MedPath

Assess Safety and Efficacy of Vilaprisan in Subjects With Uterine Fibroids (ASTEROID 3)

Phase 3
Terminated
Conditions
Uterine Fibroids
Interventions
Registration Number
NCT03400943
Lead Sponsor
Bayer
Brief Summary

The primary objective of this study was to show superiority in the treatment of HMB of vilaprisan in subjects with uterine fibroids compared to placebo.

The secondary objectives of this study were to additionally evaluate the efficacy and safety of vilaprisan in subjects with uterine fibroids.

Detailed Description

Not available

Recruitment & Eligibility

Status
TERMINATED
Sex
Female
Target Recruitment
93
Inclusion Criteria
  • Women, 18 years or older in good General health
  • Diagnosis of uterine fibroid(s) documented by ultrasound at screening with at least 1 fibroid with largest Diameter ≥ 30 mm and < 120 mm
  • Heavy menstrual bleeding (HMB) in at least 2 bleeding periods during the Screening period each with blood loss volume of >80.00 mL documented by alkaline hematin (AH) method
  • An endometrial biopsy performed during the Screening period without significant histological disorder such as endometrial hyperplasia (including simple hyperplasia) or other significant endometrial pathology
  • Use of an acceptable non-hormonal method of contraception (ie, either male condom, cap, diaphragm or sponge, each in combination with spermicide) starting at Visit 1 until the end of the study
Read More
Exclusion Criteria
  • Pregnancy or lactation (less than 3 month since delivery, abortion, or lactation before start of Treatment)
  • Hypersensitivity to any ingredient of the study drug
  • Any condition requiring immediate blood transfusion
  • Laboratory values outside inclusion range before randomization and considered as clinically relevant.
  • Any diseases, conditions, or medications that can compromise the function of the body systems and could result in altered absorption, excessive accumulation, impaired metabolism, or altered excretion of the study drug
  • Any diseases or conditions that might interfere with the conduct of the study or the interpretation of the results
  • Abuse of alcohol, drugs, or medicines (eg, laxatives)
  • Use of other treatments that might interfere with the conduct of the study or the interpretation of the results
  • Undiagnosed abnormal genital bleeding
Read More

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
Vilaprisan (A2)Vilaprisan (BAY1002670)Vilaprisan (2 mg) in treatment period 1 for 12 weeks and in treatment period 2 for 12 weeks without a break.
Placebo+Vilaprisan (B1)Vilaprisan (BAY1002670)Placebo in treatment period 1 for 12 weeks, and vilaprisan (2 mg) in treatment period 2 for 12 weeks, separated by 1 bleeding episode.
Vilaprisan (A1)PlaceboVilaprisan (2 mg) in treatment period 1 for 12 weeks and in treatment period 2 for 12 weeks, separated by 1 bleeding episode.
Vilaprisan (A1)Vilaprisan (BAY1002670)Vilaprisan (2 mg) in treatment period 1 for 12 weeks and in treatment period 2 for 12 weeks, separated by 1 bleeding episode.
Vilaprisan+Placebo (B2)PlaceboVilaprisan (2 mg) in treatment period 1 for 12 weeks and placebo in treatment period 2 for 12 weeks, separated by 1 bleeding episode.
Vilaprisan+Placebo (B2)Vilaprisan (BAY1002670)Vilaprisan (2 mg) in treatment period 1 for 12 weeks and placebo in treatment period 2 for 12 weeks, separated by 1 bleeding episode.
Placebo+Vilaprisan (B1)PlaceboPlacebo in treatment period 1 for 12 weeks, and vilaprisan (2 mg) in treatment period 2 for 12 weeks, separated by 1 bleeding episode.
Primary Outcome Measures
NameTimeMethod
Number of Participants With AmenorrheaThe last 28 days of treatment period 1

Amenorrhea was defined as menstrual blood loss (MBL) \<2 mL during the last 28 days of treatment measured by the alkaline hematin (AH) method.

Secondary Outcome Measures
NameTimeMethod
Number of Participants With Heavy Menstrual Bleeding (HMB) ResponseThe last 28 days of treatment period 1 and treatment period 2

HMB response was defined as MBL \<80 mL during the last 28 days of treatment and \>50% reduction from baseline based on AH-method.

Time to Onset of AmenorrheaIn treatment period 1 (12 weeks) and in treatment period 2 (12 weeks)

Onset of amenorrhea was defined by the first day for which the MBL for all subsequent 28-day periods up to the end of a treatment period was \< 2 mL (amenorrhea defined similar to primary endpoint).

Time to Onset of Controlled BleedingIn treatment period 1 (12 weeks) and in treatment period 2 (12 weeks)

Onset of controlled bleeding was defined by the first day for which the MBL for all subsequent 28-day periods up to the end of a treatment period was \<80.00 mL based on AH-method.

Number of Participants With Absence of Bleeding (Spotting Allowed)The last 28 days of treatment period 1 and treatment period 2

Absence of bleeding was defined as no scheduled or unscheduled bleeding (spotting allowed) during the last 28 days of a treatment period based on subjects' daily responses to the Uterine Fibroid Daily Bleeding Diary (UF-DBD).

Number of Participants With Endometrial Histology Findings by Endometrial Biopsy Main Results (Majority Read, Main Diagnosis)Up to 2 weeks after end of treatment

Number of participants with endometrial histology findings, e.g. benign endometrium, Malignant Neoplasm, Hyperplasia WHO 2014, no atypia or Hyperplasia WHO 2014, atypia and Endometrial Polyps.

Change From Baseline of Endometrial ThicknessTreatment phase (up to 2 weeks after end of treatment) and follow-up phase (starts on the day after the end of the treatment until the last study visit [up to approximately 2 years])

Ultrasound examinations were performed. Endometrial thickness was measured in the medio-sagittal section as double-layer in millimeters. Summary statistics for change from baseline in endometrial thickness was provided in below table.

Trial Locations

Locations (103)

South Florida Medical Research

🇺🇸

Aventura, Florida, United States

Chattanooga Medical Research, LLC

🇺🇸

Chattanooga, Tennessee, United States

Sweet Hope Research Specialty, Inc. - Hialeah

🇺🇸

Hialeah, Florida, United States

One Health Research Clinic

🇺🇸

Norcross, Georgia, United States

PharmaSite Research, Inc.

🇺🇸

Baltimore, Maryland, United States

Houston Center for Clinical Research, LLC

🇺🇸

Sugar Land, Texas, United States

Georgia Center For Women

🇺🇸

Atlanta, Georgia, United States

Atlanta Women's Research Institute, Inc. - Alpharetta

🇺🇸

Atlanta, Georgia, United States

Medisense, Inc.

🇺🇸

Atlanta, Georgia, United States

Dr. Victoria Garcia & Associates, LLC Doral Medical Research

🇺🇸

Doral, Florida, United States

Centex Studies, Inc.

🇺🇸

Houston, Texas, United States

The Center for Clinical Trials, Inc.

🇺🇸

Houston, Texas, United States

Beijing Tiantan Hospital, Captial Medical University

🇨🇳

Beijing, China

MHAT Dr. Bratan Shukerov AD

🇧🇬

Smolyan, Bulgaria

Umhlanga Medical Centre

🇿🇦

Durban, Kwazulu-Natal, South Africa

Ideal Clinical Research

🇺🇸

Aventura, Florida, United States

National Research Institute - Los Angeles

🇺🇸

Los Angeles, California, United States

California Center for Clinical Research

🇺🇸

Arcadia, California, United States

Core Healthcare Group

🇺🇸

Cerritos, California, United States

AVIVA Research

🇺🇸

Escondido, California, United States

Helix Biomedics, LLC

🇺🇸

Boynton Beach, Florida, United States

Altus Research

🇺🇸

Lake Worth, Florida, United States

Axcess Medical Research, LLC

🇺🇸

Loxahatchee Groves, Florida, United States

Ocean Blue Medical Research Center, Inc.

🇺🇸

Miami Springs, Florida, United States

Clinical Neurosciences Solutions, Inc. DBA CNS Healthcare

🇺🇸

Jacksonville, Florida, United States

ONCOVA Clinical Research, Inc.

🇺🇸

Saint Cloud, Florida, United States

Agile Clinical Research Trials, LLC

🇺🇸

Atlanta, Georgia, United States

Discovery Clinical Research

🇺🇸

Plantation, Florida, United States

Paramount Research Solutions-College Park

🇺🇸

College Park, Georgia, United States

GTC Research

🇺🇸

Shawnee Mission, Kansas, United States

Simmonds, Martin and Helmbrecht

🇺🇸

Gaithersburg, Maryland, United States

Advantia Health, LLC Obstetrics & Gynecology Assoc.

🇺🇸

Silver Spring, Maryland, United States

Carolinas Healthcare System

🇺🇸

Charlotte, North Carolina, United States

SUNY Downstate Medical Center

🇺🇸

Brooklyn, New York, United States

Unified Women's Clinical Research - Morehead City

🇺🇸

Morehead City, North Carolina, United States

Fellows Research Alliance, Inc.

🇺🇸

Bluffton, South Carolina, United States

Clinical Research of Philadelphia, LLC

🇺🇸

Philadelphia, Pennsylvania, United States

Wake Research, Inc.

🇺🇸

Raleigh, North Carolina, United States

Fusion Clinical Research of Spartanburg, LLC

🇺🇸

Spartanburg, South Carolina, United States

Eastern Carolina Women's Center

🇺🇸

New Bern, North Carolina, United States

Main Line Fertility Center

🇺🇸

Bryn Mawr, Pennsylvania, United States

Clinical Neurosciences Solutions, Inc DBA CNS Healthcare

🇺🇸

Memphis, Tennessee, United States

Paramount Research Solutions-Nashville

🇺🇸

Nashville, Tennessee, United States

Willowbend Health & Wellness Associates

🇺🇸

Frisco, Texas, United States

Biopharma Informatic, Inc.

🇺🇸

Houston, Texas, United States

Family Medicine Clinic

🇺🇸

Georgetown, Texas, United States

Multiprofile Hospital for Active Treatment-Dr. T. Venkova AD

🇧🇬

Gabrovo, Bulgaria

Millennium Clinical Trials, LLC

🇺🇸

Arlington, Virginia, United States

Hospital for Active Treatment - Prof.Paraskev Stoyanov AD

🇧🇬

Lovech, Bulgaria

900th Hospital of Joint Logistics Support Force

🇨🇳

Fuzhou, Fujian, China

Guangzhou Women and Children's Medical Center

🇨🇳

Guangzhou, Guangdong, China

MHAT for Women's Health - Nadezhda OOD

🇧🇬

Sofia, Bulgaria

The Third Affiliated Hospital, Sun Yat-Sen University

🇨🇳

Guangzhou, Guangdong, China

Boai Hospital of Zhongshan

🇨🇳

Zhongshan, Guangdong, China

Nanjing Maternity and Child Health Care Hospital

🇨🇳

Nanjing, Jiangsu, China

Wuhan Tongji Reproductive Medicine Hospital

🇨🇳

Wuhan, Hubei, China

NJ Drum Tower Hospital, the Affil Hos of NJ Univ Med School

🇨🇳

Nanjing, Jiangsu, China

Zhongda Hospital Southeast University

🇨🇳

Nanjing, Jiangsu, China

Hainan General Hospital

🇨🇳

Haikou, Hainan, China

The First Hospital of Jilin University

🇨🇳

Changchun, Jilin, China

1st Affiliated hospital of Soochow University

🇨🇳

Suzhou, Jiangsu, China

Jiangxi Maternal and Child Health Hospital

🇨🇳

Nanchang, Jiangxi, China

Lady Davis Carmel Medical Center

🇮🇱

Haifa, Israel

The Second Affiliated Hospital of Nanchang University

🇨🇳

Nanchang, Jiangxi, China

The First Affiliated Hospital of Dalian Medical University

🇨🇳

Dalian, Liaoning, China

Shengjing Hospital of China Medical University

🇨🇳

Shenyang, Liaoning, China

General Hospital of Ningxia Medical University

🇨🇳

Yinchuan, Ningxia, China

Second Affiliated Hospital of Xi'an Jiaotong University

🇨🇳

Xi'an, Shaanxi, China

Women's Hospital School of Medicine Zhejiang University

🇨🇳

Hangzhou, Zhejiang, China

The First Affiliated Hospital of Xinjiang Medical University

🇨🇳

Urumqi, Xinjiang, China

Sarawak General Hospital

🇲🇾

Sarawak, Malaysia

The First Affiliated Hospital of Xi'an Jiaotong University

🇨🇳

Xi'an, Shaanxi, China

The Second Affiliated Hospital of Shanxi Medical University

🇨🇳

Taiyuan, Shanxi, China

Sir Run Run Shaw Hospital, Zhejiang University School of Med

🇨🇳

Hangzhou, Zhejiang, China

The Second Affliated Hospital of Wenzhou Medicial University

🇨🇳

Wenzhou, Zhejiang, China

Beijing Friendship Hospital, Capital Medical University

🇨🇳

Beijing, China

Beijing Hospital of Traditional Chinese Medicine

🇨🇳

Beijing, China

Peking University First Hospital

🇨🇳

Beijing, China

Tianjin Medical University General Hospital

🇨🇳

Tianjin, China

Shanghai East Hospital Affiated to Tongji University

🇨🇳

Shanghai, China

Gynekologie MEDA s.r.o.

🇨🇿

Brno, Czechia

Gynekologie Studentsky dum s.r.o.

🇨🇿

Praha 6, Czechia

Hillel Yaffe Medical Center

🇮🇱

Hadera, Israel

Soukroma gynekologicka ambulance

🇨🇿

Fulnek, Czechia

MUDr. Ivana Salamonova s.r.o.

🇨🇿

Vysoke Myto, Czechia

Hospital Wanita dan Kanak-Kanak Sabah

🇲🇾

Sabah, Malaysia

Clalit Health Services through HaEmek Medical Center

🇮🇱

Afula, Israel

Meir Medical Center

🇮🇱

Kfar Saba, Israel

University Hospital Kebangsaan Malaysia

🇲🇾

Kuala Lumpur, Malaysia

KK Women's and Children's Hospital

🇸🇬

Singapore, Singapore

P3 Research Ltd Hawkes Bay

🇳🇿

Hawkes Bay, New Zealand

P3 Research

🇳🇿

Tauranga, New Zealand

Dr L Reynders Practice

🇿🇦

Lyttelton Manor, Gauteng, South Africa

Wilgeheuwel Hospital

🇿🇦

Roodepoort, Gauteng, South Africa

Ethekwini Hospital & Heart Centre

🇿🇦

Durban, Kwazulu-Natal, South Africa

Omni Fertility and Laser Institute

🇺🇸

Shreveport, Louisiana, United States

Harbor - UCLA Medical Center

🇺🇸

Torrance, California, United States

Fellows Research Alliance - Savannah

🇺🇸

Savannah, Georgia, United States

Texas Health Care, PLLC

🇺🇸

Fort Worth, Texas, United States

University of Alabama at Birmingham

🇺🇸

Birmingham, Alabama, United States

Accelerated Enrollment Solutions a business of PPD

🇺🇸

Orlando, Florida, United States

Medical University of South Carolina

🇺🇸

Charleston, South Carolina, United States

Synexus Research, LLC

🇺🇸

Richmond, Virginia, United States

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