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Effects of Alogliptin on Pancreatic Beta Cell Function

Not Applicable
Conditions
Diabetes Mellitus, Type 2
Interventions
Registration Number
NCT01303055
Lead Sponsor
Aichi Gakuin University
Brief Summary

It is reported that pancreatic beta cell function is already declined at pre-diabetic stage, impaired glucose tolerance (IGT). It has not been clarified whether inhibitors of the dipeptidyl peptidase IV enzyme (DPP-IV inhibitors) improve beta cell function on human pancreas, however, if efficacy is ensured, they may become the first medicine to be chosen for treatments of type 2 diabetes and IGT.

In this trial, a DPP-IV inhibitor, Alogliptin, or Metformin are given to diabetic patients whose HbA1c level is below 7.9%. Oral glucose tolerance test (OGTT) will be conducted before, a year after, and two years after the beginning of the trial and beta cell function will be evaluated.

Detailed Description

Patients will be randomly allocated to two groups. They will receive either Alogliptin or Metformin.

Alogliptin: The investigators will start with 25 mg QD and the dose will be maintained.

Metformin: The investigators will start with 250 mg QD and the dose will be slowly increased to 750 mg TID. The dose increase is possible up to its maximum, 2250 mg, so that HbA1c is maintained below 6.9%. However, increase in dose with elder patients requires careful consideration.

Participants taking part in this study will receive dietary and exercise coaching. Participation in this study is expected to last up to 2 years.

Patients will terminate from the trial when their HbA1c exceeds 8.4% for more than three months.

The investigators will evaluate beta cell function by conducting 75 g OGTT before, a year after, and two years after the beginning of the trial. Alogliptin or Metformin will be stopped three days before the OGTT. The investigators will make sure that urine ketone is negative before an oral glucose load.

Recruitment & Eligibility

Status
UNKNOWN
Sex
All
Target Recruitment
80
Inclusion Criteria
  • Patients who are diagnosed as type 2 diabetes with HbA1c level below 7.9% and haven't received oral hypoglycemic agents or insulin treatments for the past three months.
Exclusion Criteria
  • Patients whose 75 g OGTT 30-minutes insulin secretion exceeds 100 μU/ml
  • Patients with renal failure with serum creatinine level ≧ 1.2
  • Patients with hepatocirrhosis
  • Patients with proliferative diabetic retinopathy or worse
  • Patients with acute infectious disease
  • Patients who are treated with steroids
  • Patients with cancer
  • Pregnant patients
  • Patients with malfunction of the heart (NYHA classification III-IV)
  • Patients who are decided to be inappropriate subjects by study physicians

Study & Design

Study Type
INTERVENTIONAL
Study Design
PARALLEL
Arm && Interventions
GroupInterventionDescription
AlogliptinAlogliptinAlogliptin 25 mg
MetforminMetformin 750 mgMetformin 750 mg
Primary Outcome Measures
NameTimeMethod
beta cell function evaluated from 75 g OGTT2 years

75 g OGTT: glucose level, blood insulin level, c-peptide immunoreactivity (pre-test, 30 mins, 60 mins, 120 mins), fasting blood proinsulin

Oral glucose tolerance test ( OGTT ) will be conducted before, a year after, and two years after the beginning of the trial.

Secondary Outcome Measures
NameTimeMethod
1,5-AG level2 years

Secondary end points include HbA1c level.

Trial Locations

Locations (4)

Diabetes Center, Yokkaichi Social Insurance Hospital

🇯🇵

Yokkaichi, Mie, Japan

Dept. of Intern. Med., School of Dentistry, Aichi Gakuin University

🇯🇵

Nagoya, Aichi, Japan

Diabetes Clinic, Okazaki East Hospital

🇯🇵

Okazaki, Aichi, Japan

Tosaki Clinic for Diabetes and Endocrinology

🇯🇵

Nagoya, Aichi, Japan

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