124 Weeks

Change from Baseline to End Time Point in iADRS will be measured in participants with early symptomatic Alzheimer's Disease (AD) with demonstrated presence of moderate levels of tau pathology

Secondary Outcome Measures
NameTimeMethod
Change From Baseline to End Time Point in Clinical Dementia Rating Scale - Sum of Boxes (CDR-SB)Baseline, 76 to 124 Weeks

Change From Baseline to End Time Point in CDR-SB

Change from Baseline to End Time Point in Alzheimer's Disease Assessment Scale - Cognitive Subscale (ADAS-Cog13)Baseline, 76 to 124 Weeks

Change from Baseline to End Time Point in ADAS-Cog13

Change from Baseline to End Time Point in Alzheimer's Disease Cooperative Study Instrumental Activities of Daily Living Inventory (ADCS-iADL)Baseline, 76 to 124 Weeks

Change from Baseline to End Time Point in ADCS-iADL

Pharmacokinetics (PK) Plasma Concentration of LY3372689Up to 124 Weeks

PK Plasma Concentration of LY3372689

Change from Baseline to End Time Point in iADRSBaseline, 76 to 124 Weeks

Change from baseline to end point time in iADRS will be measured in the full study population (moderate + high levels of tau pathology) with early symptomatic AD

Change from Baseline to End Time Point in Brain Tau Deposition as Measured by Flortaucipir F18 PET scanBaseline, 76 to 124 Weeks

Change from Baseline to End Time Point in Brain Tau Deposition as Measured by Flortaucipir F18 PET scan

Change from Baseline to End Time Point in Volumetric Magnetic Resonance Imaging (vMRI) MeasuresBaseline, 76 to 124 Weeks

Change from Baseline to End Time Point in Volumetric MRI Measures

Change from Baseline to End Time Point in Mini Mental State Examination (MMSE)Baseline, 76 to 124 Weeks

Change from Baseline to End Time Point in MMSE

Trial Locations

Locations (68)

Memory Clinic Toride

🇯🇵

Toride, Ibaraki, Japan

St Vincent's Hospital

🇦🇺

Sydney, New South Wales, Australia

Box Hill Hospital

🇦🇺

Box Hill, Victoria, Australia

Hope Clinical Research, Inc.

🇺🇸

Canoga Park, California, United States

Neuro-Pain Medical Center

🇺🇸

Fresno, California, United States

Irvine Clinical Research

🇺🇸

Irvine, California, United States

Sharp Mesa Vista Hospital

🇺🇸

San Diego, California, United States

Institute for Neurodegenerative Disorders

🇺🇸

New Haven, Connecticut, United States

JEM Research Institute

🇺🇸

Atlantis, Florida, United States

VIN-Julie Schwartzbard

🇺🇸

Aventura, Florida, United States

Neurology Offices of South Florida

🇺🇸

Boca Raton, Florida, United States

Brain Matters Research

🇺🇸

Stuart, Florida, United States

Neuropsychiatric Research Center of Southwest Florida

🇺🇸

Fort Myers, Florida, United States

K2 Medical Research

🇺🇸

Maitland, Florida, United States

ClinCloud - Viera

🇺🇸

Melbourne, Florida, United States

Merritt Island Medical Research, LLC

🇺🇸

Merritt Island, Florida, United States

VIN-Andrew Lerman

🇺🇸

Miami, Florida, United States

IMIC, Inc.

🇺🇸

Miami, Florida, United States

VIN-Victor Faradji

🇺🇸

Miami, Florida, United States

Suncoast Clinical Research, Inc.

🇺🇸

New Port Richey, Florida, United States

Renstar Medical Research

🇺🇸

Ocala, Florida, United States

VIN- Margarita Almeida El-Ramey

🇺🇸

Pembroke Pines, Florida, United States

Charter Research - Lady Lake

🇺🇸

The Villages, Florida, United States

Josephson Wallack Munshower Neurology, PC

🇺🇸

Indianapolis, Indiana, United States

Boston Center for Memory

🇺🇸

Newton, Massachusetts, United States

Donald S. Marks M.D., P.C.

🇺🇸

Plymouth, Massachusetts, United States

MedVadis Research Corporation

🇺🇸

Waltham, Massachusetts, United States

The Cognitive and Research Center of New Jersey

🇺🇸

Springfield, New Jersey, United States

Adams Clinical

🇺🇸

Watertown, Massachusetts, United States

Advanced Memory Research Institute of New Jersey

🇺🇸

Toms River, New Jersey, United States

University at Buffalo - UBMD Neurology

🇺🇸

Buffalo, New York, United States

Abington Neurological Associates, Ltd.

🇺🇸

Abington, Pennsylvania, United States

Keystone Clinical Studies

🇺🇸

Plymouth Meeting, Pennsylvania, United States

Rhode Island Mood & Memory Research Institute

🇺🇸

East Providence, Rhode Island, United States

Kerwin Medical Center

🇺🇸

Dallas, Texas, United States

The University of Texas Health Science Center at Houston

🇺🇸

Houston, Texas, United States

The Memory Clinic

🇺🇸

Bennington, Vermont, United States

Central Coast Neurosciences Research (Tumbi Umbi)

🇦🇺

Central Coast, New South Wales, Australia

HammondCare Greenwich Hospital

🇦🇺

Sydney, New South Wales, Australia

Hornsby Ku-Ring-Gai Hospital

🇦🇺

Sydney, New South Wales, Australia

KARA Institute for Neurological Diseases

🇦🇺

Sydney, New South Wales, Australia

Private Practice - Dr PL Morris

🇦🇺

Southport, Queensland, Australia

The Queen Elizabeth Hospital

🇦🇺

Woodville, South Australia, Australia

NeuroCentrix

🇦🇺

Carlton, Victoria, Australia

Delmont Private Hospital

🇦🇺

Glen Iris, Victoria, Australia

HammondCare

🇦🇺

Malvern, Victoria, Australia

Bruyère Research Institute

🇨🇦

Ottawa, Ontario, Canada

Clinique de la Mémoire de l'Outaouais

🇨🇦

Ottawa, Ontario, Canada

Ottawa Memory Clinic

🇨🇦

Ottawa, Ontario, Canada

Toronto Memory Program

🇨🇦

Toronto, Ontario, Canada

Diex Recherche Sherbrooke Inc.

🇨🇦

Sherbrooke, Quebec, Canada

National Center for Geriatrics and Gerontology

🇯🇵

Obu City, Aichi, Japan

Himeji Central Hospital Affiliated Clinic

🇯🇵

Himeji, Hyogo, Japan

Kobe City Medical Center General Hospital

🇯🇵

Kobe, Hyogo, Japan

Oita University Hospital

🇯🇵

Yufu, Oita, Japan

Katayama Medical Clinic

🇯🇵

Kurashiki, Okayama, Japan

Nozomi Memory Clinic

🇯🇵

Mitaka-shi, Tokyo, Japan

Kikukawa Clinic

🇯🇵

Nerima, Tokyo, Japan

Memory Clinic Ochanomizu

🇯🇵

Tokyo, Japan

Wroclawskie Centrum Alzheimerowskie

🇵🇱

Wroclaw, Dolnośląskie, Poland

Centrum Medyczne NEUROMED

🇵🇱

Bydgoszcz, Kujawsko-pomorskie, Poland

Centrum Medyczne NeuroProtect

🇵🇱

Warszawa, Mazowieckie, Poland

Diamond Clinic

🇵🇱

Krakow, Małopolskie, Poland

Podlaskie Centrum Psychogeriatrii

🇵🇱

Białystok, Podlaskie, Poland

Centrum Badan Klinicznych PI-House sp. z o.o.

🇵🇱

Gdansk, Pomorskie, Poland

Centrum Medyczne SENIOR

🇵🇱

Sopot, Pomorskie, Poland

Nzoz Neuro-Kard Ilkowski i Partnerzy SPL

🇵🇱

Poznan, Wielkopolskie, Poland

Centrum Medyczne Euromedis

🇵🇱

Szczecin, Zachodniopomorskie, Poland

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