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To Investigate the Efficacy and Safety of Individualized Doses of BioChaperone Insulin Lispro in Comparison to Humalog® U-100 in Patients With Type 1 Diabetes Mellitus

Phase 1
Completed
Conditions
Type 1 Diabetes Mellitus
Interventions
Drug: BioChaperone insulin lispro
Registration Number
NCT02528396
Lead Sponsor
Adocia
Brief Summary

This is a double-blind, randomised, controlled, two period crossover phase Ib trial using an individualized standard meal with a fixed nutrient ratio in subjects with type 1 diabetes mellitus to investigate postprandial blood glucose control with BioChaperone insulin lispro compared to Humalog®. The assessments will be conducted before and after a period of multiple daily dose administrations for 14 days. The meal tolerance test will be performed on day 1-3 and on day 14 of each period. Furthermore the study aims at investigating Post-prandial glucose (PPG) profiles with BioChaperone insulin lispro and Humalog® when injected at various injection meal intervals (-15min, 0 minutes, +15 minutes).

Each subject will be randomised to a sequence of two treatments, either BioChaperone insulin lispro-Humalog® or Humalog®-Biochaperone insulin lispro, and three different sequences of injection-meal intervals. A blinded to patient continuous monitoring of glucose (CGM) will be performed during the 14 day treatment periods.

Detailed Description

Not available

Recruitment & Eligibility

Status
COMPLETED
Sex
All
Target Recruitment
36
Inclusion Criteria
  • Type 1 diabetes mellitus (as diagnosed clinically) ≥ 12 months
  • Treated with multiple daily insulin injections (no pump users) ≥ 12 months
  • Current total daily insulin treatment <1.2 (I)U/kg/day
  • Body mass index (BMI) 18.5-28.0 kg/m² (both inclusive)
  • HbA1c (N-(1-deoxy)-fructosyl-haemoglobin) ≤ 9.0% by local laboratory analysis
  • Fasting C-peptide ≤ 0.30 nmol/L
Exclusion Criteria
  • Known or suspected hypersensitivity to trial products or related products
  • Type 2 diabetes mellitus
  • Patients using continuous subcutaneous insulin infusion (CSII)
  • Previous participation in this trial. Participation is defined as randomised
  • The receipt of any investigational product within 3 months prior to this trial
  • Clinically significant abnormal haematology, biochemistry, lipids, or urinalysis screening tests, as judged by the Investigator considering the underlying disease
  • Presence of clinically significant acute gastrointestinal symptoms (e.g. nausea, vomiting, heartburn or diarrhoea), as judged by the Investigator
  • Known slowing of gastric emptying and or gastrointestinal surgery that in the opinion of the investigator might change gastrointestinal motility and food absorption
  • Unusual meal habits and special diet requirements or unwillingness to eat the food provided in the trial

Study & Design

Study Type
INTERVENTIONAL
Study Design
CROSSOVER
Arm && Interventions
GroupInterventionDescription
Humalog®Humalog®-
BioChaperone insulin lisproBioChaperone insulin lispro-
Primary Outcome Measures
NameTimeMethod
AUCΔBG0-2h (timepoint 0 = administration of the meal)2 hours

Incremental area under the blood glucose (BG) concentration-time curve from 0-2 hours after a meal on day 1-3 \[comparison between treatments Biochaperone insulin lispro vs. lispro (Humalog®)\]

AUClispro 0-30min (timepoint 0 = time of dosing)30 minutes

Area under the serum insulin lispro concentration-time curve from 0-30 minutes after bolus dose on one of days 1, 2 or 3 (comparison between treatments BioChaperone insulin lispro vs. lispro (Humalog®))

Secondary Outcome Measures
NameTimeMethod
AUClispro_0-6h6 Hours

Area under the serum insulin lispro concentration-time curve from 0-6 hours after bolus dose

Cmax_lisproup to 6 Hours

Maximum serum insulin lispro concentration

Tmax_lisproup to 6 Hours

Time to maximum observed serum insulin lispro concentration

AUCBG_0-6h6 Hours

Area under the curve under the blood glucose (BG) concentration time curve from 0-6 hours

ΔBGmax6 Hours

Maximum blood glucose (BG) excursion after a standard meal (0-6 hours)

Adverse eventsUp to 3 months

Number of Adverse events

Local tolerability injection site reactions14 days

Injection site reactions over 14 days of exposure

Trial Locations

Locations (1)

Profil GmbH

🇩🇪

Neuss, Germany

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