MedPath

PGL4001 Versus GnRH-agonist in Uterine Myomas

Phase 3
Completed
Conditions
Uterine Myomas
Interventions
Registration Number
NCT00740831
Lead Sponsor
PregLem SA
Brief Summary

This trial will assess the efficacy and safety of PGL4001 versus GnRH agonist, over a 3-month period for the pre-operative treatment of pre-menopausal women suffering from excessive uterine bleeding due to uterine myoma.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
Female
Target Recruitment
301
Inclusion Criteria
  • Be a pre-menopausal woman between 18 and 50 years inclusive.
  • Have excessive uterine bleeding due to myoma
  • Have a myomatous uterus with at least one myoma of ≥ 3 cm diameter in size
  • Be eligible for one surgical procedure: e.g. hysterectomy, myomectomy or others.
  • If of childbearing potential the subject must be practicing a non-hormonal method of contraception.
  • Have a Body Mass Index (BMI) ≥ 18 and ≤ 40.
Exclusion Criteria
  • Has a history of or current uterine, cervical, ovarian or breast cancer.
  • Has a history of or current endometrium atypical hyperplasia or adenocarcinoma.
  • Has a known severe coagulation disorder.
  • Has a history of or current treatment for myoma with a Selective Progesterone Receptor Modulator (SPRM) or a GnRH-agonist.
  • Has a history of or known current osteoporosis.
  • Has abnormal hepatic function at study entry.
  • Has a positive pregnancy test at baseline or is nursing or planning a pregnancy during the course of the study.
  • Has a current (within twelve months) problem with alcohol or drug abuse.
  • Is currently enrolled in an investigational drug or device study or has participated in such a study within the last 30 days.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
A (PGL4001 5 mg)PGL4001Drug: PGL4001 5mg (oral tablets) and leuproreline matching placebo (intramuscular injection)
B (PGL4001 10mg)PGL4001Drug: PGL4001 10 mg (oral tablets) and leuproreline matching placebo (intramuscular injection)
C (GnRH-agonist)leuprorelinPGL4001 matching placebo (oral tablets) and leuprorelin 3.75 mg (intramuscular injection)
Primary Outcome Measures
NameTimeMethod
Percentage of Subjects With Reduction of Uterine Bleeding at Week 13 Visit Defined as Pictorial Blood-loss Assessment Chart (PBAC) Score < 75 at End-of-treatment Visit (Week 13 Visit)3 months

Uterine bleeding was assessed with the use of the PBAC, a validated self-reporting method to estimate menstrual blood loss.

Patients recorded daily the number of tampons and towels used and the degree to which individual items were soiled with blood (plus small or large clots). Monthly scores range from 0 (amenorrhea) to more than 500, with higher numbers indicating more bleeding.

A slightly stained tampon/towel scores 1, a partially stained tampon/towel scores 5, a completely saturated tampon scores 10 and a completely saturated towel scores 20. Small clots/flooding (2cm) score 1. Large clots/flooding (3cm) score 5.

Menorrhagia is defined as a PBAC \> 100 during one menstrual period which approximates to a blood loss of \> 80 mL. A PBAC of 400 corresponds to a blood loss of around 300 mL or approximately 80 tampons/towels used.

The week 13 PBAC score was calculated using the last 28 days of treatment.

Co-primary Safety Endpoint: Serum Estradiol Levels at End of Treatment Visit (Week 13 Visit) for PGL4001 Compared With GnRHagonistWeek 13 visit

Measured by log 10 (log pg/ml) transformed values for estradiol (E2) in blood samples

Co-primary Safety Endpoint: % of Subjects Reporting Moderate or Severe Hot Flushes as Adverse Events Throughout the Treatment Period for PGL4001 Compared With GnRH-agonistUp to week 17

Difference in percentage of subjects reporting moderate or severe hot flushes:

Frequency and severity of this adverse event(as spontaneously reported by patients or elicited by nonleading questions) were recorded on standard forms at every visit up to week 17.

Secondary Outcome Measures
NameTimeMethod
Change in the Total Volume of the Three Largest Myomas From Baseline to Week 133 months

Assessment of PGL4001 capacity to decrease volume of the three largest myomas was performed at each center by means of ultrasonography at baseline and at week 13.

The total volume of the three largest myomas assessed at screening and at end-of-treatment visit (Week 13) was analysed on a logarithm transformed scale (to base 10).

Trial Locations

Locations (44)

Hospital Universitario Vall d'Hebrón

🇪🇸

Barcelona, Spain

Clinica Obstetrica - Azienda Ospedaliera Universitaria di Cagliari

🇮🇹

Cagliari, Italy

Policlinico Universitario Federico II

🇮🇹

Napoli, Italy

Hospital Universitaris La Fe

🇪🇸

Valencia, Spain

Hospital Virgen de la Arrixaca Servicio de Ginecología Carretera Madrid-Cartagena

🇪🇸

Murcia, Spain

Hospital Universitario Dr. Peset

🇪🇸

Valencia, Spain

Azienda Ospedaliera S. Gerardo - U. O. Ostetricia e Ginecologia

🇮🇹

Monza, Italy

Prywatna Klinika Polozniczo-Ginekologiczna

🇵🇱

Bialystok, Poland

INVICTA Sp. Z o.o.

🇵🇱

Gdańsk, Poland

Policlinico Universitario "Agostino Gemelli"

🇮🇹

Roma, Italy

Institut Universitari Dexeus

🇪🇸

Barcelona, Spain

Clinica Ostetrica e Ginecologica - A. O. U. Policlinico Paolo Giaccone

🇮🇹

Palermo, Italy

Cabinet de Gynécologie Chirurgicale

🇫🇷

Bordeaux, France

Universita di Padova-Dip scienze ginecologiche e della riproduzione umana

🇮🇹

Padova, Italy

Hospital Clínic i Provincial

🇪🇸

Barcelona, Spain

Clínica Ginecológica CEOGA

🇪🇸

Lugo, Spain

Samodzielny Publiczny Szpital Klinika Ginekologii Onkologicznej i Ginekologii

🇵🇱

Lublin, Poland

Gabinet Lekarski Specjalistyczny "Sonus"

🇵🇱

Warszawa, Poland

Medical University Graz

🇦🇹

Graz, Austria

CHU de Clermont-Ferrand - Polyclinique Gynécologie-Obstétrique

🇫🇷

Clermont Ferrand, France

Private Practice

🇪🇸

Madrid, Spain

Medizinische Hochschule Hannover, Frauenklinik, Abt. I für Frauenheilkunde und Geburtshilfe,

🇩🇪

Hannover, Germany

Universitätsklinikum Köln Klinik und poliklinik für Frauenheilkunde und Geburtshilfe

🇩🇪

Köln, Germany

Universitätsklinikum Tübingen

🇩🇪

Tübingen, Germany

Universität zu Lübeck, Klinik für Gynäkologie und Geburtshilfe

🇩🇪

Lübeck, Germany

Hadassah University Hospital

🇮🇱

Jerusalem, Israel

Meir Medical Center

🇮🇱

Kfar-Saba, Israel

Poliklinik fur Frauenheilkunde und Geburtshilfe

🇩🇪

Münster, Germany

Soroka University Medical Center, Division of Obstetrics & Gynecology

🇮🇱

Be'er Sheva, Israel

Western Galilee Hospital Nahariya

🇮🇱

Nahariya, Israel

Rabin Medical Center, Helen Schneider Hospital for Women

🇮🇱

Petach Tikva, Israel

Ammerland-Klinik GmbH Frauenklinik

🇩🇪

Westerstede, Germany

Clinica Ostetrica e Ginecologica II - Università degli Studi di Bari

🇮🇹

Bari, Italy

Hadassah University Hospital, Mount Scopus

🇮🇱

Jerusalem, Israel

Hospital Universitario Doce de Octubre

🇪🇸

Madrid, Spain

Klinik für Gynäkologie und Geburtshilfe

🇩🇪

Chemnitz, Germany

Medical University of Innsbruck

🇦🇹

Innsbruck, Austria

CHR de la Citadelle

🇧🇪

Liège, Belgium

Medical University Vienna

🇦🇹

Vienna, Austria

Landesklinikum Thermenregion Neunkirchen; Dept. For Gynecology

🇦🇹

Neunkirchen, Austria

Clinique Universitaire St-Luc

🇧🇪

Brussels, Belgium

University Medical Center Utrecht, Gynecologist Reproductive Medicine and Surgery, Division for Reproductive Medicine

🇳🇱

Utrecht, Netherlands

Hopital Erasme, Department of Obstetrics and Gynecology,

🇧🇪

Brussels, Belgium

Clinique Universitaire de Mont-Godinne

🇧🇪

Yvoir, Belgium

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