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A Study to Evaluate CC-486/Onureg in Participants With Moderate or Severe Hepatic Impairment Compared With Normal Hepatic Function in Participants With Myeloid Malignancies

Phase 1
Recruiting
Conditions
Neoplasms
Hepatic Insufficiency
Interventions
Registration Number
NCT05209295
Lead Sponsor
Bristol-Myers Squibb
Brief Summary

The purpose of this study is to evaluate the effect of moderate or severe liver impairment on the drug levels of oral azacitidine and the safety and tolerability of oral azacitidine in participants with myeloid malignancies.

Detailed Description

Not available

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
32
Inclusion Criteria
  • Documented diagnosis of Myelodysplastic syndrome, Acute myeloid leukemia, Non-acute promyelocytic leukemia, Chronic myelomonocytic leukemia, Philadelphia-negative myeloproliferative neoplasms, Myelodysplastic syndrome Myeloproliferative neoplasms overlap, Accelerated phase and blast phase Myeloproliferative neoplasms, Blastic plasmacytoid dendritic cell neoplasm according to the World Health Organization (WHO) 2016 classification
  • Life expectancy of ≥ 3 months
  • Stable renal function without dialysis for at least 2 months prior to investigational product administration
  • Has moderate or severe hepatic impairment as defined by National Cancer Institute Organ Dysfunction Working Group criteria
Exclusion Criteria
  • Chemotherapy or radiotherapy within 2 weeks or 5 half-lives, whichever is longer, prior to the first day of investigational product administration
  • Persistent, clinically significant non-hematologic toxicities from prior therapies which have not recovered to < Grade 2
  • Any condition including the presence of laboratory abnormalities, which places the participant at unacceptable risk if he/she were to participate in the study
  • History of inflammatory bowel disease, celiac disease, prior gastrectomy, gastric bypass, upper bowel removal, or any other gastrointestinal disorder or defect that would interfere with the absorption of the investigational product and/or predispose the participant to an increased risk of gastrointestinal toxicity

Other protocol-defined inclusion/exclusion criteria apply

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Group 3OnuregControl - participants with normal hepatic function
Group 2Onureg-
Group 1Onureg-
Primary Outcome Measures
NameTimeMethod
AUC0-∞: Estimation of AUC calculated from time zero to infinityDay 1
AUC0-t: Estimation of area under the plasma concentration-time curve (AUC) calculated from time zero to the last measured time pointDay 1
Cmax: Observed maximum concentrationDay 1
Secondary Outcome Measures
NameTimeMethod
Incidence of clinically significant changes in clinical laboratory results: Clinical Chemistry testsUp to 9 Months
Incidence of clinically significant changes in clinical laboratory results: Liver Function testsUp to 9 Months
Number of participants with a recording of concomitant medicationsUp to 9 Months
Incidence of adverse eventsUp to 9 Months
Incidence of serious adverse eventsUp to 9 Months
Number of participants with clinically significant changes in electrocardiogram parametersUp to 9 Months
Incidence of clinically significant changes in vital signs: Body temperatureUp to 9 Months
Incidence of clinically significant changes in vital signs: Blood pressureUp to 9 Months
Incidence of clinically significant changes in vital signs: Heart rateUp to 9 Months
Incidence of clinically significant changes in clinical laboratory results: Hematology testsUp to 9 Months
Number of participants with a recording of concomitant proceduresUp to 9 Months
Incidence of clinically significant changes in vital signs: Respiratory rateUp to 9 Months
Incidence of clinically significant changes in clinical laboratory results: Urinalysis testsUp to 9 Months
Number of Participants with clinically significant changes in Eastern Cooperative Oncology Group (ECOG) performance statusUp to 9 Months
Number of clinically significant changes in physical examinationsUp to 9 Months

Trial Locations

Locations (22)

Hospital Universitario Austral

🇦🇷

Pilar, Buenos Aires, Argentina

Instituto Nacional De Cancerologia

🇨🇴

Bogota, Cundinamarca, Colombia

University of Iowa

🇺🇸

Iowa City, Iowa, United States

Tulane Cancer Center

🇺🇸

New Orleans, Louisiana, United States

Local Institution - 0068

🇺🇸

Worcester, Massachusetts, United States

Henry Ford Hospital

🇺🇸

Detroit, Michigan, United States

Local Institution - 0007

🇺🇸

Port Jefferson Station, New York, United States

Local Institution

🇺🇸

Cleveland, Ohio, United States

University of Virginia Cancer Center

🇺🇸

Charlottesville, Virginia, United States

Hospital Italiano de Buenos Aires

🇦🇷

ABB, Ciudad Autónoma De Buenos Aires, Argentina

Hospital Aleman

🇦🇷

Buenos Aires, Ciudad Autónoma De Buenos Aires, Argentina

Clínica Zabala

🇦🇷

Buenos Aires, Argentina

Fundacion Ctic Centro de Tratamiento E Investigacion Sobre Cancer Luis Carlos Sarmiento Angulo

🇨🇴

Bogotá, Distrito Capital De Bogotá, Colombia

Fundación Cardiovascular de Colombia

🇨🇴

Piedecuesta, Santander, Colombia

Klinikum Augsburg

🇩🇪

Augsburg, Bayern, Germany

Local Institution - 0075

🇩🇪

Halle, Sachsen-Anhalt, Germany

Local Institution - 0074

🇩🇪

Hamburg, Germany

Local Institution - 9000

🇬🇷

Thessaloniki, Greece

Local Institution - 0018

🇪🇸

Badalona, Barcelona [Barcelona], Spain

Hospital Universitari Vall d'Hebron

🇪🇸

Barcelona, Barcelona [Barcelona], Spain

Clinica Universidad de Navarra

🇪🇸

Pamplona, Navarra, Spain

Local Institution - 0078

🇪🇸

Salamanca, Spain

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