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A rotation study of different albuminuria lowering drug classes to study individual drug response in diabetic and non diabetic CKD

Phase 1
Conditions
Chronic Kidney Disease
MedDRA version: 21.1Level: LLTClassification code 10009119Term: Chronic renal failureSystem Organ Class: 100000004857
Therapeutic area: Diseases [C] - Nutritional and Metabolic Diseases [C18]
Registration Number
EUCTR2017-004641-25-IT
Lead Sponsor
IVERSITY MEDICAL CENTER GRONINGE
Brief Summary

Not available

Detailed Description

Not available

Recruitment & Eligibility

Status
Authorised-recruitment may be ongoing or finished
Sex
All
Target Recruitment
46
Inclusion Criteria

eGFR > 30 and < 90 ml/min/1.73m2
Albuminuria = 100 mg/24 hour and = 3500 mg/24 hour
Serum potassium = 5.0 mmol/L
Treatment with ACEi or ARB
Age = 18 years
Written informed consent

Are the trial subjects under 18? no
Number of subjects for this age range:
F.1.2 Adults (18-64 years) yes
F.1.2.1 Number of subjects for this age range 20
F.1.3 Elderly (>=65 years) yes
F.1.3.1 Number of subjects for this age range 26

Exclusion Criteria

Diagnosis of type 1 diabetes mellitus

Urinary protein excretion > 3500 mg/24 hour

Autosomal dominant polycystic kidney disease or autosomal recessive polycystic kidney disease, lupus nephritis, or ANCA-associated vasculitis

Indication for immunosuppressants as per the treating physician’s judgment.

Receiving cytotoxic therapy, immunosuppressive therapy, or other immunotherapy for primary or secondary renal disease within 6 months prior to enrolment.

Active malignancy aside from treated squamous cell or basal cell carcinoma of the skin.

Diabetes type 2 patients with recent (last 6 months) of hyperosmolar hyperglicemic state who are prone to development redistributive hyperkalemia (movement of potassium out of the cells)

Pregnant women and women of child-bearing potential who are not using reliable contraception

Cardiovascular disease: myocardial infarction, angina pectoris, percutanous transluminal coronary angioplasty, coronary artery bypass grafting, stroke, heart failure (NYHA I-IV) < 6 months before inclusion

Uncontrolled blood pressure (office blood pressure > 160 / 100 mmHg)

History of autonomic dysfunction (e.g. history of fainting or clinically significant orthostatic hypotension)

History of amputations

eGFR change > 30% in the last six months before study randomization

Current therapy with renin inhibitor or MRA

Concomitant treatment with ACEi and ARB

Intolerance or contraindications to drugs inhibiting the Renin-Angiotensin-Aldosterone System (RAAS). Cyclosporine A, tacrolimus, trimethoprim due to increased risk of hyperkalemia in combination with eplerenone. Ketoconazole, itraconazole, ritonavir, nelfinavir, clarithromycin, telithromycin and nefazadone, lithium, amiodarone, diltiazem, verapamil due to increase in toxicity when combined with eplerenone. Rifampicin, carbamazepine, phenytoin, phenobarbital due the risk of decreased eplerenone efficacy.

Participation in any clinical investigation within 3 months prior to initial dosing or longer if required by local regulations, and for any other limitation of participation based on local regulations.

Donation or loss of 400 ml or more of blood within 8 weeks prior to initial dosing

History of drug or alcohol abuse within the 12 months prior to dosing, or evidence of such abuse as indicated by the laboratory assays conducted during the screening.

Any medication, surgical or medical condition which might significantly alter the absorption, distribution, metabolism, or excretion of medications

Study & Design

Study Type
Interventional clinical trial of medicinal product
Study Design
Not specified
Primary Outcome Measures
NameTimeMethod
Main Objective: To determine the correlation between individual albuminuria lowering responses of the MRA eplerenone, SGLT2 inhibitor dapagliflozin and their combination in patients with chronic kidney disease ;Secondary Objective: To determine the correlation between office/home blood pressure-lowering responses of eplerenone, dapaglifozin and their combination.<br>To determine which patients characteristics predict the albuminuria and blood pressure response to eplerenone, dapagliflozin and their combination;Primary end point(s): Correlation between individual albuminuria response between eplerenone and dapagliflozin.;Timepoint(s) of evaluation of this end point: 24 weeks which corresponds to the sum of the three treatment periods plus the three wash-out periods
Secondary Outcome Measures
NameTimeMethod
Secondary end point(s): the degree of correlation in either office or home blood pressure-lowering responses with eplerenone and dapagliflozin<br>; Correlation between selected biomarkers of interest at baseline such as NT-proBNP and change in albuminuria from baseline during interventions;Timepoint(s) of evaluation of this end point: 24 weeks which corresponds to the sum of the three treatment periods plus the three wash-out periods; 24 weeks which corresponds to the sum of the three treatment periods plus the three wash-out periods
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