MedPath

Study to Assess the Short- and Long-term Efficacy of Certolizumab Pegol Plus Methotrexate Compared to Adalimumab Plus Methotrexate in Subjects With Moderate to Severe Rheumatoid Arthritis (RA) Inadequately Responding to Methotrexate

Phase 4
Completed
Conditions
Rheumatoid Arthritis
Interventions
Biological: Certolizumab Pegol (CZP)
Biological: Adalimumab (ADA)
Registration Number
NCT01500278
Lead Sponsor
UCB Pharma SA
Brief Summary

This study is conducted to evaluate the short (12 Weeks) and long term (104 Weeks) efficacy of Certolizumab Pegol compared with Adalimumab both in combination with Methotrexate (MTX) in the treatment of moderate to severe Rheumatoid Arthritis (RA) that is not responding adequately to MTX.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
915
Inclusion Criteria
  • Subject must have a diagnosis of Rheumatoid Arthritis (RA) at Screening, as defined by the 2010 European League Against Rheumatism (EULAR)/American College of Rheumatology (ACR) classification criteria (Aletaha D et al, 2010)

  • Subject must have a positive Rheumatoid Factor (RF) and/or a positive anti-Cyclic Citrullinated Peptide antibody (anti-CCP) as determined by the central laboratory at Screening

  • Subject must have moderate to severe RA disease at Screening and Baseline defined as:

    1. Screening (all criteria required)

      • ≥ 4 swollen joints (of 28 prespecified joints)
      • Disease Activity Score [Erythrocyte Sedimentation Rate] (DAS28[ESR]) > 3.2
      • C-Reactive Protein (CRP) concentration ≥ 10 mg/L (or 1.0 mg/dL) or Erythrocyte Sedimentation Rate (ESR) (Westergren) ≥ 28 mm/hr
    2. Baseline (both criteria required)

      • ≥ 4 swollen joints (of 28 prespecified joints)
      • Disease Activity Score [Erythrocyte Sedimentation Rate] (DAS28[ESR]) > 3.2
  • Subject must have inadequately responded previously to Methotrexate (MTX)

  • Subject is using MTX 15 to 25 mg/week orally or subcutaneously at Screening and has used the same MTX regimen for a minimum of 28 days prior to Baseline

Exclusion Criteria
  • Subject has previously received any biological Disease Modifying Antirheumatic Drug (DMARD) or has received treatment with cyclophosphamide, chlorambucil, Janus Kinase, phosphodiesterase 4 inhibitors or investigational agents such as spleen tyrosine kinase
  • Diagnosis of any other inflammatory arthritis
  • Infected with Tuberculosis (TB) or high risk of acquiring TB infection
  • Subjects with concurrent acute or chronic viral hepatitis B or C infection
  • Subjects with a history of chronic or recurrent infections or subjects at high risk of infection
  • Use of prohibited medications like nonbiological DMARDs (excluding MTX), biological DMARDs excluding study medications, experimental therapy, IA hyaluronic acid

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Certolizumab Pegol + Methotrexate (CZP + MTX)Certolizumab Pegol (CZP)-
Adalimumab + Methotrexate (ADA + MTX)Adalimumab (ADA)-
Adalimumab + Methotrexate (ADA + MTX)Methotrexate (MTX)-
CZP + MTX followed by ADA + MTXMethotrexate (MTX)Those subjects who received Certolizumab Pegol (400 mg at Weeks 0, 2, 4 followed by 200 mg every two weeks) + Methotrexate (CZP+ MTX) at Baseline and are Non-Responders at Week 12, switch to Adalimumab (40 mg) + Methotrexate (ADA + MTX) after Week 12.
CZP + MTX followed by ADA + MTXCertolizumab Pegol (CZP)Those subjects who received Certolizumab Pegol (400 mg at Weeks 0, 2, 4 followed by 200 mg every two weeks) + Methotrexate (CZP+ MTX) at Baseline and are Non-Responders at Week 12, switch to Adalimumab (40 mg) + Methotrexate (ADA + MTX) after Week 12.
CZP + MTX followed by ADA + MTXAdalimumab (ADA)Those subjects who received Certolizumab Pegol (400 mg at Weeks 0, 2, 4 followed by 200 mg every two weeks) + Methotrexate (CZP+ MTX) at Baseline and are Non-Responders at Week 12, switch to Adalimumab (40 mg) + Methotrexate (ADA + MTX) after Week 12.
ADA + MTX followed by CZP + MTXCertolizumab Pegol (CZP)Those subjects who received Adalimumab (40 mg + Placebo at Weeks 0, 2, 4 followed by 40 mg ADA every two weeks) + Methotrexate (ADA+ MTX) at Baseline and are Non-Responders at Week 12, switch to Certolizumab Pegol (400 mg at Weeks 12, 14, 16 followed by 200 mg every two weeks) + Methotrexate (CZP+ MTX) after Week 12.
ADA + MTX followed by CZP + MTXAdalimumab (ADA)Those subjects who received Adalimumab (40 mg + Placebo at Weeks 0, 2, 4 followed by 40 mg ADA every two weeks) + Methotrexate (ADA+ MTX) at Baseline and are Non-Responders at Week 12, switch to Certolizumab Pegol (400 mg at Weeks 12, 14, 16 followed by 200 mg every two weeks) + Methotrexate (CZP+ MTX) after Week 12.
Certolizumab Pegol + Methotrexate (CZP + MTX)Methotrexate (MTX)-
ADA + MTX followed by CZP + MTXMethotrexate (MTX)Those subjects who received Adalimumab (40 mg + Placebo at Weeks 0, 2, 4 followed by 40 mg ADA every two weeks) + Methotrexate (ADA+ MTX) at Baseline and are Non-Responders at Week 12, switch to Certolizumab Pegol (400 mg at Weeks 12, 14, 16 followed by 200 mg every two weeks) + Methotrexate (CZP+ MTX) after Week 12.
Primary Outcome Measures
NameTimeMethod
Percentage of Subjects Who Met the American College of Rheumatology 20 % (ACR20) Criteria at Week 12Week 12

Subjects who met the ACR20 criteria were those subjects with at least 20% improvement from Baseline for Tender Joint Count (TJC), Swollen Joint Count (SJC), and at least 3 of the 5 remaining core set measures: 1) Health Assessment Questionnaire-Disability Index (HAQ-DI), 2) C-reactive Protein (CRP), 3) Patient's Assessment of Arthritis Pain-Visual Analog Scale (PAAP-VAS), 4) Patient's Global Assessment of Disease Activity-Visual Analog Scale (PtGADA-VAS), 5) Physician's Global Assessment of Disease Activity-Visual Analog Scale (PhGA-VAS).

Percentage of Subjects Who Had a Disease Activity Score 28 [Erythrocyte Sedimentation Rate] (DAS28 [ESR]) ≤ 3.2 at Week 104Week 104

DAS28 \[ESR\] was calculated using the Tender Joint Count (TJC), Swollen Joint Count (SJC), Erythrocyte Sedimentation Rate (ESR in mm/hour), and the Patient's Global Assessment of Disease Activity - Visual Analog Scale (PtGADA-VAS in mm) using the following formula: 0.56 x √ (TJC) + 0.28 x √ (SJC) + 0.70 x lognat (ESR) + 0.014 x Patient Global Assessment of Arthritis, where 28 joints were examined and a lower score indicates less disease activity.

Secondary Outcome Measures
NameTimeMethod
Percentage of Week 12 Responders Who Had a Disease Activity Score 28 [Erythrocyte Sedimentation Rate] (DAS28 [ESR]) ≤ 3.2 at Week 104Week 104

DAS28 \[ESR\] was calculated using the Tender Joint Count (TJC), Swollen Joint Count (SJC), Erythrocyte Sedimentation Rate (ESR in mm/hour), and the Patient's Global Assessment of Disease Activity - Visual Analog Scale (PtGADA-VAS in mm) using the following formula: 0.56 x √ (TJC) + 0.28 x √ (SJC) + 0.70 x lognat (ESR) + 0.014 x Patient Global Assessment of Arthritis, where 28 joints were examined and a lower score indicates less disease activity.

The definition of Week 12 responders was DAS28\[ESR\] Low Disease Activity (LDA) (ie ≤ 3.2) or an improvement of ≥ 1.2 in DAS28\[ESR\] relative to Baseline.

Percentage of Subjects Who Met the American College of Rheumatology 20 % (ACR20) Criteria at Week 6Week 6

Subjects who met the ACR20 criteria were those subjects with at least 20% improvement from Baseline for Tender Joint Count (TJC), Swollen Joint Count (SJC), and at least 3 of the 5 remaining core set measures: 1) Health Assessment Questionnaire-Disability Index (HAQ-DI), 2) C-reactive Protein (CRP), 3) Patient's Assessment of Arthritis Pain-Visual Analog Scale (PAAP-VAS), 4) Patient's Global Assessment of Disease Activity-Visual Analog Scale (PtGADA-VAS), 5) Physician's Global Assessment of Disease Activity-Visual Analog Scale (PhGA-VAS).

Percentage of Subjects Who Had a Disease Activity Score 28 [Erythrocyte Sedimentation Rate] (DAS28 [ESR]) ≤ 3.2 at Week 6Week 6

DAS28 \[ESR\] was calculated using the Tender Joint Count (TJC), Swollen Joint Count (SJC), Erythrocyte Sedimentation Rate (ESR in mm/hour), and the Patient's Global Assessment of Disease Activity - Visual Analog Scale (PtGADA-VAS in mm) using the following formula: 0.56 x √ (TJC) + 0.28 x √ (SJC) + 0.70 x lognat (ESR) + 0.014 x Patient Global Assessment of Arthritis, where 28 joints were examined and a lower score indicates less disease activity.

Percentage of Subjects Who Had a Disease Activity Score 28 [Erythrocyte Sedimentation Rate] (DAS28 [ESR]) ≤ 3.2 at Week 12Week 12

DAS28 \[ESR\] was calculated using the Tender Joint Count (TJC), Swollen Joint Count (SJC), Erythrocyte Sedimentation Rate (ESR in mm/hour), and the Patient's Global Assessment of Disease Activity - Visual Analog Scale (PtGADA-VAS in mm) using the following formula: 0.56 x √ (TJC) + 0.28 x √ (SJC) + 0.70 x lognat (ESR) + 0.014 x Patient Global Assessment of Arthritis, where 28 joints were examined and a lower score indicates less disease activity.

Percentage of Subjects With a Disease Activity Score 28 [Erythrocyte Sedimentation Rate] (DAS28 [ESR]) ≤ 3.2 at Week 104, in Subjects Responding at Both Week 6 and Week 12Week 104

DAS28 \[ESR\] was calculated using the Tender Joint Count (TJC), Swollen Joint Count (SJC), Erythrocyte Sedimentation Rate (ESR in mm/hour), and the Patient's Global Assessment of Disease Activity - Visual Analog Scale (PtGADA-VAS in mm) using the following formula: 0.56 x √ (TJC) + 0.28 x √ (SJC) + 0.70 x lognat (ESR) + 0.014 x Patient Global Assessment of Arthritis, where 28 joints were examined and a lower score indicates less disease activity.

The definition of Week 6/12 responders was DAS28\[ESR\] Low Disease Activity (LDA) (ie ≤ 3.2) or an improvement of ≥ 1.2 in DAS28\[ESR\] relative to Baseline.

Change From Baseline in the Health Assessment Questionnaire-Disability Index (HAQ-DI) at Week 104From Baseline to Week 104

HAQ-DI was derived based on the mean of individual scores in 8 categories of daily living actives (using 20 questions). Each question was scored 0-3 (0 = without any difficulty, 1 = with some difficulty, 2 = with much difficulty, and 3 = unable to do), and the total HAQ-DI was scored on the scale of 0-3 as well. Change from Baseline was computed as the value at Week 104 minus the Baseline value. A negative value in Change from Baseline indicates an improvement.

Kaplan-Meier Estimates of Proportion of Subjects Who Discontinued After Response at Week 12From Week 12 up to Week 104

Response at Week 12 means that a subject had either a Disease Activity Score 28 \[Erythrocyte Sedimentation Rate\] (DAS28 \[ESR\]) ≤ 3.2 at Week 12 or had a reduction of DAS28 \[ESR\] ≥ 1.2 from Baseline to Week 12. Kaplan-Meier Estimates of Proportion of Subjects Discontinued are presented per study week (days relative to Week 12 visit).

Trial Locations

Locations (175)

166

🇺🇸

Houston, Texas, United States

35

🇧🇬

Plovdiv, Bulgaria

14

🇵🇹

Ponte De Lima, Portugal

4

🇦🇺

Hobart, Tasmania, Australia

100

🇭🇺

Kistarcsa, Hungary

113

🇵🇱

Warszawa, Poland

76

🇵🇹

Lisboa, Portugal

96

🇷🇴

Galati, Romania

8

🇦🇺

Fitzroy, Victoria, Australia

85

🇦🇹

Stockerau, Austria

107

🇵🇱

Bydgoszcz, Poland

69

🇵🇹

Coimbra, Portugal

57

🇷🇴

Bucharest, Romania

1

🇦🇺

Malvern, Victoria, Australia

18

🇧🇬

Pleven, Bulgaria

108

🇵🇱

Wroclaw, Poland

159

🇺🇸

Tucson, Arizona, United States

144

🇺🇸

Menifee, California, United States

161

🇺🇸

Fullerton, California, United States

147

🇺🇸

Covina, California, United States

142

🇺🇸

Aventura, Florida, United States

148

🇺🇸

Whittier, California, United States

202

🇺🇸

Maywood, Illinois, United States

145

🇺🇸

Coeur d'Alene, Idaho, United States

178

🇺🇸

Baltimore, Maryland, United States

137

🇺🇸

Battle Creek, Michigan, United States

190

🇺🇸

Wyomissing, Pennsylvania, United States

155

🇺🇸

Lansing, Michigan, United States

170

🇺🇸

Reno, Nevada, United States

219

🇺🇸

Orchard Park, New York, United States

201

🇺🇸

Teaneck, New Jersey, United States

154

🇺🇸

Albany, New York, United States

132

🇺🇸

Duncansville, Pennsylvania, United States

146

🇺🇸

Dallas, Texas, United States

133

🇺🇸

Jackson, Tennessee, United States

151

🇺🇸

Corpus Christi, Texas, United States

67

🇮🇹

Prato, Italy

213

🇺🇸

Dallas, Texas, United States

212

🇺🇸

Houston, Texas, United States

6

🇦🇺

Camperdown, New South Wales, Australia

2

🇦🇺

Maroochydore, Queensland, Australia

163

🇺🇸

Clarksburg, West Virginia, United States

3

🇦🇺

Subiaco, Western Australia, Australia

22

🇦🇹

Wien, Austria

21

🇧🇬

Sofia, Bulgaria

29

🇧🇬

Sofia, Bulgaria

34

🇧🇬

Sofia, Bulgaria

70

🇫🇷

Le Mans, France

221

🇨🇦

Barrie, Canada

171

🇨🇦

Quebec, Canada

103

🇨🇿

Brno, Czechia

49

🇨🇿

Praha, Czechia

61

🇨🇿

Hradec Kralove, Czechia

31

🇩🇪

Heidelberg, Germany

64

🇩🇪

Köln, Germany

37

🇩🇪

Herne, Germany

72

🇫🇷

Montpellier Cedex 5, France

17

🇩🇪

Hamburg, Germany

63

🇩🇪

Osnabrück, Germany

68

🇭🇺

Gyula, Hungary

33

🇭🇺

Veszprem, Hungary

194

🇲🇽

Chihuahua, Mexico

106

🇵🇱

Poznan, Poland

11

🇩🇪

Ratingen, Germany

20

🇮🇪

Limerick, Ireland

88

🇮🇹

Genova, Italy

13

🇭🇺

Budapest, Hungary

51

🇮🇪

Dublin, Ireland

195

🇲🇽

Chihuahua, Mexico

79

🇮🇹

Magenta, Italy

98

🇮🇹

Napoli, Italy

80

🇮🇹

Bergamo, Italy

38

🇮🇹

Genova, Italy

36

🇮🇹

Roma, Italy

39

🇮🇹

Verona, Italy

193

🇲🇽

Guadalajara, Mexico

192

🇲🇽

Monterrey, Mexico

191

🇲🇽

San Luis Potosi, Mexico

60

🇲🇨

Monaco, Monaco

27

🇵🇹

Lisbon, Portugal

24

🇷🇴

Bucharest, Romania

74

🇷🇴

Braila, Romania

25

🇷🇴

Bucharest, Romania

52

🇪🇸

A Coruna, Spain

73

🇬🇧

Upton, United Kingdom

99

🇬🇧

Wigan, United Kingdom

30

🇪🇸

Madrid, Spain

86

🇬🇧

Ashford, United Kingdom

59

🇬🇧

Leeds, United Kingdom

77

🇬🇧

Poole, United Kingdom

89

🇫🇷

Brest, France

62

🇫🇷

Lyon, France

172

🇨🇦

Hamilton, Ontario, Canada

174

🇨🇦

Hamilton, Ontario, Canada

177

🇨🇦

Ottawa, Ontario, Canada

40

🇨🇿

Uherske Hradiste, Czechia

141

🇺🇸

Birmingham, Alabama, United States

140

🇺🇸

Cincinnati, Ohio, United States

184

🇺🇸

Oklahoma City, Oklahoma, United States

139

🇺🇸

San Antonio, Texas, United States

207

🇺🇸

Plainview, New York, United States

181

🇺🇸

Sugar Land, Texas, United States

217

🇺🇸

La Mesa, California, United States

179

🇨🇦

Edmonton, Alberta, Canada

214

🇺🇸

Tuscaloosa, Alabama, United States

152

🇺🇸

Hot Springs, Arkansas, United States

149

🇺🇸

Los Angeles, California, United States

189

🇺🇸

Van Nuys, California, United States

220

🇺🇸

Lewes, Delaware, United States

216

🇺🇸

Fort Lauderdale, Florida, United States

153

🇺🇸

Detroit, Michigan, United States

209

🇺🇸

Vero Beach, Florida, United States

204

🇺🇸

Eagan, Minnesota, United States

143

🇺🇸

Saint Louis Park, Minnesota, United States

180

🇺🇸

Rochester, Minnesota, United States

135

🇺🇸

Omaha, Nebraska, United States

150

🇺🇸

Voorhees, New Jersey, United States

167

🇺🇸

Syracuse, New York, United States

136

🇺🇸

Brooklyn, New York, United States

187

🇺🇸

Myrtle Beach, South Carolina, United States

164

🇺🇸

Bethlehem, Pennsylvania, United States

160

🇺🇸

Knoxville, Tennessee, United States

131

🇺🇸

Dallas, Texas, United States

203

🇺🇸

Orangeburg, South Carolina, United States

211

🇺🇸

Arlington, Virginia, United States

215

🇺🇸

Glendale, Wisconsin, United States

218

🇨🇦

Rimouski, Quebec, Canada

46

🇧🇬

Sofia, Bulgaria

183

🇨🇦

Halifax, Nova Scotia, Canada

206

🇨🇦

Ottawa, Ontario, Canada

175

🇨🇦

St. Catharines, Ontario, Canada

169

🇨🇦

Sainte Foy, Quebec, Canada

58

🇨🇿

Plzen, Czechia

90

🇫🇷

Orleans, France

43

🇭🇺

Szeged, Hungary

95

🇬🇷

Larisa, Greece

56

🇩🇪

Berlin, Germany

105

🇫🇷

Toulouse Cedex 9, France

47

🇩🇪

Fulda, Germany

71

🇩🇪

Traunstein, Germany

66

🇩🇪

Rheine, Germany

94

🇬🇷

Heraklion, Greece

44

🇩🇪

Zerbst, Germany

48

🇩🇪

Rostock, Germany

42

🇭🇺

Budapest, Hungary

23

🇮🇪

Dublin, Ireland

115

🇵🇱

Warszawa, Poland

81

🇵🇹

Porto, Portugal

54

🇷🇴

Bacau, Romania

12

🇷🇴

Cluj-Napoca, Romania

28

🇷🇴

Bucharest, Romania

32

🇷🇴

Bucharest, Romania

26

🇷🇴

Iasi, Romania

65

🇪🇸

Vigo, Spain

16

🇪🇸

A Coruna, Spain

83

🇪🇸

Madrid, Spain

82

🇪🇸

Sabadell, Spain

53

🇨🇭

St. Gallen, Switzerland

50

🇨🇭

Zürich, Switzerland

78

🇬🇧

Brighton, United Kingdom

55

🇬🇧

Sheffield, United Kingdom

19

🇬🇧

London, United Kingdom

208

🇺🇸

Sacramento, California, United States

185

🇺🇸

Roseville, California, United States

157

🇺🇸

Spokane, Washington, United States

5

🇦🇺

Kogarah, New South Wales, Australia

162

🇺🇸

Gainesville, Florida, United States

134

🇺🇸

Lexington, Kentucky, United States

205

🇺🇸

Albuquerque, New Mexico, United States

210

🇺🇸

Charleston, South Carolina, United States

138

🇺🇸

Austin, Texas, United States

7

🇦🇺

Clayton, Victoria, Australia

176

🇨🇦

St. John's, Newfoundland and Labrador, Canada

165

🇺🇸

Victoria, Texas, United States

168

🇨🇦

St. John's, Newfoundland and Labrador, Canada

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