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The Safety and Efficacy of Multiple-dose of WJ01024 in Subject With Advanced Cancer

Phase 1
Terminated
Conditions
Advanced Hematologic Malignancies
Advanced Solid Tumors
Interventions
Registration Number
NCT04991129
Lead Sponsor
Suzhou Junjing BioSciences Co., Ltd.
Brief Summary

A clinical study of WJ01024 in subjects with advanced cancer in China, to evaluate the safety, tolerability, PK and efficacy of WJ01024. This study includes a dose escalation part and a dose expansion part. Patients receive WJ01024 on Day 1 and Day 3 of each week, 4 weeks as a cycle, until disease progression, or intolerable toxicity , withdrawal of consent, or end of the study, whichever occurs first.

Detailed Description

Not available

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
23
Inclusion Criteria

Not provided

Exclusion Criteria

Not provided

Study & Design

Study Type
INTERVENTIONAL
Study Design
SEQUENTIAL
Arm && Interventions
GroupInterventionDescription
WJ01024 80mg QW repeat dose every 28 daysWJ01024-
WJ01024 5mg QD repeat dose every 28 daysWJ01024-
WJ01024 5mg BID repeat dose every 28 daysWJ01024-
WJ01024 10mg BID repeat dose every 28 daysWJ01024-
WJ01024 40mg BIW repeat dose every 28 daysWJ01024-
WJ01024 60mg BIW repeat dose every 28 daysWJ01024-
WJ01024 50mg QW repeat dose every 28 daysWJ01024-
WJ01024 40mg QW repeat dose every 28 daysWJ01024-
WJ01024 80mg BIW repeat dose every 28 daysWJ01024-
WJ01024 60mg QW repeat dose every 28 daysWJ01024-
Primary Outcome Measures
NameTimeMethod
The incidence of adverse events (AE) and serious adverse events (SAE) were assessed2 years

Incidence and severity of adverse events (AE) and serious adverse events (SAE) as assessed according to NCI-CTCAE 5.0, as well as abnormalities in vital signs, electrocardiogram, and laboratory tests

Secondary Outcome Measures
NameTimeMethod
Kel2 years

Elimination rate constant

t1/22 years

Elimination half life time

CL/F2 years

Clearance

Vd/F2 years

Apparent volume of distribution

Rac2 years

Accumulation factor

PFS2 years

Progression-free survival

DOR2 years

Duration of Response

DCR2 years

Disease Control Rate

Cmax2 years

Maximum Plasma Concentration

Tmax2 years

Time to Cmax

AUC0-t2 years

Area under the concentration versus time curve from time 0 to the last measurable concentration

AUC0-inf2 years

AUC from time 0 to infinity

ORR2 years

DLT, MTD, RP2D, Number of participants and severity with treatment-related Adverse events as assessed by CTCAE V5.0

Trial Locations

Locations (4)

Sun Yat-Sen University Cancer Center

🇨🇳

Guangzhou, Guangdong, China

Harbin The First Hospitall

🇨🇳

Harbin, Heilongjiang, China

Jilin Cancer Hospital

🇨🇳

Changchun, Jilin, China

Beijing Cancer Hospital

🇨🇳

Beijing, 北京市, China

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