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Single Dose Study in Subjects With Severe Hemophilia A Comparing Pharmacokinetic Parameters for BAY81-8973 and Advate

Phase 1
Completed
Conditions
Hemophilia A
Interventions
Drug: BAY81-8973
Registration Number
NCT02483208
Lead Sponsor
Bayer
Brief Summary

The purpose of this study is to compare the pharmacokinetics of BAY81-8973 and Advate after intravenous administration.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
Male
Target Recruitment
18
Inclusion Criteria
  • Males, age 18 to 65 years

    • Subjects with Severe hemophilia A with a documented plasma FVIII level of <1%
    • ≥ 150 exposure days with FVIII concentrate(s) as supported by medical records
Exclusion Criteria
  • Evidence of current or past inhibitor antibody

    • History of any congenital or acquired coagulation disorders other than hemophilia A
    • Platelet count <75,000/mm3
    • Abnormal renal function (serum creatinine >2 times the upper limit of the normal [ULN] range)
    • Active liver disease verified by medical history or persistently elevated alanine aminotransferase (ALT) or aspartate aminotransferase (AST) >5 times the ULN or severe liver disease as evidenced by, but not limited to any of the following: International Normalized Ratio (INR) >1.4, hypoalbuminemia, portal vein hypertension including presence of otherwise unexplained splenomegaly and history of esophageal varices.

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
BAY81-8973BAY81-8973BAY81-8973 infusion to analyze pharmacokinetics
AdvateAdvateAdvate infusion to analyze pharmacokinetics.
Primary Outcome Measures
NameTimeMethod
AUC(0-tlast)Pre-Dose, 0.25, 0.5, 1, 3, 6, 8, 24, 30, 48 hours after treatment

Area under the blood concentration vs time curve from zero to the last data point \> lower limit of quantification

Secondary Outcome Measures
NameTimeMethod
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