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Tofacitinib in the Treatment of Rheumatoid Arthritis-related Interstitial Lung Disease.

Phase 2
Recruiting
Conditions
Interstitial Lung Disease
Rheumatoid Arthritis
Interventions
Registration Number
NCT05246293
Lead Sponsor
National Institute of Respiratory Diseases, Mexico
Brief Summary

Nowadays, no single drug is approved to treat rheumatoid arthritis-related interstitial lung disease (RA-ILD). The medical management of this clinical condition is empirical and controversial. There is preliminary data that tofacitinib may have a beneficial effect in treating RA-ILD. Tofacitinib may have a double role in treating RA-ILD: treat RA disease activity and an anti-fibrotic possible impact. Moreover, tofacitinib may be used as monotherapy for the treatment of rheumatoid arthritis (RA) This is a phase IIa clinical trial to evaluate the safety and tolerability of tofacitinib in RA-ILD patients.

Detailed Description

This is a phase 2 open-label study designed to evaluate the safety and tolerability of tofacitinib in RA-ILD patients. Patients who met the inclusion criteria of the study protocol will receive tofacitinib 5 mg BID for 12 months.

Objectives

Primary objectives:

1. To evaluate the safety and tolerability of tofacitinib 5 mg PO BID as monotherapy for managing RA-ILD in RA-ILD patients.

2. To evaluate the pulmonary function of patients treated with tofacitinib PO BID as monotherapy to manage RA-ILD in RA-ILD patients, at baseline, at three months of follow-up, at six months of follow-up, and one year of follow-up.

3. To estimate the efficacy of tofacitinib 5 mg PO BID as monotherapy for the management of RA-ILD, in RA-ILD patients, at three months of follow-up, at six months of follow-up, and at one year of follow-up, according to the ACR 20, 50, 70 response criteria, and the following disease activity scores index: DAS 28, CDAI and SDAI.

All the included patients will receive Tofacitinib in doses of 5 mg BID until the end of the protocol.

Recruitment & Eligibility

Status
RECRUITING
Sex
All
Target Recruitment
60
Inclusion Criteria
  1. Patients must fulfill ACR/EULAR 2010 RA classification criteria.
  2. Patients must have an interstitial lung disease confirmed by a high-resolution computed tomography scan or a surgical lung biopsy. Nonspecific interstitial pneumonia, usual interstitial pneumonia, lymphocytic pneumonia, and organized pneumonia, either by HRCT or surgical biopsy, will be included.
  3. Patients must be 18 years of age or older.
  4. There is no evidence of active, latent, or inadequately treated infection with Mycobacterium tuberculosis (TB).
  5. Patients must discontinue using the non-permitted medications: leflunomide, azathioprine, cyclosporine, tacrolimus, cyclophosphamide, and any biologic disease-modifying drug (bDMDARDs) such as anti-TNF therapy, rituximab, tocilizumab, etc. Patients must have a stable prednisone dose of ≤ 10 mg/ PO/day for at least three months.
  6. All patients must have stable doses of prednisone during the last three months of follow-up, and the prednisone dose must be ≤ 10 mg/day. Patients without a prednisone history in the previous three months may also be included in the protocol.
Exclusion Criteria
  1. Seropositivity for the following infections: HIV, HBV, and HCV.
  2. Absolute neutrophil count ≤ 1,200/L
  3. Absolute platelet count ≤ 100,000 /L
  4. Severe renal damage with GFR < 30 ml/min based on CKD-EPI formula.
  5. AST or ALT greater than 1.5 times the upper limit of normal AST and ALT levels
  6. Severe hepatic, hematologic, gastrointestinal, cardiac, and neurological disease may put the patient´s life at risk regardless of ILD severity.
  7. Severe active infections at baseline evaluation, such as pneumonia, urinary tract infections, meningitis.

8 History of drug abuse or alcoholism. 9. History of any malignancy 10. Patients with an FVC < 40% of what is expected will be excluded from the study.

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
Tofacitinib ArmTofacitinibTofacitinib in doses of 5 mg BID, in RA-ILD patients at stable doses of prednisone ≤ 10 mg/day during the last three months.
Primary Outcome Measures
NameTimeMethod
Incidence and severity of adverse events52 weeks

Adverse event: Any untoward medical occurrence in a subject being included in the trial, in which the event may not necessarily have a causal relationship with the treatment. Examples of adverse events are as follows: abnormal test findings, clinically significant symptoms and signs, hypersensitivity reactions, and progression or worsening of RA or RA-ILD.

Secondary Outcome Measures
NameTimeMethod
6 minutes walk test52 weeks

walked metters in 6 minutes

Rheumatoid arthritis disease activity according to the simplified disease activity (SDAI) index.52 weeks

The SDAI index consists of the algebraic sum of the following items: tender joint count, swollen joint count, c-reactive protein, rheumatoid arthritis activity according to the patient, disease activity according to the attending physician.

Rheumatoid arthritis disease activity according to the Disease Activity Score Index (DAS28)52 weeks

The DAS28 score is calculated with the tender joint count, swollen joint count, eritrosedimentation rate, patients' global health assesment aacording with the following formula DAS28 = ( 0.56 \* sqr(TJC)) + (0.28 \* sqr(SJC)) + ( 0.7 \* ln(VSG)) + (0.014 \* GH)

Forced Vital Capacity (liters)52 weeks

Forced vital capacity (FVC) on spirometry, the data will be presented as percentages of predicted values, according to sex, age, height, and weight.

Carbon monoxide diffusing capacity (DLCO) (mil/min/mmHg)52 weeks

The data will be presented as percentages of predicted values, according to sex, age, height, and weight.

Trial Locations

Locations (1)

Instituto Nacional de Enfermedades Respiratorias, Ismael Cosío Villegas

🇲🇽

Mexico City, Tlalpan, Mexico

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