MedPath

AVT03 With Prolia in Healthy Male Subjects

Phase 1
Completed
Conditions
Healthy Male Subjects
Interventions
Biological: Prolia
Biological: AVT03
Registration Number
NCT05126784
Lead Sponsor
Alvotech Swiss AG
Brief Summary

This study has been designed as a randomized, double-blind, single-dose, parallel-group study in healthy adult male subjects 28 years to 55 years old. The study will assess the PK, PD, safety, tolerability and immunogenicity of AVT03 compared to Prolia when administered as a single SC dose.

Detailed Description

The study will consist of a 4 week screening period, a 252 day (36 weeks) treatment and assessment period, and an End of Study (EOS) visit on week 36 on Day 252. Subjects will undertake a screening visit between Day -28 and Day -1 to determine their eligibility for the study. On Day 1, eligible subjects will be randomized and will receive a single dose of AVT03 or Prolia as subcutaneous injection.

Recruitment & Eligibility

Status
COMPLETED
Sex
Male
Target Recruitment
209
Inclusion Criteria
  • Male subjects who are 28 to 55 years old, inclusive
  • Have a body weight of 50.0 to 90.0 kg (inclusive) and body mass index (BMI) of 17.0 to 32.0 kg/m2 (inclusive)at Screening and Day -1
  • Medical history without evidence of a clinically significant disorder, condition, or disease that, in the opinion of the Investigator, would pose a risk to subject safety
Exclusion Criteria
  • Any evidence of clinically relevant pathology, especially prior diagnosis of bone disease, or any uncontrolled condition that will affect bone metabolism (such as, but not limited to osteoporosis, osteogenesis imperfecta, hyperparathyroidism, hyperthyroidism, hypothyroidism, osteomalacia, rheumatoid arthritis, psoriatic arthritis, ankylosing spondylitis, current flare-up of osteoarthritis and/or gout, active malignancy, renal disease, Paget's disease of the bone, recent bone fracture [within 6 months], and malabsorption syndrome)
  • Have osteonecrosis of the jaw (ONJ) or risk factors for ONJ such as invasive dental procedures (eg, tooth extraction, dental implants, oral surgery) within 6 months prior to Day 1 or intend to undergo such procedures during the study period, poor oral hygiene, periodontal, and/or pre existing dental disease
  • Have bone fractures within 6 months prior to Day -1.
  • Have a history of immunodeficiency
  • Those with skin allergies, or are susceptible to autoinflammatory skin disorders, or prone to the development of allergic skin inflammation
  • Abnormal serum calcium: current hypocalcemia or hypercalcemia at Screening. Serum calcium levels must be within reference ranges.
  • Known vitamin D deficiency

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Prolia ArmProliaProlia(denosumab) is the proposed comparator for AVT03 (denosumab). Subjects in this arm will receive a single 60mg dose of Prolia (denosumab) as a subcutaneous injection.
AVT03 ArmAVT03AVT03 (denosumab) is the proposed biosimilar for Prolia (denosumab). Subjects in this arm will receive a single 60mg dose of AVT03 (denosumab) as a subcutaneous injection.
Primary Outcome Measures
NameTimeMethod
Area under the serum concentration-time curve (AUC0-last) from day 0 to day 252Day 1(week 1) to Day 252 (week 36)

Venous blood samples will be collected for measurement of Area under serum concentration-time curve (AUC 0-t) AVT03 and Prolia

Area under the serum concentration-time curve (AUC0-inf) from day 0 to day 252Time Frame: Day 1(week 1) to Day 252 (week 36)]

Venous blood samples will be collected for measurement of CTX-1 serum biomarker for AVT03 and Prolia.

Maximum serum concentration Cmax from day 0 to day 252Day 1(week 1) to Day 252 (week 36)

Venous blood samples will be collected for measurement of maximum serum concentration (Cmax) of AVT03 and Prolia.

Secondary Outcome Measures
NameTimeMethod
PK area under the concentration-time curve (AUC0-24) from Day 0 to Day 252Day 1(week 1) to Day 162 (week 24)]

Venous blood samples will be collected for measurement of serum concentration of AVT03 and Prolia

Immunogenicity presence and titers of ADAs and presence of nAbs against AVT03 and ProliaTime Frame: Day 1(week 1) to Day 252 (week 36)

Venous blood samples will be collected for measurement of antidrug-antibodies against of AVT03 and Prolia

Safety incidence, nature and severity of adverse eventsScreening to Day 252 (week 36)
PD_AUCE0 for CTX-1 (% inhibition)Day 1(week 1) to Day 252 (week 36)

Venous blood samples will be collected for measurement of serum concentration of AVT03 and Prolia

Trial Locations

Locations (4)

NZCR Auckland

🇳🇿

Auckland, New Zealand

NZCR Christchurch

🇳🇿

Christchurch, Christchuch, New Zealand

Nucleus Network

🇦🇺

Herston, Australia

Farmovs

🇿🇦

Bloemfontein, South Africa

© Copyright 2025. All Rights Reserved by MedPath