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Safety, Tolerability and Pharmacodynamics Evaluation of CBT-009 Eye Drop

Phase 1
Completed
Conditions
Myopia, Progressive
Interventions
Registration Number
NCT05372991
Lead Sponsor
Cloudbreak Therapeutics, LLC
Brief Summary

This is a Two-Stage Phase 1/2 study to evaluate the safety, tolerability and pharmacodynamics of CBT-009 eye drop in healthy volunteers.

CBT-009 has the active ingredient of atropine, which at low doses, has shown to be effective in slowing down myopic deterioration. Current atropine products are prone to degradation once the container is open to the air. ADS Pharmaceutical has developed a novel atropine formulation.

Detailed Description

Type of Study:

Stage 1: Single center, open-labeled, vehicle-controlled, single ascending dose.

Stage 2: Parallel, double-masked, randomized, vehicle-controlled with dosing once-daily in one eye.

Study Population:

Male or female healthy volunteers aged 18-36 years.

Number of Subjects and Sites:

Stage 1: Enrollment is planned for approximately 32 healthy volunteers with 8 subjects per cohort for a total of 4 cohorts.

Stage 2: Enrollment is planned for approximately 50 healthy volunteers with 25 subjects per cohort for a total of 2 cohorts.

Duration of Study Participation:

Stage 1: One day. Stage 2: 28 days of treatment with no follow-up observations.

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
84
Inclusion Criteria

Healthy volunteer without any active ocular diseases

  • 18-36 years of age
  • Able to provide written informed consent and comply with study assessments for the full duration of the study
Exclusion Criteria

Uncontrolled systemic disease

  • Active ocular disease
  • Any ocular surgical procedure within the last 3 months
  • Current enrollment in an investigational drug or device study or participation in such as study within 30 days prior to entry into this study
  • Any condition or situation which, in the investigator's opinion, may put the volunteer at significant risk, may confound the study results, or may interfere significantly with the volunteer's participation in the study. Allergic or sensitive to Atropine study medication or formulation excipient
  • Smoking during the study
  • Female patients who are pregnant, nursing, or planning a pregnancy during the study
  • Current or anticipated use of topical ophthalmic medications are prohibited during the study. Volunteers must have discontinued use of ophthalmic medications for at least 2 weeks prior to Day 1 visit

Study & Design

Study Type
INTERVENTIONAL
Study Design
SEQUENTIAL
Arm && Interventions
GroupInterventionDescription
vehicleVehicleCBT-009 vehicle formulation is a proprietary sterile ophthalmic solution that does not contain CBT-009 drug substance.
CBT-009, Low DoseCBT-009CBT-009 low dose formulation is a proprietary sterile ophthalmic solution that contain low dose of CBT-009 drug substance.
CBT-009, Mid DoseCBT-009CBT-009 mid dose formulation is a proprietary sterile ophthalmic solution that contain mid dose of CBT-009 drug substance.
CBT-009, High DoseCBT-009CBT-009 high dose formulation is a proprietary sterile ophthalmic solution that contain high dose of CBT-009 drug substance.
0.025% atropine sulphateAtropine SulfateThe comparator formulation of 0.025% atropine sulfate monohydrate in normal saline will be prepared by diluting commercial 1% atropine sulphate solution with physiologic saline.
Primary Outcome Measures
NameTimeMethod
Safety on near visual acuity28 days

Near visual acuity will be assessed using best-corrected distance spectacle correction with a reduced logMAR reading chart placed at 40 cm under well-lit conditions at Day 28.

Safety on accommodation28 days

The accommodation will be measured using a near point rule with best-corrected distance spectacle correction at Day 28.

Safety on mesopic and photopic pupil28 days

Mesopic pupil size and photopic pupil size will be measured with a pupillometer at Day 28.

Secondary Outcome Measures
NameTimeMethod

Trial Locations

Locations (1)

USC

🇦🇺

Brisbane, Australia

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