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A Trial to Find Out How Safe REGN5668 is and How Well it Works When Given With Either Cemiplimab or REGN4018

Phase 1
Recruiting
Conditions
Ovarian Cancer
Fallopian Tube Cancer
Primary Peritoneal Cancer
Endometrial Cancer
Interventions
Registration Number
NCT04590326
Lead Sponsor
Regeneron Pharmaceuticals
Brief Summary

This study is researching an investigational drug called REGN5668. Participants will receive additional investigational drugs in combination with REGN5668. These additional drugs include cemiplimab or REGN4018 (with or without sarilumab).

The main purposes of this study are to:

* Learn about the safety and profile of any side effects from the study drugs and to determine the highest, safe dose that can be given to participants with ovarian cancer or cancer of the uterus

* Look for signs that the study drugs can treat ovarian cancer or cancer of the uterus

This study has 2 parts. The purpose of Part 1 (Escalation) to find the highest, safe dose of the study drug(s). The purpose of Part 2 (Expansion) is to use the doses chosen in Part 1. Participants with cancer of the uterus will only participate in Part 2.

The study is looking at several other research questions, including:

* Side effects that may be experienced by participants taking REGN5668 alone and/or in combination with cemiplimab or REGN4018

* How REGN5668 works in the body either alone and/or in combination with cemiplimab or REGN4018

* How much of the study drugs (REGN5668, cemiplimab, REGN4018) are in the blood

* To see if REGN5668 in combination with cemiplimab or REGN4018 works to treat cancer

* To find out how safe, tolerable, and effective in mitigating Cytokine Release Syndrome (CRS) sarilumab pretreatment is when given before REGN4018

Detailed Description

Not available

Recruitment & Eligibility

Status
RECRUITING
Sex
Female
Target Recruitment
612
Inclusion Criteria
  1. Ovarian Cancer Cohorts Only: Has histologically or cytologically confirmed diagnosis of advanced epithelial ovarian cancer (except carcinosarcoma), primary peritoneal, or fallopian tube cancer that has received at least 1 line of platinum-based systemic therapy as defined in the protocol
  2. Expansion cohorts only: Has at least 1 lesion that is measurable by RECIST 1.1 as described in the protocol.
  3. Has a serum CA-125 level ≥2x ULN (in screening, not applicable to endometrial cohorts)
  4. Has adequate organ and bone marrow function as defined in the protocol
  5. Has an Eastern Cooperative Oncology Group (ECOG) performance status of 0 or 1.
  6. Has a life expectancy of at least 3 months
  7. Endometrial Cancer Cohorts Only: histologically confirmed endometrial cancer that has progressed or recurrent after prior anti-PD-1 therapy and platinum-based chemotherapy as described in the protocol

Key

Exclusion Criteria
  1. Prior anti-cancer immunotherapy as defined in the protocol
  2. Recent treatment with anti-Programmed Cell Death (PD-1)/PDL-1 therapy
  3. Has had another malignancy within the last 5 years that is progressing, requires active treatment, or has a high likelihood of recurrence as defined in the protocol
  4. Prior treatment with a MUC16-targeted therapy
  5. Expansion cohorts only: More than 4 prior lines of cytotoxic chemotherapy (including antibody drug conjugates)
  6. Has any condition that requires ongoing/continuous corticosteroid therapy as defined in the protocol within 1 week prior to the first dose of study drug
  7. Has ongoing or recent (within 5 years) evidence of significant autoimmune disease that required treatment with systemic immunosuppressive treatments as defined in the protocol
  8. Has untreated or active primary brain tumor, CNS metastases, leptomeningeal disease, or spinal cord compression as defined in the protocol
  9. Has history of clinically significant cardiovascular disease as defined in the protocol
  10. Has known allergy or hypersensitivity to cemiplimab and/or components of study drug(s).

Note: Other protocol-defined Inclusion/Exclusion criteria apply

Study & Design

Study Type
INTERVENTIONAL
Study Design
SEQUENTIAL
Arm && Interventions
GroupInterventionDescription
Module 2REGN5668REGN5668 and REGN4018
Module 2REGN4018REGN5668 and REGN4018
Module 2SarilumabREGN5668 and REGN4018
Module 1REGN5668REGN5668 and cemiplimab
Module 1CemiplimabREGN5668 and cemiplimab
Primary Outcome Measures
NameTimeMethod
Incidence of laboratory abnormalities (Grade 3 or higher per National Cancer Institute Common Terminology Criteria for Adverse Events [NCI-CTCAE] version 5.0 [v5.0])Through study completion, up to 5 years

Primary: Dose escalation phase Secondary: Dose expansion phase

Concentrations of REGN5668 in serum when dosed alone and in combination with cemiplimab or REGN4018Through study completion, up to 5 years

Primary: Dose escalation phase Secondary: Dose expansion phase

Incidence of dose limiting toxicities (DLT)42 days

Dose escalation phase, Module 1

Incidence of DLTs21 days post combination administration

Dose escalation phase, Module 2

Incidence of treatment-emergent adverse events (TEAEs)Through study completion, up to 5 years

Primary: Dose escalation phase Secondary: Dose expansion phase

Incidence of serious adverse events (SAEs)Through study completion, up to 5 years

Primary: Dose escalation phase Secondary: Dose expansion phase

Incidence of deathsThrough study completion, up to 5 years

Primary: Dose escalation phase Secondary: Dose expansion phase

ORR defined by Response Evaluation Criteria in Solid Tumors (RECIST) 1.1 (Eisenhauer, 2009) in combination with cemiplimab or REGN4018 (separately by cohort and combination)Through study completion, up to 5 years

Primary: Dose expansion phase Secondary: Dose escalation phase

Secondary Outcome Measures
NameTimeMethod
BOR based on RECIST 1.1 and iRECISTThrough study completion, up to 5 years

Dose escalation and expansion phases

DOR based on RECIST 1.1 and iRECISTThrough study completion, up to 5 years

Dose escalation and expansion phases

Concentration of REGN4018 in serum over timeThrough study completion, up to 5 years

Dose expansion phase

Concentration of cemiplimab in serum over timeThrough study completion, up to 5 years

Dose expansion phase

ORR based on Immune-based therapy RECIST (iRECIST)Through study completion, up to 5 years

Dose escalation and expansion phases

DCR based on RECIST 1.1 and iRECISTThrough study completion, up to 5 years

Dose escalation and expansion phases

PFS based on RECIST 1.1 and iRECISTThrough study completion, up to 5 years

Dose escalation and expansion phases

CA-125 change from baseline after treatment with REGN5668 in combinations with cemiplimab or REGN4018 (separately by cohort and combination)Through study completion, up to 5 years

Dose escalation and expansion phases

Presence or absence of anti-drug antibodies against REGN5668Through study completion, up to 5 years

Dose escalation and expansion phases

Presence or absence of anti-drug antibodies against REGN4018Through study completion, up to 5 years

Dose escalation and expansion phases

Presence or absence of anti-drug antibodies against cemiplimabThrough study completion, up to 5 years

Dose escalation and expansion phases

Trial Locations

Locations (23)

Hopital Lyon Sud

🇫🇷

Pierre-Benite, Lyon, France

Institut Gustave Roussy

🇫🇷

Villejuif, France

The City of Hope Orange County Lennar Foundation Cancer Center

🇺🇸

Irvine, California, United States

Robert H. Lurie Comprehensive Cancer Center of Northwestern University

🇺🇸

Chicago, Illinois, United States

City of Hope Comprehensive Cancer Center

🇺🇸

Duarte, California, United States

Memorial Sloan Kettering Cancer Center

🇺🇸

New York, New York, United States

The Ohio State University Wexner Medical Center

🇺🇸

Columbus, Ohio, United States

Perelman School of Medicine at the University of Pennsylvania

🇺🇸

Philadelphia, Pennsylvania, United States

H. Lee Moffitt Cancer Center

🇺🇸

Tampa, Florida, United States

University of Chicago Medical Center

🇺🇸

Chicago, Illinois, United States

Massachusetts General Hospital

🇺🇸

Boston, Massachusetts, United States

Centre Francois Baclesse (CFB)

🇫🇷

Caen, Normandy, France

Institut Bergonie

🇫🇷

Bordeaux, France

Hospital Clinico Universitario Santiago de Compostela

🇪🇸

Santiago de Compostela, A Coruna, Spain

Dana Farber Cancer Institute Brookline Avenue

🇺🇸

Boston, Massachusetts, United States

Karmanos Cancer Institute

🇺🇸

Detroit, Michigan, United States

Seattle Cancer Care Alliance at South Lake Union - G3630

🇺🇸

Seattle, Washington, United States

Universitair Ziekenhuis Leuven

🇧🇪

Leuven, Vlaams Brabant, Belgium

Centre Georges Francois Leclerc

🇫🇷

Dijon, Bourgogne, France

Institut Catala dOncologia Girona

🇪🇸

Girona, Spain

Ciudad Universitaria

🇪🇸

Madrid, Spain

Hospital Universitario Fundacion Jimenez

🇪🇸

Madrid, Spain

Hospital Universitario 12 de Octubre Universidad Complutense de Madrid UCM

🇪🇸

Madrid, Spain

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