MedPath

Bioequivalence Study With Clinical Endpoint for Diclofenac Sodium Topical Gel 1%

Phase 3
Completed
Conditions
Osteoarthritis, Knee
Interventions
Registration Number
NCT02913521
Lead Sponsor
Akorn, Inc.
Brief Summary

A Double-Blind, Randomized, Placebo-Controlled, Parallel Group, Three-Arm, Multi-Site Study to Evaluate the Therapeutic Equivalence of Diclofenac Sodium Topical Gel 1% (Hi-Tech Pharmacal Co., Inc.) With Voltaren® Gel (Diclofenac Sodium Topical Gel) 1% (Novartis) in Patients With Osteoarthritis of the Knee

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
934
Inclusion Criteria
  1. Ambulatory male and non-pregnant females 35 years and older diagnosed with osteoarthritis according to the American College of Rheumatology Criteria (ACR) in one knee. Target knee is the one with higher level of pain.

    ACR Criteria includes: Knee Pain and at least 3 of the following: age ≥ 50, stiffness lasting < 30 mins, bony tenderness, crepitus, bony enlargement, and no palpable warmth.

  2. Symptom onset of > 6 Months prior to Screening for the target knee.

  3. If female and of child-bearing potential, prepare to abstain from sexual intercourse or use a reliable method of contraception during the study (e.g., IUD, oral, transdermal, injected, implanted hormonal contraceptives or condom + spermicide).

  4. Periarticular knee pain due to osteoarthritis (not bursitis, tendonitis etc.) that required the use of oral or topical treatments (e.g., NSAIDs or acetaminophen).

  5. Radiograph of the target knee within the previous year with a Grade 1, 2 or 3 disease based upon the Kellgren-Lawrence disease severity scale.

  6. After a minimum of 7-day wash out of all pain medication has Baseline pain on movement score of ≥ 50mm on a 0-100-mm Visual Analogue Scale for the target knee.

  7. After a minimum of 7-day wash out of all pain medication has Baseline WOMAC Pain sub scale of ≥ 9 on a 5 question, 5 point (0 to 4) Likert scale for the target knee.

  8. Willing and able to use only acetaminophen as rescue medication.

  9. Willing and able to comply with the study requirements.

Exclusion Criteria
  1. Females who are pregnant, breast feeding, or planning a pregnancy.
  2. Radiograph of the target knee within the previous year with a Grade 4 score on the Kellgren-Lawrence disease severity scale.
  3. History of osteoarthritis in the contralateral knee requiring medication (OTC or prescription) within 12 months of screening.
  4. After a minimum of 7-day wash out of all pain medication has Baseline pain on movement score of ≥ 20mm on a 0-100-mm Visual Analogue Scale for the contralateral knee immediately prior to randomization.
  5. Known history of secondary osteoarthritis (e.g. congenital, traumatic, gouty arthritis) of the knee or rheumatoid arthritis.
  6. Known history of other chronic inflammatory diseases, (e.g., colitis) or fibromyalgia during last 5 years. Patients whose disease was diagnosed at least 5 (five) years prior to screening visit and have had no known disease activity (i.e., no disease related complaints nor disease treatment prescribed) since then may enter into the study.
  7. History of asthma, hypertension, myocardial infarction, thrombotic events, stroke, congestive heart failure, impaired renal function or liver disease. Patients who have had high blood pressure measured at least 2 (two) years prior to screening visit and have had no disease activity (i.e., no record of hypertension or anti-hypertensive treatment prescribed) for at least 2 (two) years prior to screening visit may enter into the study.
  8. History of coronary artery bypass graft within 6 months of screening.
  9. Concomitant acetylsalicylic acid therapy other than a stable low dose used for cardiac prophylaxis (max. 162 mg daily) taken for at least 3 months prior to enrollment and maintained throughout the duration of the study.
  10. Use of warfarin or other anticoagulant therapy within 30 days of screening.
  11. Use of ACE inhibitors, cyclosporine, diuretics, lithium or methotrexate, within 30 days of screening or during the study.
  12. Known history of gastrointestinal bleeding or peptic ulcer disease.
  13. Abnormal screening clinical laboratory evaluations which the Investigator deems clinically significant.
  14. Known allergy to aspirin or NSAIDs.
  15. Skin lesions or wounds in the affected area.
  16. Significant (requiring surgery) injury or major knee surgery to either knee within six months prior to screening.
  17. Transaminase levels that are more than two times the upper limit of the normal range at screening.
  18. Any other acute or chronic illness that in the opinion of the investigator could compromise the integrity of study data or place the Patient at risk by participating in the study.
  19. Concomitant use of corticosteroids (any formulation) or use within 30 days of study randomization.
  20. Receipt of any drug as part of a research study within 30 days prior to screening.
  21. Previous randomization into this study.
  22. Known allergy (hypersensitivity) to acetaminophen.

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
PlaceboPlaceboApply 4 g of gel to the knee four times a day
Diclofenac Sodium Gel 1%Diclofenac Sodium Gel 1%Apply 4 g of gel to the knee four times a day
Voltaren GelVoltaren GelApply 4 g of gel to the knee four times a day
Primary Outcome Measures
NameTimeMethod
Mean Change From Baseline to Week 8 in WOMAC Pain Scale, Bioequivalence of Test to Reference.8 weeks

WOMAC = Western Ontario and McMaster Universities Arthritis Index. The higher number is more pain. Change from baseline to Week 8 as indicated in the title. Scale is 5 questions with a scale of 0-4, higher number is more pain. Therefore, if you have 5 questions and the max score for each is 4, the maximum number on the scale is 20 (5 questions x 4 units on the scale = 20).

Secondary Outcome Measures
NameTimeMethod
Clinically Significant Changes From Baseline in Physical Examination Results8 weeks
An Evaluation to Determine Superiority of Test and Reference Against Placebo in the Mean Change From Baseline to Week 8 in the Total WOMAC Pain Score.8 weeks

WOMAC = Western Ontario and McMaster Universities Arthritis Index. The higher number is more pain. Change from baseline to Week 8 as indicated in the title. Scale is 5 questions with a scale of 0-4, higher number is more pain. Therefore, if you have 5 questions and the max score for each is 4, the maximum number on the scale is 20 (5 questions x 4 units on the scale = 20).

Incidences of Abnormal Vital Signs8 weeks
Incidences of Treatment Emergent Adverse Events8 weeks

Trial Locations

Locations (50)

Medicum Ltd.

🇪🇪

Tallinn, Estonia

Dr.Monika Vask Ltd.

🇪🇪

Tartu, Estonia

Ltd. Elli Kahar

🇪🇪

Tartu, Estonia

CERMED

🇵🇱

Bialystok, Poland

SIS Klinika ALma

🇱🇻

Riga, Latvia

OU Perearstikeskus Remedium

🇪🇪

Tallinn, Estonia

"REUMA TIKA- Centrnrn Reurnatologii" NZOZ

🇵🇱

Warsaw, Poland

Spital Judetean De Urgenta Bacau

🇷🇴

Bacau, Romania

Communal Institution "Cherkasy Regional Hospital of Cherkasy Regional Council"

🇺🇦

Cherkasy, Ukraine

MI Pyogrov Vinnystya Regional Clinical Hospital

🇺🇦

Vinnytsya, Ukraine

Clinical Best Solutions

🇵🇱

Lublin, Poland

Linnamoisa Perearstikeskus

🇪🇪

Tallinn, Estonia

D.Saulites-Kandevicas private practice

🇱🇻

Liepaja, Latvia

Health Center 4

🇱🇻

Riga, Latvia

JSC Mano Seimos Gydytojas

🇱🇹

Klaipeda, Lithuania

Medical Chamber in Warsaw Nr 5718455

🇵🇱

Warsaw, Mazovia, Poland

Duo Medical

🇷🇴

Bucharest, Romania

RK Medcenter SRL

🇷🇴

Iasi, Romania

Communal Institution of Kyiv Regional Council "Kyiv Regional Clinical Hospital"

🇺🇦

Kyiv, Ukraine

InMedica

🇱🇹

Kaunas, Lithuania

ClinicMed Badurski i Wspolnicy Spolka Jawna

🇵🇱

Bialystok, Poland

ZOZ w Olawie

🇵🇱

Olawa, Poland

Spiratul Judetean de Urgenta Bacau

🇷🇴

Bacau, Romania

Emergency County Hospital SF Gheorghe

🇷🇴

Bucharest, Romania

State Institution "Professor M.I. Sytenko Institute of Spine and Joint Patholo of the National Academ of Medical Sciences of Ukraine

🇺🇦

Kharkiv, Ukraine

Communal Institution of.Lviv Regional Council "Yu. Lypa Lviv Regional Hospital of Disabled War Veterans and Former Political Prisoners"

🇺🇦

Lviv, Ukraine

East Tallinn Central Hospital

🇪🇪

Tallinn, Estonia

Linna Health Cerntre

🇪🇪

Tallinn, Estonia

Association of Health Centres, Medical Centre "OLVI"

🇱🇻

Daugavpils, Latvia

JSC Vita Longa

🇱🇹

Kaunas, Lithuania

Private medical practice Jacek Niski

🇵🇱

Czestochowa, Poland

Dr Ion Stoia Rheumatology Center

🇷🇴

Bucharest, Romania

S.C. Clinica Somesan

🇷🇴

Marasti, Romania

State Institution D.F.Chebotariov Institute ofGerontolo!.!v ofNAMS of Ukraine - Dept of Age related changes to Muscoskeletal system

🇺🇦

Kyiv, Ukraine

Pirita Family Doctors Centre

🇪🇪

Tallinn, Estonia

Vee Family Doctor's Center OY

🇪🇪

Paide, Estonia

OU Mai Perearstid

🇪🇪

Parnu, Estonia

West Tallinn Central Hospital

🇪🇪

Tallinn, Estonia

Orthopaedic and Clinical Research Center

🇪🇪

Tartu, Estonia

JSC Saules seimos medicinos centras

🇱🇹

Kaunas, Lithuania

Private Doctor Family Clinic JSc Ausveja

🇱🇹

Vilnius, Lithuania

St. Luke's hospital in Bielsko-Biala

🇵🇱

Bielsko-Biala, Poland

Niepubliczny Zaklad Opieki Zdrowotnej ORTMED sp. z o.o.

🇵🇱

Lodz, Poland

MEDICOME Sp. z o.o.

🇵🇱

Oswiecim, Poland

Centrum Medyczne Luxmed, Przezmierowo

🇵🇱

Poznan, Poland

State Institution D.F.Chebotariov Institute of Gerontology of NAMS of Ukraine

🇺🇦

Kyiv, Ukraine

S.C. lanuli Med Consult Str Intr Lt. Dumitru Lemnea

🇷🇴

Bucharest, Romania

Ploiești Municipal Hospital

🇷🇴

Ploiesti, Romania

State Institution "Ukrainian State Scientific and Research Institute of Medical and Social Problems of Disability of the Ministry of Health of Ukraine

🇺🇦

Dnipropetrovsk, Ukraine

Odesa Regional Clinical Hospital

🇺🇦

Odesa, Ukraine

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