MedPath

Phase I/II CT 2106 and 5-FU/FA in Colorectal Cancer

Phase 1
Completed
Conditions
Colorectal Cancer
Registration Number
NCT00291785
Lead Sponsor
CTI BioPharma
Brief Summary

CT-2106, a camptothecin (CPT) conjugate, is a new generation of topoisomerase I inhibitors designed to deliver higher, more effective chemotherapy to tumor tissue with less toxicity to normal tissues. The objective of this study is to determine the dose limiting toxicities, safety profile and antitumor activity of CT-2016 in combination with 5-FU and folic acid for the treatment of colorectal cancer.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
48
Inclusion Criteria
  • Histologically proven metastatic colorectal adenocarcinoma, failing one prior treatment containing oxaliplatin plus 5-FU/FA
  • At least one measurable lesion according to RECIST criteria for both Phase I and II
  • ECOG performance status 0 or 1
  • Adequate hematologic, renal and hepatic function
  • Wash out period of at least 4 weeks from surgery, 4 weeks from radiotherapy
Exclusion Criteria
  • Past or concurrent history of neoplasm other than colorectal adenocarcinoma, except curatively treated non melanoma skin cancer or in situ carcinoma of the cervix.
  • Pregnant or lactating patients
  • Prior treatment with camptothecins
  • Presence or history of CNS metastasis or carcinomatous leptomeningitis
  • Current active infection per investigator assessment
  • Unresolved bowel obstruction or partial obstruction, uncontrolled Crohn's disease or ulcerative colitis
  • Current history of chronic diarrhea greater than or equal to grade 1 (CTCAE version 3)

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Primary Outcome Measures
NameTimeMethod
Phase I: determine the Maximum Tolerated Dose, dose limiting toxicities, safety profile and antitumor activityEach cycle
Secondary Outcome Measures
NameTimeMethod

Trial Locations

Locations (2)

Policlinico Universitario "A.Gemelli"

🇮🇹

Rome, Italy

Istituto Clinico Humanitas

🇮🇹

Rozzano, Italy

© Copyright 2025. All Rights Reserved by MedPath