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Study of ABT-199 (GDC-0199) in Combination With Azacitidine or Decitabine (Chemo Combo) in Subjects With Acute Myelogenous Leukemia (AML)

Phase 1
Terminated
Conditions
Acute Myelogenous Leukemia
Myelogenous Leukemia
Treatment Naive AML
Interventions
Registration Number
NCT02203773
Lead Sponsor
AbbVie
Brief Summary

This is a Phase 1b, open-label, non-randomized, multicenter study to evaluate the safety and pharmacokinetics of orally administered venetoclax (ABT-199) combined with decitabine or azacitidine and the preliminary efficacy of these combinations. In addition, there is a drug-drug interaction (DDI) sub-study only at a single site, to assess the pharmacokinetics and safety of venetoclax (ABT-199) in combination with posaconazole.

Detailed Description

Not available

Recruitment & Eligibility

Status
TERMINATED
Sex
All
Target Recruitment
212
Inclusion Criteria
  • Subjects must have confirmation of Acute Myeloid Leukemia (AML) by WHO criteria and be ineligible for treatment with a standard cytarabine and anthracycline induction regimen due to co-morbidity or other factors.
  • Subject must have received no prior treatment for AML with the exception of hydroxyurea
  • Subjects must have Eastern Cooperative Oncology Group (ECOG) Performance Status of 0 to 2 for subjects greater than or equal to 75 years of age, or 0 to 3 for subjects greater than or equal to 60 to 74 years of age
  • Subject must have adequate kidney and liver function as described in the protocol
Exclusion Criteria
  • Subject has received treatment with the following hypomethylating agent and/or chemo therapeutic agent for for an antecedent hematologic disorder (AHD) (Subjects may have been treated with other agents for AHD i.e., Myelodysplastic syndrome [MDS])

  • Subject has history of Myeloproliferative Neoplasm (MPN).

  • Subject has favorable risk cytogenetics as categorized by the National Comprehensive Cancer Network Guidelines Version 2, 2014 for AML.

  • Subject has t(8;21), inv(16), t(16;16) or t(15;17) karyotype abnormalities.

  • Subject has acute promyelocytic leukemia.

  • Subject has known active central nervous system involvement with AML.

  • Subject has received a strong and/or moderate CYP3A inducer within 7 days prior to the initiation of study treatment.

  • Subject has a history of other malignancies prior to study entry, with the exception of:

    • Adequately treated in situ carcinoma of the cervix uteri or carcinoma in situ of breast;
    • Basal cell carcinoma of the skin or localized squamous cell carcinoma of the skin;
    • Previous malignancy confined and surgically resected (or treated with other modalities) with curative intent.
  • Subject has a white blood cell count > 25 × 10^9/L. Note: Hydroxyurea is permitted to meet this criterion.

Study & Design

Study Type
INTERVENTIONAL
Study Design
SINGLE_GROUP
Arm && Interventions
GroupInterventionDescription
ABT-199 + AzacitidineAzacitidineTreatment Naive Acute Myelogenous Leukemia
ABT-199 + AzacitidineABT-199Treatment Naive Acute Myelogenous Leukemia
ABT-199 + DecitabineABT-199Treatment Naive Acute Myelogenous Leukemia
ABT-199 + DecitabineDecitabineTreatment Naive Acute Myelogenous Leukemia
ABT-199+Decitabine+PosaconazolePosaconazoleTreatment Naive Acute Myelogenous Leukemia
ABT-199+Decitabine+PosaconazoleABT-199Treatment Naive Acute Myelogenous Leukemia
ABT-199+Decitabine+PosaconazoleDecitabineTreatment Naive Acute Myelogenous Leukemia
Primary Outcome Measures
NameTimeMethod
Number of Participants Experiencing Adverse Events (AEs)Measured up to 1 year after the last subject last dose

An adverse event (AE) is defined as any untoward medical occurrence in a patient or clinical investigation participant administered a pharmaceutical product which does not necessarily have a causal relationship with this treatment. The investigator assesses the relationship of each event to the use of study drug.

Maximum observed plasma concentration (Cmax)For approximately 5 days following a single dose of ABT-199.

Maximum observed concentration, occurring at Tmax.

Time to Cmax (peak time, Tmax),For approximately 5 days following a single dose of ABT-199.

The time at which maximum plasma concentration (Cmax) is observed.

The area under the plasma concentration-time curve (AUC) from 0 to 24 hours (AUC0-24)For approximately 5 days following a single dose of ABT-199.

The area under the plasma concentration-time curve (AUC) over a 24-hour dose interval.

Half-Life (t1/2)For approximately 5 days following a single dose of ABT-199.

The time required for the concentration of the drug to reach half of its original value.

Clearance (CL)For approximately 5 days following a single dose of ABT-199.

Clearance is defined as the rate at which drug is cleared from the blood.

Complete Remission RateMeasured up to 1 year after the last subject last dose

Complete Remission Rate will be determined by the number of subjects who achieve a Complete Remission.

Complete Remission with incomplete blood count recovery rateMeasured up to 1 year after the last subject last dose

Complete Remission with incomplete blood count recovery rate will be determined by the number of subjects who achieve a Complete Remission with incomplete blood count recovery.

Overall Response RateMeasured up to 1 year after the last subject last dose

Overall response rate will be defined as the proportion of subjects who achieve a complete remission (CR), complete remission incomplete (CRi), or partial remission (PR) per the International Working Group criteria for AML.

Overall SurvivalMeasured up to 1 year after the last subject last dose

Overall survival will be defined as the number of days from the date of first dose to the date of death.

Secondary Outcome Measures
NameTimeMethod
Event Free SurvivalMeasured up to 1 year after the last subject last dose

Event-free survival (EFS) will be defined as the number of days from the date of first dose to the date of earliest evidence of relapse, subsequent treatment other than stem cell transplant while in composite complete response (CR + CRi), or death.

Duration of ResponseMeasured up to 1 year after the last subject last dose

Duration of response will be defined as the number of days from the date of first response per the IWG criteria for AML to the earliest recurrence or progressive disease (PD).

Trial Locations

Locations (23)

Johns Hopkins University /ID# 129699

🇺🇸

Baltimore, Maryland, United States

Northwestern University Feinberg School of Medicine /ID# 128741

🇺🇸

Chicago, Illinois, United States

Dana-Farber Cancer Institute /ID# 127857

🇺🇸

Boston, Massachusetts, United States

University of Texas MD Anderson Cancer Center /ID# 141581

🇺🇸

Houston, Texas, United States

University of Washington /ID# 129717

🇺🇸

Seattle, Washington, United States

University of California, Davis Comprehensive Cancer Center /ID# 129719

🇺🇸

Sacramento, California, United States

Duke Cancer Center /ID# 129720

🇺🇸

Durham, North Carolina, United States

AP-HP - Hopital Saint-Louis /ID# 130349

🇫🇷

Paris, France

Peter MacCallum Cancer Ctr /ID# 130352

🇦🇺

Melbourne, Victoria, Australia

Columbia University Medical Center /ID# 130289

🇺🇸

New York, New York, United States

City of Hope /ID# 129718

🇺🇸

Duarte, California, United States

The University of Chicago Medical Center /ID# 128742

🇺🇸

Chicago, Illinois, United States

Hopital Haut-Lévêque /ID# 134388

🇫🇷

Pessac CEDEX, Gironde, France

Alfred Health /ID# 130353

🇦🇺

Melbourne, Victoria, Australia

Emory Midtown Infectious Disease Clinic /ID# 129715

🇺🇸

Atlanta, Georgia, United States

Univ of Colorado Cancer Center /ID# 127859

🇺🇸

Aurora, Colorado, United States

Universitaetsklinikum Leipzig /ID# 130346

🇩🇪

Leipzig, Sachsen, Germany

Universitaetsklinikum Ulm /ID# 130341

🇩🇪

Ulm, Baden-Wuerttemberg, Germany

Universitaetsklinikum Carl Gustav Carus an der TU Dresden /ID# 130342

🇩🇪

Dresden, Germany

University of Texas MD Anderson Cancer Center /ID# 127860

🇺🇸

Houston, Texas, United States

St George Hospital /ID# 130356

🇦🇺

Kogarah, New South Wales, Australia

Duplicate_Klinikum Rechts der Isar /ID# 130347

🇩🇪

Munich, Germany

Duplicate_Hopital Universitaire Purpan /ID# 134389

🇫🇷

Toulouse, Haute-Garonne, France

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