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Clinical trial/study for lung cancer patients with ROS1 positive

Phase 3
Conditions
Health Condition 1: C349- Malignant neoplasm of unspecifiedpart of bronchus or lung
Registration Number
CTRI/2022/04/041861
Lead Sponsor
F HoffmannLa Roche Ltd
Brief Summary

Not available

Detailed Description

Not available

Recruitment & Eligibility

Status
Closed to Recruitment of Participants
Sex
Not specified
Target Recruitment
0
Inclusion Criteria

1. Histologically or cytologically confirmed diagnosis of advanced or recurrent (Stage IIIB/C,

not amenable for radical treatment) or metastatic (Stage IV) NSCLC that harbors a documented ROS1 gene rearrangement

2. No prior treatment with a ROS1 tyrosine kinase inhibitor, chemotherapy, or other systemic therapy for advanced or recurrent (Stage IIIB/C not amenable for radical treatment) or metastatic (Stage IV) NSCLC

3. Prior radiotherapy is allowed if more than 14 days have elapsed between the end of treatment and randomization. Patients who received brain irradiation must have completed whole brain radiotherapy at least 14 days prior and/or stereotactic radiosurgery at least 7 days prior to the start of entrectinib treatment.

4. Measurable systemic disease according to RECIST v1.1

5. Life expectancy of at least 12 weeks

6. ECOG Performance Status of 0, 1, or 2

7. Adequate hematologic, renal, liver functions

8. Participants must have recovered from effects of any major surgery or significant traumatic injury at least 28 days before the first dose of study treatment

9. Ability to swallow entrectinib and crizotinib intact without chewing, crushing, or opening the

capsules

10. Ability to comply with the study protocol, in the investigator’s judgment

11. For women of childbearing potential: agreement to remain abstinent (refrain from heterosexual intercourse) or use contraceptive methods with a failure rate of <1% per year during the treatment period and for up to 5 weeks after the last dose of entrectinib or for at least 90 days after the last dose of crizotinib

12. For men: agreement to remain abstinent (refrain from heterosexual intercourse) or use contraceptive measures, and agreement to refrain from donating sperm.

Exclusion Criteria

1. Current participation in another therapeutic clinical trial

2. Prior treatment with a ROS1 tyrosine kinase inhibitor, chemotherapy or other systemic therapy for advanced or recurrent (Stage IIIB/C not amenable for radical treatment) or metastatic (Stage IV) NSCLC

3. NCI-CTCAE v5.0 Grade 3 or higher toxicities due to any prior therapy (excluding alopecia, fatigue, nausea and lack of appetite), which have not shown improvement and are strictly considered to interfere with current study drug

4. History of recent (within the past 3 months) symptomatic congestive heart failure or ejection

fraction ? 50% observed during screening for the study

5. History of prolonged corrected QT interval

6. History of additional risk factors for torsades de pointes

7. Grade = 2 peripheral sensory neuropathy

8. Known interstitial lung disease, interstitial fibrosis, or history of tyrosine kinase inhibitor-induced pneumonitis

9. Previous malignancy within the past 3 years

10. Incomplete recovery from any surgery prior to the start of study treatment that would

interfere with the determination of safety or efficacy

11. Active GI disease (e.g., Crohn’s disease, ulcerative colitis, or short gut syndrome) or other malabsorption syndrome that would reasonably impact drug absorption

12. History of prior therapy-induced pneumonitis

13. Any condition (in the past 3 months) e.g., myocardial infarction, unstable angina, coronary/peripheral artery bypass graft, cerebrovascular accident or transient ischemic attack, stroke, symptomatic bradycardia, or uncontrolled arrhythmias requiring medication

14. Known active infections that would interfere with the assessment of safety or efficacy of

study treatments (bacterial, fungal or viral), with the exceptions of HIV, hepatitis B virus

(HBV), and hepatitis C virus (HCV) infections

15. History of hypersensitivity to any of the additives in the entrectinib and/or crizotinib drug formulations

16. Pregnant or breastfeeding, or intending to become pregnant during the study or within 3 months after the final dose of entrectinib or crizotinib

17. Any clinically significant concomitant disease or condition that could interfere with, or for

which the treatment might interfere with, the conduct of the study or the absorption of oral

medications or that would, in the opinion of the Principal Investigator, pose an unacceptable

risk to the patient in this study

18. Any psychological, familial, sociological or geographical condition potentially hampering

compliance with the study protocol requirements and/or follow-up procedures; those conditions should be discussed with the patient before trial entry

Study & Design

Study Type
Interventional
Study Design
Not specified
Primary Outcome Measures
NameTimeMethod
PFS (Progression-free survival) defined by RECIST v1.1 <br/ ><br>Timepoint: Screening <br/ ><br>Visit 1 <br/ ><br>Visit 2 <br/ ><br>All subsequent visit after 8 weeks <br/ ><br>
Secondary Outcome Measures
NameTimeMethod
CNS-PFS defined by RECIST v1.1Timepoint: Screening <br/ ><br>Visit 1 <br/ ><br>Visit 2 <br/ ><br>All subsequent visit after 8 weeks <br/ ><br>
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